DB818|cas 790241-43-9|DC Chemicals

Cas No.:	790241-43-9
Chemical Name:	1H-Benzimidazole-5-carboximidamide,2-[5-[4-(aminoiminomethyl)phenyl]-2-thienyl]-
SMILES:	N\N=C\C1=CC=C(C=C1)C2SC(=CC=2)C3=NC4=C(C=CC(C(N)=N)=C4)N3
Formula:	C₁₉H₁₆N₆S
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

DB818 (DB-818, DB 818) is a small molecule inhibitor of HOXA9/DNA interaction through binding as minor groove DNA ligand on the HOXA9 cognate sequence; directly bind to HOXA9-cognate sequence with Kd value of 4.6 nM (HBS sequence); alters HOXA9-mediated transcription, cell survival and cell cycle inHOXA9-mediated HOXA9-expressing murine MigA9 cell line.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

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