DC22456 |
GLPG-0492 R enantiomer |
The R enantiomer of GLPG-0492, a non-steroidal selective androgen receptor modulator (SARM) for treatment for Duchenne muscular dystrophy (DMD). |
|
DC24174 |
Refametinib R enantiomer |
The R enantiomer of Refametinib, a potent, non–ATP-competitive, highly selective, allosteric inhibitor of MEK1/2 with IC50 of 19/47 nM respectively.. |
|
DC24133 |
Bay 65-1942 R form |
The R form of Bay 65-1942. which is a potent, selective, ATP-competitive inhibitor of IKKβ kinase with Ki of 2 nM.. |
|
DC23865 |
LOXO-195 R racemate |
The R racemate of LOXO-195, a potent, selective, next-generation Trk tyrosine kinase inhibitor with IC50 of 0.6 nM and <2.5 nM for WT TrkA and WT TrKC, respectively.. |
|
DC23174 |
GNE-140 racemate
Featured
|
GNE-140 racemate consists of equal parts (R)-GNE-140 and (S)-GNE-140 enantiomers, functioning as a potent inhibitor of lactate dehydrogenase A (LDHA). |
|
DC22558 |
Pemafibrate racemate |
The racemate of Pemafibrate, which is a highly potent, specific PPARα agonist with EC50 of 1 nM.. |
|
DC23999 |
(R)-Oxiracetam |
the R-enantiomer of the nootropic drug oxiracetam (ISF 2522), which is a nootropic drug of the racetam family and stimulant.. |
|
DC23866 |
LOXO-195 RS-isomer |
The RS-isomer of LOXO-195, a potent, selective, next-generation Trk tyrosine kinase inhibitor with IC50 of 0.6 nM and <2.5 nM for WT TrkA and WT TrKC, respectively.. |
|
DC22480 |
5-FAM |
The single isomer, 5-FAM, contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid. Fluorescein is the most common fluorescent derivatization reagent for labeling biomolecules. In addition |
|
DC20816 |
BMS 830216 |
The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM. |
|
DC10469 |
ST-271
Featured
|
The tyrosine kinase inhibitor ST271 inhibited phospholipase D (PLD) activity in human neutrophils stimulated by fMet-Leu-Phe, platelet-activating factor and leukotriene B4. |
|
DC11272 |
AG-126
Featured
|
The tyrphostin AG-126 selectively inhibits the phosphorylation of ERK1 (p44) and ERK2 (p42) at 25-50 μM. |
|
DC22593 |
KPT-8602 Z-isomer |
The Z-isomer of Eltanexor (KPT-8602), which is a second-generation SINE with markedly reduced brain penetration compared to selinexor.. |
|
DC22541 |
R-80123 |
The Z-isomer of R 79595, a highly selective PDE inhibitor, 10-fold more potent than R 79595.. |
|
DC20173 |
Acefylline;Theophyllineacetic acid; Theophylline-7-acetic acid |
Theophylline-7-acetic acid (Acefylline), acting as an adenosine receptor antagonist, is a stimulant drug of the xanthine chemical class. |
|
DC8759 |
Thiamet G
Featured
|
Thiamet G is a potent and selective inhibitor of O-GlcNAcase that demonstrates a Ki value of 21 nM. |
|
DCAPI1077 |
Thiamphenicol (Thiophenicol) |
Thiamphenicol (Thiophenicol) |
|
DC8673 |
Thifluzamide |
Thifluzamide is a powerful and effective fungicide. When used safely and correctly it can be effective on rice and other crops because of improved water dispersal techniques. Thifluzamide is highly active against Basidiomycete fungi, in particular Rhizoct |
|
DC12363 |
Thionin acetate (Thionine acetate) |
Thionin (acetate) is a metachromic cationic histology dye used in biological staining widely. |
|
DC12573 |
THIQ40 |
THIQ 40 (THIQ40) is a potent, orally available ERα antagonist and selective estrogen receptor degrader (SERD) with IC50 of 17 nM (ERα binding) and 30 nM (ERα transcription), IC50 of 0.9 nM (ERα degradation). |
|
DC7678 |
R-P7C3-Ome
Featured
|
This compound is a methoxy derivative of parent compound P7C3. |
|
DC8126 |
CALCIUM IONOPHORE II
Featured
|
This is a very good carrier of Ca+2-ions, induces a selectivity in membranes for Ca+2over Mg+2 by a factor of about 10. |
|
DC21746 |
Thr-Asp-F-amidine
Featured
|
Thr-Asp-F-amidine (TDFA) is a highly potent, selective PAD4 (protein arginine deiminase 4) inhibitor with IC50 of 2.3 uM, displays ≥15-fold selectivity for PAD4 versus PAD1 and ≥50-fold versus PADs 2 and 3. |
|
DC23429 |
THRX-198321 |
THRX-198321 is a bifunctional mAChR antagonist and β2-adrenoceptor agonist (MABA) with pKi of 9.69/10.05 for M1/M2 respectively, pEC50 of 9.25 for β2AR. |
|
DC24135 |
THS-044 |
THS-044 is a low micromolar HIF2α PAS-B binding compound (Kd=2 uM). |
|
DC11384 |
Thymogen(Oglufanide)
Featured
|
Thymogen(Oglufanide) is a new immunomodulating drug. |
|
DC23984 |
Thyroxine sulfate |
Thyroxine sulfate (T4) is a major Thyroid hormone metabolite secreted by follicular cells of the Thyroid gland, T4 is involved in controlling the rate of metabolic processes in the body and influencing physical development, a prohormone and a reservoir fo |
|
DC8656 |
Tiamulin fumarate |
Tiamulin is a diterpenic veterinary drug widely used in swine for the control of infectious diseases, including swine dysentery and enzootic pneumonia. |
|
DC8868 |
TIC10
Featured
|
TIC10 inactivates Akt and ERK to induce TRAIL through Foxo3a, possesses superior drug properties: delivery across the blood-brain barrier, superior stability and improved pharmacokinetics |
|
DCAPI1144 |
Ticarcillin sodium |
Ticarcillin is a semisynthetic antibiotic with a broad spectrum of bactericidal activity against many gram-positive and gram-negative aerobic and anaerobic bacteria. |
|