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Cat. No.	Product Name	Field of Application
DC23061	L-45	PCAF BRD inhibitor L-45 is a potent, selective, and cell-active PCAF bromodomain inhibitor with Ki of 47 nM in HTRF assays, >4,500-fold selectivity over BRD4.
DC23651	PCARBTP	PCARBTP is a derivative, potent, specific Kv1.3 channel inhibitor, reduces cell viability and efficiently kills B16F10 cancer cells at 1 uM.
DC11169	PCC0104005	PCC0104005 (PCC-0104005) is a novel modulator of serotonin, dopamine, and noradrenaline receptors, including partial agonism at dopamine D2, D3, D4, serotonin 5-HT1A, and 5-HT2A receptors and antagonism at 5-HT2B, 5-HT6, and 5-HT7 receptors.
DC10757	PCI-29732 Featured	PCI 29732 is a selective and irreversible Btk inhibitor with IC50 of 8.2 nM in a FRET based biochemical enzymology assay.
DC8844	PCI-27483 Featured	PCI-27483 is a selective small molecule inhibitor of activated coagulation factor VII (FVIIa), which is in preclinical development as a novel anti-cancer agent.
DC1106	PCI-32765 (Ibrutinib) Featured	PCI-32765 (Ibrutinib) is a potent and highly selective Btk inhibitor with IC50 of 0.5 nM.
DC12080	PCI-33380	PCI-33380 is an irreversible Bruton's Tyrosine Kinase (BTK) inhibitor (fluorescent probe).
DC1109	PCI-34051 Featured	PCI-34051 is a potent and specific HDAC8 inhibitor with IC50 of 10 nM.
DC10531	PCO371 Featured	PCO371 is a novel, orally active small molecule that acts as a full agonist of PTHR1.
DC23759	PCSK9 modulator 10	PCSK9 modulator 10 is a highly potent, orally active PCSK9 modulator that inhibits PCSK9 production in HepG2 cells with IC50 of 0.036 nM.
DC23758	PCSK9-IN-7l	PCSK9-IN-7l is a potent, small molecule PCSK9 mRNA translation inhibitor with IC50 of 1.37 uM, shows limited bone marrow toxicity (IC50=27.1 uM)..
DC7224	PD 123319 Featured	PD 123319 is a potent, selective AT2 angiotensin II receptor antagonist with IC50 of 34 nM.
DC8283	PD 150606 Featured	PD 150606 is a selective, cell-permeable non-peptide calpain inhibitor (Ki values for ν and m-calpains are 0.21 and 0.37 μM respectively).
DC8747	PD-151746 Featured	PD 151746 is a selective, cell-permeable calpain inhibitor with Ki of 0.26 μM for μ-Calpain, about 20-fold selectivity over m-calpain.
DC8078	PD 153035(AG-1517) Featured	PD 153035(AG-1517) is an ultra-potent inhibitor of epidermal growth factor receptor tyrosine kinase (EGFRK), with an IC50 of 25 pM.
DC5100	PD 98059 Featured	PD 98059 is a selective inhibitor of MEK and blocker of MAPK
DC9744	PD0166285 Featured	PD0166285 is a potent Wee1 and Chk1 inhibitor with activity at nanomolar concentrations.PD0166285 is a novel G2 checkpoint abrogator.
DC1056	PD0325901 (Mirdametinib) Featured	PD0325901 (PD325901) is selective and non ATP-competitive MEK inhibitor with IC50 of 0.33 nM.
DC9280	BMS-1 (PD1/PDL1 inhibitor 1) Featured	PD-1/PD-L1 inhibitor 1 is a PD-1/PD-L1 interaction inhibitor,IC50 values: 0.006-0.10 μM,a useful immunomodulator compound.
DC8381	PD-1/PD-L1 inhibitor 2(BMS-202) Featured	PD-1/PD-L1 inhibitor 2 is reported to prevent the interaction of PD-L1 with PD-1 with an IC50 value of 18 nM,a useful compound immunomodulator compound.
DC5021	PD153035 HCl (SU-5271, AG1517) Featured	PD153035 is a potent and specific inhibitor of EGFR with Ki and IC50 of 5.2 pM and 29 pM; little effect noted against PGDFR, FGFR, CSF-1, InsR and Src.
DC7842	PD158780 Featured	PD158780 is a very potent inhibitor of EGFR with IC50 of 0.08 nM; pan-specific antagonist of ErbB receptor.
DC21466	PD166285 Featured	PD166285 (PD 0166285) is a broad-spectrum receptor tyrosine kinase (RTK) inhibitor that inhibits PDGFR-β, EGFR, and FGFR1 and c-Src with IC50 of 7-85 nM.
DC10068	PD166866 Featured	PD-166866 is a selective inhibitor of the FGF-1 receptor tyrosine kinase (FGFR1) with IC50 = 55 nM, and no effect on c-Src, PDGFR-b, EGFR or insulin receptor tyrosine kinases or MEK, PKC, and CDK4.
DC12316	PD-168077 maleate Featured	PD-168077 maleate is a selective dopamine D4 receptor agonist, with a Ki of 9 nM.
DC9258	PD168393 Featured	PD168393 is potent, cell-permeable, irreversible and selective inhibitor of EGF receptor (EGFR) tyrosine kinase and ErbB2.
DC5095	PD169316 Featured	PD169316 is a potent and selective p38 MAP kinase inhibitor
DC2054	PD-173074 Featured	PD173074 is a potent FGFR1 inhibitor with IC50 of ~25 nM and also inhibits VEGFR2 with IC50 of 100-200 nM.
DC7571	PD173955 Featured	PD-173955 is a src tyrosine kinase inhibitor. PD173955 inhibited Bcr-Abl-dependent cell growth.
DC12219	PD1-IN-2	PD1-IN-2 is a PD1 signaling pathway inhibitor, which acts as an immunomodulator.

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