CALP1 TFA

  Cat. No.:  DC41566  
Chemical Structure
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Field of application
CALP1 TFA is a calmodulin (CaM) agonist (Kd of 88 μM) with binding to the CaM EF-hand/Ca2+-binding site. CALP1 TFA blocks calcium influx and apoptosis (IC50 of 44.78 μM) through inhibition of calcium channel opening. CALP1 TFA blocks glutamate receptor channels and blocks a store-operated nonselective cation channel. CALP1 TFA activates CaM-dependent phosphodiesterase activity.
Cas No.:
Chemical Name: CALP1 TFA
Synonyms: VAITVLVK
Formula: C42H76F3N9O12
M.Wt: 956.10
Sotrage: Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS
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COA
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