Cat. No. | Product name | CAS No. |
DC9666 |
Ro 46-2005
Featured
Ro 46-2005 is a novel synthetic non-peptide endothelin receptor antagonist, inhibits the specific binding of 125I-ET-1 to human vascular smooth muscle cells (ETA receptor) with IC50 of 220 nM. |
150725-87-4 |
DC10583 |
RO 5028442
Featured
RO5028442 is a highly potent and selective Brain-Penetrant Vasopressin 1a (V1a) receptor antagonist with Kis of 1 nM (hV1a) and 39 nM (mV1a). |
920022-47-5 |
DC5015 |
Rotigotine Hydrochloride
Rotigotine is dopamine D2 and D3 receptor agonist. Ki values are 13 and 0.71 nM for D2 and D3 respectively. Rotigotine also has significant affinity for 5-HT1A and adrenergic α2B receptors. Rotigotine exhibits antiparkinsonian acitivity. |
125572-93-2 |
DCAPI1584 |
Roxatidine Acetate Hydrochloride
Roxatidine Acetate Hydrochloride is a histamine H2-receptor antagonist used in ulcer treatment. This compound has been found to inhibit platelet function in vitro. |
93793-83-0 |
DC9251 |
RS-102895 hydrochloride
Featured
RS 102895 hydrochloride is a chemokine receptor CCR2 antagonist. |
1173022-16-6 |
DC12250 |
RS 17053 hydrochloride (RS-17053)
RS 17053 hydrochloride is a potent and selective α1A adrenoceptor antagonist, with a pKi value of 9.1 in native cell membrane and a pA2 value of 9.8 in functional assays. |
169505-93-5 |
DC8334 |
RS-127445
Featured
RS-127445 is a potent and selective antagonist at the serotonin 5-HT2B receptor, with around 1000x selectivity over the closely related 5-HT2A and 5-HT2C receptors. |
199864-87-4 |
DC11039 |
RTI-13951-33
Featured
RTI-13951-33 is a potent, selective, brain-penetrant agonist of the orphan receptor GPR88 with EC50 of 25 nM in in vitro cAMP functional assay. |
2244884-08-8 |
DCAPI1593 |
Rupatadine
Featured
Rupatadine is a dual histamine H1 and PAF antagonist |
182349-12-8 |
DC11271 |
S38093 HCl
Featured
S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors. |
1222097-72-4 |
DC10392 |
S1p receptor agonist 1
S1p receptor agonist 1 is an S1P receptor agonist extracted from patent WO 2015039587 A1, compound example 2. |
1514888-56-2 |
DC7274 |
S1RA
Featured
S1RA(E-52862) is a potent and selective sigma-1 receptor(σ1R, Ki=17 nM), showed good selectivity against σ2R (Ki > 1000 nM). |
878141-96-9 |
DC9264 |
S1RA hydrochloride
Featured
S1RA(E-52862) is a potent and selective sigma-1 receptor(σ1R, Ki=17 nM), showed good selectivity against σ2R (Ki > 1000 nM). |
1265917-14-3 |
DC11346 |
Salbutamol (hydrochloride)
Featured
Salbutamol is an agonist of the β2-adrenergic receptor (β2-AR; Kd = 759 nM in a radioligand binding assay using CHO cells expressing the human receptor). |
50293-90-8 |
DC8436 |
Salmeterol Xinafoate
Featured
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptoms. |
94749-08-3 |
DC8610 |
Salmeterol
Featured
Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstructive pulmonary disease (COPD) symptoms. |
89365-50-4 |
DC10925 |
SAR-100842
SAR-100842 (SAR100842) is a potent, selective, orally available antagonist of the Lysophosphatidic Acid 1 Receptor (LPA1 receptor) with IC50 of 31 nM in β-arrestin assays. |
1195941-38-8 |
DC9313 |
Sarpogrelate (hydrochloride)
Featured
Sarpogrelate(MCI-9042) hydrochloride, a selective 5-HT2 antagonist, has been widely used as an anti-platelet agent for the treatment of PAD. |
135159-51-2 |
DC7245 |
SB 222200
SB 222200 is a selective, reversible and competitive antagonist of human NK-3 receptor(Ki=4.4 nM) that effectively crosses the blood-brain barrier. |
174635-69-9 |
DC8878 |
SB 242084
SB 242084 is a potent and selective antagonist of 5-HT2C receptor. |
181632-25-7 |
DC7913 |
SB225002
Featured
SB225002 is a potent, and selective CXCR2 antagonist with IC50 of 22 nM for inhibiting interleukin IL-8 binding to CXCR2, > 150-fold selectivity over the other 7-TMRs tested. |
182498-32-4 |
DC4102 |
SB-269970,SB 269970
Featured
SB269970 is a potent and selective 5-HT7 receptor antagonist. |
201038-74-6 |