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Cat. No.	Product Name	Field of Application
DC33513	D-alpha-Methylbenzyl isothiocyanate	D-alpha-Methylbenzyl isothiocyanate is an antioxidant that induces phase II enzyme activity. It is also used as a chiral agent.
DC33514	L-alpha-Methylbenzyl isothiocyanate	L-alpha-Methylbenzyl isothiocyanate is an antioxidant that induces phase II enzyme activity. It is also used as a chiral agent.
DC33515	S-Methyl-L-cysteine	S-Methylcysteine is an antioxidant found in Brassicaceae family plants. It decreases oxidative stress and inhibits oil drop formation in white pre-adipose tissue.
DC33516	Methyiin	NSC-226572, also known as Alanine, 3-(methylsulfinyl)-, L-, pyrolyzate, S-methyl-L-cysteine-S-oxide; S-Methylcysteine sulfoxide, is a synthetic analog of alliin found in cruciferous vegetables including cabbage, turnip, cauliflower, and kale. NSC-226572 is converted through alliinase activity into a volatile thiosulfinate.
DC33517	7-Methyl-6-mercaptopurine	7-Methyl-6-mercaptopurine is a 6-mercaptopurine derivative and inhibitor of PRPP amidotransferase used to treat autoimmune diseases, leukemia,s and lymphomas. It inhibits IMP metabolism, preventing the synthesis of purines, DNA and RNA.
DC33518	Kavatin	Methysticin is found in Piper methysticum (kava plant). It inhibits activation of NF-χB in lung adenocarcinoma tissue, activates Nrf2 in neurons and astroglia, decreases peak amplitude of voltage-gated Na+ channels in hippocampal neurons, and suppresses growth of Fusarium, Trichoderma, and Colletotrichum.
DC33519	Andergin	Miconazole nitrate is an 14-α demethylase inhibitor and potential glucocorticoid receptor antagonist that inhibits ergosterol synthesis and fungal cell wall formation. It is used to treat fungal infections and is especially active against Candida. It also decreases expression of HIF-1α and VEGF in breast cancer and glioma cells.
DC33520	BW-B 1090U	Mivacurium chloride is a non-depolarizing NMJ blocker and nAChR antagonist used as an anesthetic. It inhibits skeletal muscle contractility and prevents atrial fibrillation.
DC33521	Coban 45	Monensin sodium is an ionophore and inhibitor of autophagy commercially used in livestock feed. It inhibits autophagy, interfering with the fusion of the autophagosome and the lysosome.
DC33522	Moniliformin	Moniliformin is a mycotoxin and potential dehydrogenase inhibitor found in Fusarium. It decreases collage synthesis, suppresses endocytosis, and may damage myocardial tissue.
DC33523	Myclobutanil	Myclobutanil is a 14-α demethylase inhibitor that inhibits ergosterol synthesis and fungal cell wall formation. It also weakly inhibits testosterone production.
DC33524	Nadifloxacine	Nadifloxacin is a bacterial DNA gyrase inhibitor used to treat acne vulgaris. It inhibits Proponibacterium-stimulated cytokine expression and decreases production of oxidative radicals by neutrophils.
DC33525	Albalon Liquifilm	Naphazoline HCl is an α1-Adrenergic receptor agonist used to treat congestion and ocular pathologies. It also induces autophagy and necrotic cell death in erythroleukemia cells and inhibits erythroid differentiation.
DC33526	Benil	Naphazoline nitrate is α1-Adrenergic receptor agonist used to treat congestion and ocular pathologies. It also induces autophagy and necrotic cell death in erythroleukemia cells and inhibits erythroid differentiation.
DC33527	beta-Naphthoflavone	beta-Naphthoflavone is a AhR agonist and antioxidant. It inhibits cigarette smoked-induced DNA damage and tumor development and induces cell cycle arrest in breast cancer cells.
DC33528	D-(+)-Neopterin	D-(+)-Neopterin is an endogenous pteridine metabolite of GTP used as an endogenous biomarker of cellular immune response and oxidative stress.
DC33529	Histomon	Nifursol is a livestock feed additive and antiobiotic used to prevent the growth of histomonas.
DC33530	HLI373	HLI373 is a water-soluble inhibitor of Hdm2. HLI373 is effective in inducing apoptosis of several tumor cells lines that are sensitive to DNA-damaging agents. HLI373 could serve as a potential lead for developing cancer therapeutics based on inhibition of the ubiquitin ligase activity of Hdm2.
DC33531	J1038	J1038 is a novel Inhibitor of Histone Deacetylase 8 (HDAC8).
DC33532	GQ-16	GQ-16 is an effective inhibitor of Cdk5-mediated phosphorylation of PPARγ. GQ-16 improves glucose tolerance and insulin sensitivity in mouse models of obesity and diabetes without inducing weight gain or edema.
DC33533	CYP3cide	PF-04981517, also known as CYP3cide, is a potent and selective time dependent inactivator of Cytochrome P450 3A4 (CYP3A4). CYP3cide is a very useful tool for understanding the relative roles of CYP3A4 versus CYP3A5 and the impact of CYP3A5 genetic polymorphism on a compound's pharmacokinetics.
DC33534	LPA5-IN-4	LPA5-IN-4 is the first non-lipid, small-molecule inhibitor for LPA5/GPR92, specifically inhibiting LPA-mediated platelet activation in vitro.
DC33535	NMS-E973 Featured	NMS-E973 is a novel, selective and potent inhibitor of heat shock protein 90 (Hsp90). NMS-E973 displays significant efficacy in a human ovarian A2780 xenograft tumor model, with a mechanism of action confirmed in vivo by typical modulation of known Hsp90 client proteins, and with a favorable pharmacokinetic and safety profile. The efficacy profile of NMS-E973 suggests a potential for development in different clinical settings, including tumors that have become resistant to molecular targeted agents, particularly in cases of tumors which reside beyond the blood-brain barrier (BBB).
DC33536	azF	4-Azido-L-phenylalanine, also known as azF, is a genetically-encoded molecular probe. azF is used to study GPCRs in their native cellular environment or under detergent solubilized conditions.
DC33537	Chlorfenson Featured	Chlorfenson is used to treat onychomycosis (nail fungus) as the primary indication.
DC33538	Monocrotophos	Monocrotophos is an organophosphate insecticide that blocks monoamine oxidase and acetylcholinesterase.
DC33539	BTT-3033	BTT-3033 is a α2β1 integrin inhibitor. BTT-3033 blocks platelet attachment under flow (90 dynes/cm(2)). The action of BTT-3033, unlike that of BTT-3034, was dependent on Tyr-285.
DC33540	CU-CPT22	CU-CPT22 is the first probe for the complex between toll-like receptors TLR1 and TLR2. CU-CPT22 binds at the interface of TLR1 and TLR2 (IC50 = 0.58 μM).
DC33541	Calpain Inhibitor VI	SJA6017, also known as Calpain Inhibitor VI, is a calpain inhibitor (calpain-1; IC50 = 7.5 nM) and m-calpain (calpain-2; IC50 = 78 nM). It also inhibits cathepsins B and L (IC50s = 15 and 1.6 nM, respectively). Treatment with SJA6017 reduces apoptotic cell death, preserves spinal cord tissue and improves functional outcome. Treating calpain-induced apoptosis with this agent may be a feasible therapeutic strategy for patients with spinal cord injury.
DC33542	D-AP7	D-AP7 is a specific NMDA antagonist and is the more active form of DL-AP7. D-AP7 enhanced motility, exhibited anxiogenic-like effect and impaired consolidation in passive avoidance.

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