MDK-8582（Hnps-PLA Inhibitor）|cas 185298-58-2

Cas No.:	185298-58-2
Chemical Name:	2-(4-(2-Amino-2-oxoethoxy)-1-benzyl-2-ethyl-1H-indol-3-yl)-2-oxoacetamide
Synonyms:	2-(4-(2-amino-2-oxoethoxy)-1-benzyl-2-ethyl-1H-indol-3-yl)-2-oxoacetamide;hnps-PLA Inhibitor;MDK-8582(Hnps-PLA Inhibitor);BCP17761;BDBM50055402;2-(1-Benzyl-4-carbamoylmethoxy-2-ethyl-1H-indol-3-yl)-2-oxo-acetamide;2-{[1-benzyl-3-(carbamoylcarbonyl)-2-ethyl-1H-indol-4-yl]oxy}acetamide
SMILES:	O(C([H])([H])C(N([H])[H])=O)C1=C([H])C([H])=C([H])C2=C1C(C(C(N([H])[H])=O)=O)=C(C([H])([H])C([H])([H])[H])N2C([H])([H])C1C([H])=C([H])C([H])=C([H])C=1[H]
Formula:	C₂₁N₃O₄H₂₁
M.Wt:	379.4091
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

MDK-8582, also known as Hnps-PLA Inhibitor, is an nhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA). The best one inhibited hnps-PLA(2) and LTA(4)H-h with IC(50) values of 9.2 ± 0.5 μM and 2.4 ± 1.4 μM, respectively.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101
2018-0101

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