N6-Cyclohexyladenosine

  Cat. No.:  DC23227   Featured
Chemical Structure
36396-99-3
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More than 5000 active chemicals with high quality for research!
Field of application
An adenosine A1 receptor agonist (EC50= 8.2 nM)..
Cas No.: 36396-99-3
Chemical Name: (2R,3R,4S,5R)-2-(6-(Cyclohexylamino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol
Synonyms: (2R,3R,4S,5R)-2-(6-(Cyclohexylamino)-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol;Adenosine,N-cyclohexyl-;CHA;N6-Cyclohexyladenosine;Cyclohexyladenosine;N-Cyclohexyladenosine
SMILES: C1(NC2N=CN=C3C=2N=CN3C2C(O)C(O)C(CO)O2)CCCCC1
Formula: C16H23N5O4
M.Wt: 349.384923219681
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM).
Target: A1 receptor
In Vivo: N6-Cyclohexyladenosine exerts anticonvulsant effects and protects against neuronal death. CHA was also found to inhibit the pressor effects of lumbar sympathetic nerve stimulation in rats.
References: [1]. Asghari AA, et al. Adenosine A1 receptor agonist, N6-cyclohexyladenosine, protects myelin and induces remyelination in an experimental model of rat optic chiasm demyelination; electrophysiological and histopathological studies. J Neurol Sci. 2013 Feb 15;3
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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