Methoxy-PEPy

  Cat. No.:  DC23215  
Chemical Structure
524924-76-3
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More than 5000 active chemicals with high quality for research!
Field of application
Methoxy-PEPy is a potent, selective mGlu5 receptor antagonist with IC50 of 1 nM.
Cas No.: 524924-76-3
Chemical Name: Pyridine, 3-methoxy-5-[2-(2-pyridinyl)ethynyl]-
SMILES: COC1C=C(C#CC2=NC=CC=C2)C=NC=1
Formula: C13H10N2O
M.Wt: 210.2313
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Methoxy-PEPy is a potent, selective mGlu5 receptor antagonist with IC50 of 1 nM; exhibits 14-fold higher binding in forebrain relative to cerebellum in mGlu5 receptor-deficient mice, the radioligand [3H]methoxy-PEPy is useful for determining the occupancy of mGlu5 receptors in the brain.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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