Cas No.: | 710654-74-3 |
Chemical Name: | 3-((2R,5S)-5-methyl-4-propylmorpholin-2-yl)phenol |
Synonyms: | PF 219061;PF219061 |
Formula: | C14H21NO2 |
M.Wt: | 235.327 |
Purity: | >98% |
Sotrage: | 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Description: | PF-219061 (PF 219061, PF219061) is a potent, selective agonist of dopamine D3 receptor with EC50 of 8 nM; has >1000-fold functional selectivity over D2, displays minimal binding activity (IC50>10 uM) against a wide panel of targets including dopamine D1 and D5 receptors; demonstrates activity in animal models of male erectile dysfunction. |