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STD-101-D1

  Cat. No.:  DC23481   Featured
Chemical Structure
2151041-09-5
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More than 5000 active chemicals with high quality for research!
Field of application
STD-101-D1 is a novel brain permeable, G protein-biased beta-1 adrenergic receptor (ADRB1) partial agonist with EC50 of 16.9 nM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2151041-09-5
Chemical Name: Schembl22279186
Synonyms: (S)-4-(2-Hydroxy-3-((2-(2-methoxyphenoxy)ethyl)amino)propoxy)phenol;Schembl22279186
SMILES: O(C1C=CC(=CC=1)O)C[C@H](CNCCOC1C=CC=CC=1OC)O
Formula: C18H23NO5
M.Wt: 333.378925561905
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: References 1. Yi B, et al. PLoS One. 2017 Jul 26;12(7):e0180319. View Related Products by Target Adrenergic Receptor
Description: STD-101-D1 is a novel brain permeable, G protein-biased beta-1 adrenergic receptor (ADRB1) partial agonist with EC50 of 16.9 nM; engages very little beta-arrestin recruitment compared to the unbiased agonist isoproterenol; also inhibits the acute peripheral and CNS TNFα response induced by LPS both in vitro and in vivo.
References: References 1. Yi B, et al. PLoS One. 2017 Jul 26;12(7):e0180319. View Related Products by Target Adrenergic Receptor
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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