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Home > Molecular Glues

NRX-252262

  Cat. No.:  DC20253   Featured
Chemical Structure
2438637-61-5
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More than 5000 active chemicals with high quality for research!
Field of application
NRX-252262 is a powerful enhancer of the interaction between β-Catenin and its cognate E3 ligase, SCFβ-TrCP. It effectively induces the degradation of mutant β-catenin, demonstrating an EC50 of 3.8 nM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2438637-61-5
Chemical Name: NRX-252262
Synonyms: NRX-252262
SMILES: C1C(Cl)=C(C(=CC=1)Cl)SC1=C(C(N([H])C(C(F)(F)F)=C1)=O)C(=O)N1CC2=C(C=C(C(OC)=C2)OC)C1
Formula: C23N2O4F3Scl2H17
M.Wt: 545.3583
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
DC67413 MRT-23227
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