PREX-in1|CAS 674801-27-5|DC Chemicals

Cas No.:	674801-27-5
Chemical Name:	PREX-in1
SMILES:	N#CC1=C(N)OC2=NNC(C3=CC=C(OC)C=C3)=C2C1C4=CC=C(C5=CC=C(Cl)C=C5)O4
Formula:	C₂₄H₁₇ClN₄O₃
M.Wt:	444.88
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

MSDS

Cat. No.	Product name	Field of application
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DC74557	PREX-in1	PREX-in1 is a specific small-molecule inhibitor of P-Rex1 and P-Rex2 Rac-GEF activity with IC50 of 4.5 uM (P-Rex1 DHPH Rac-GEF activity) in liposome-based GEF assay, inhibits P-Rex1 and P-Rex2 through their catalytic DH domain.