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BI-0314

  Cat. No.:  DC12406   Featured
Chemical Structure
2244560-46-9
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More than 5000 active chemicals with high quality for research!
Field of application
BI-0314 (BI0314) is an allosteric activator of protein tyrosine phosphatase non-receptor type 5 (PTPN5, STEP) with potency of 56% at 500 uM, displays no activity against hPTP1B and hTCPTP.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2244560-46-9
Chemical Name: 1-(3-(piperidin-4-yl)-5-(trifluoromethyl)phenyl)guanidine
Synonyms: BI0314;BI 0314
SMILES: N(C1=CC(C(F)(F)F)=CC(C2CCNCC2)=C1)C(=N)N
Formula: C13H17F3N4
M.Wt: 286.302
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: 1. Tautermann CS, et al. J Med Chem. 2018 Sep 12. doi: 10.1021/acs.jmedchem.8b00857.
Description: BI-0314 (BI0314) is an allosteric activator of protein tyrosine phosphatase non-receptor type 5 (PTPN5, STEP) with potency of 56% at 500 uM, displays no activity against hPTP1B and hTCPTP.
References: References 1. Tautermann CS, et al. J Med Chem. 2018 Sep 12. doi: 10.1021/acs.jmedchem.8b00857. View Related Products by Target Protein Phosphatase/PTP
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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