Thr-Asp-F-amidine

  Cat. No.:  DC21746   Featured
Chemical Structure
1345019-64-8
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Field of application
Thr-Asp-F-amidine (TDFA) is a highly potent, selective PAD4 (protein arginine deiminase 4) inhibitor with IC50 of 2.3 uM, displays ≥15-fold selectivity for PAD4 versus PAD1 and ≥50-fold versus PADs 2 and 3.
Cas No.: 1345019-64-8
Chemical Name: TDFA
Synonyms: TDFA
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Thr-Asp-F-amidine (TDFA) is a highly potent, selective PAD4 (protein arginine deiminase 4) inhibitor with IC50 of 2.3 uM, displays ≥15-fold selectivity for PAD4 versus PAD1 and ≥50-fold versus PADs 2 and 3; active in cells and can be used to inhibit PAD4 activity in cellulo.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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