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QQN52061

  Cat. No.:  DC44603   Featured
Chemical Structure
907952-06-1
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More than 5000 active chemicals with high quality for research!
Field of application
QQN52061 is GPR34 receptor modulator, which can control function of GPR34 receptor (as antagonist or inverse agonist). QQN52061 was first reported in PCT Int. Appl. (2006), WO 2006088246. This product has not formal name. For the convenience of scientific communication, we named it by combining its Inchi key (3 letters from the first letter of each section) with the last 5 digit of its CAS#) according to MedKoo Chemical Nomenclature .
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 907952-06-1
Chemical Name: N-[(2E)-3-(4'-Chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)tyrosine
Synonyms: QQN52061; QQN-52061; QQN 52061;
SMILES: O=C(O)[C@H](CC1=CC=C(OCC2=CC=CC=C2)C=C1)NC(/C=C/C3=CC=C(C4=CC=C(Cl)C=C4)C=C3)=O
Formula: C31H26ClNO4
M.Wt: 512.002
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: QQN52061 is a GPR34 receptor antagonist. GPR34 receptor antagonist 2 can be used for immune diseases, inflammatory diseases research[1].
Target: GPR34 receptor[1]
In Vitro: Endogenous ligands of GPR34, a G protein-coupled receptor, act on histamine-releasing activity on antigen- or concanavalin A-stimulated rat mast cells and synergize with nerve growth factor on rat mast cells. It is a lipid such as lysophosphatidylserine having the activity of releasing histamine. GPR34 antagonists can be used, for example, for histamine release inhibitors, immune diseases, edema, hyperacidity, etc[1].
References: [1]. Fumio Ito, et al. Agent for controlling function of gpr34 receptor. WO2006088246 A1.
MSDS
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MSDS_28309_DC44603_907952-06-1
COA
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Cat. No. Product name Field of application
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