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PF 750

  Cat. No.:  DC20027   Featured
Chemical Structure
959151-50-9
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More than 5000 active chemicals with high quality for research!
Field of application
PF 750 is a selective and covalent fatty acid amide hydrolase (FAAH) inhibitor, with IC50s varied from 16.2-595 nM in different pre-incubation times. Covalently modifies the enzyme’s active site serine nucleophile.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 959151-50-9
Chemical Name: PF 750
Synonyms: PF 750;N-phenyl-4-(quinolin-3-ylmethyl)piperidine-1-carboxamide;PF-750;Nisoxetine hydrochloride
SMILES: O=C(N1CCC(CC2C=NC3=C(C=CC=C3)C=2)CC1)NC1=CC=CC=C1
Formula: C22H23N3O
M.Wt: 345.437525033951
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: PF 750 is a selective and covalent fatty acid amide hydrolase (FAAH) inhibitor, with IC50s varied from 16.2-595 nM in different pre-incubation times. Covalently modifies the enzyme’s active site serine nucleophile[1].
Target: IC50: 16.2-595 nM (FAAH)[1].
References: [1]. Ahn K, et al. Novel mechanistic class of fatty acid amide hydrolase inhibitors with remarkable selectivity. Biochemistry. 2007 Nov 13;46(45):13019-30.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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