Saclofen|GABAB receptor antagonist|DC Chemicals

Cas No.:	125464-42-8
Chemical Name:	3-AMino-2-(4-chlorophenyl)propane-1-sulfonic acid
Synonyms:	Saclofen
SMILES:	ClC1=CC=C(C(CN)CS(O)(=O)=O)C=C1
Formula:	C₉H₁₂ClNO₃S
M.Wt:	249.71
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

Saclofen is a competitive antagonist of the GABAB receptor with an IC50 of 7.8 μM. Saclofen can be used to determine the functional roles for the GABAB receptor as a mediator of slow inhibitory postsynaptic potentials in the brain[1].

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101
2018-0101

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