Cat. No. | Product name | CAS No. |
DC22418 |
CCX-771
A potent, selective CXCR7 antagonist with IC50 of 4.1 nM. |
|
DC22912 |
SCH39166
A potent, selective D1 dopamine receptor antagonist with Ki of 3.6 nM, >300-fold selectivity over D2 and 5-HT2 receptors. |
1227675-51-5 |
DC11897 |
Garvagliptin
A potent, selective dipeptidyl peptidase-4 (DPP-4) inhibitor for treatment for type 2 diabetes.. |
1601479-87-1 |
DC12015 |
SKF 83566 hydrobromide
A potent, selective dopamine D1 receptor antagonist with Ki of 0.56 nM. |
108179-91-5 |
DC22910 |
ABT-724
A potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors. |
70006-24-5 |
DC22909 |
ABT-724 trihydrochloride
A potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors. |
587870-77-7 |
DC11973 |
A-412997
A potent, selective dopamine D4 receptor agonist with Ki of 12.1 and 7.9 nM for rat and human D4 receptors, respectively. |
1347744-96-0 |
DC11866 |
AZD 3147
Featured
A potent, selective dual mTORC1 and mTORC2 inhibitor with enzyme IC50 of 1.5 nM. |
1101810-02-9 |
DC22586 |
AZD9496 maleate
A potent, selective estrogen receptor downregulator (SERD) with ER downregulation pIC50 of 9.68. |
1639042-28-6 |
DC20378 |
FABP4 inhibitor 1
A potent, selective FABP4 inhibitor with Ki of 30 nM.. |
1526928-21-1 |
DC11956 |
CCG 258748
A potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM. |
|
DC22881 |
GLP1-agonist-1
A potent, selective GLP-1 agonist. |
281208-76-2 |
DC20392 |
GLUT4-IN-17
A potent, selective glucose transporter 4 (GLUT4) inhibitor with IC450 of 10.8 uM, inhibits MM cell proliferation. |
1061081-61-5 |
DC22747 |
AICP
A potent, selective GluN2C-selective NMDA receptor glycine site superagonist with EC50 of 1.7 nM at GluN1/2C. |
861213-66-3 |
DC11838 |
Org 25935
A potent, selective glycine transporter 1 (GlyT1) inhibitor with IC50 of 100 nM. |
949588-40-3 |
DC23558 |
(+)-NFPS
A potent, selective GlyT1 inhibitor that demonstrates >10-fold greater activity in in vitro functional glycine reuptake assay than racemic (±)-NFPS. |
571147-18-7 |
DC11616 |
KUNG94
A potent, selective Grp94 inhibitor with IC50 of 8 nM. |
2134571-29-0 |
DC11619 |
KUNG29
A potent, selective Grp94 inhibitor with Kd of 0.2 uM. |
1887032-92-9 |
DC11618 |
KUNG38
A potent, selective Grp94 inhibitor with Kd of 0.44 uM. |
1887033-00-2 |
DC11617 |
PU-H54
Featured
PU-H54 is potent, selective Grp94 inhibitor. |
1454619-13-6 |
DC20400 |
HDAC1,2-IN-2
A potent, selective HDAC1 and HDAC2 inhibitor with IC50 of 6 nM and 45 nM, respectively. |
937727-03-2 |
DC11597 |
SB-429201
A potent, selective HDAC1 inhibitor with IC50 of 1.5 uM. |
1027971-34-1 |