ALG1001 (Risuteganib)|CAS 1307293-62-4|DC Chemicals

Cas No.:	1307293-62-4
Chemical Name:	Luminate
Synonyms:	123DNA66IA;Risuteganib;Luminate;Risuteganib [USAN];ALG1001;Glycyl-L-arginylglycyl-3-sulfo-L-alanyl-L-threonyl-L-proline;L-Proline, glycyl-L-arginylglycyl-3-sulfo-L-alanyl-L-threonyl-
SMILES:	S(C[C@@H](C(N[C@@H]([C@@H](C)O)C(N1CCC[C@H]1C(=O)O)=O)=O)NC(CNC([C@H](CCC/N=C(\N)/N)NC(CN)=O)=O)=O)(=O)(=O)O
Formula:	C₂₂H₃₉N₉O₁₁S
M.Wt:	637.666
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

ALG1001 (Risuteganib, ALG-1001) is a first-in-class, RGD class oligopeptide that inhibits integrin receptors (αvβ3, αvβ5, and α5β1) associated with angiogenesis; ALG1001 inhibits an integrin-mediated pathway of the vitreoretinal interface, connecting the posterior aspect of the vitreous with the internal limiting membrane of the retina. In blocking this pathway, ALG-1001 helps to achieve vitreous breakdown and separation from the retina. Other Indication Phase 2 Clinical

MSDS

COA

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2018-0101

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