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Tipifarnib S enantiomer

  Cat. No.:  DC24098   Featured
Chemical Structure
192185-71-0
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More than 5000 active chemicals with high quality for research!
Field of application
Tipifarnib S enantiomer is a potent and selective inhibitor of FTase (farnesyltransferase).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 192185-71-0
Chemical Name: 2(1H)-Quinolinone, 6-[(S)-amino(4-chlorophenyl)(1-methyl-1H-imidazol-5-yl)methyl]-4-(3-chlorophenyl)-1-methyl-
Synonyms: (S)-(-)-R-115777;IND-58359 S enantiomer
SMILES: O=C1C=C(C2C=C(Cl)C=CC=2)C2C=C(C=CC=2N1C)C(C1N(C)C=NC=1)(N)C1C=CC(Cl)=CC=1
Formula: C27H22Cl2N4O
M.Wt: 489.3958
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: Tipifarnib S enantiomer is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase (FTase) inhibitor with IC50 of 0.6 nM. Tipifarnib S enantiomer is the less active isomer.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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