| Cat. No. | Product Name | Field of Application | Chemical Structure |
|---|---|---|---|
| DC11955 | Takeda compound 101 Featured | Compound 101 (GRK2 inhibitor 101, Takeda compound 101, Cmpd101) is a novel membrane-permeable, small-molecule inhibitor of GRK2 and GRK3. |
|
| DC10933 | Compound 3-110-22 | Compound 3-110-22 is a small molecule that inhibits dengue virus (DENV) by binding to its envelope protein E. |
|
| DC22270 | Compound 621433144 | Compound 621433144 (ZINC000621433144, Z3269026405) is a potent, selective full agonist of the D4 receptor with 2,500-fold subtype selectivity. |
|
| DC22117 | Compound 7004 | Compound 7004 (IRAK2 mimetic 7004) is a small molecule mimetic of a-helical domain of IRAK2, inhibit IL-33–induced NF-κB transcriptional activity (IC50=9.7 uM) by disrupting Myddosome formation. |
|
| DC11164 | Compound 919278 | Compound 919278 is a specific inhibitor of lymphotoxin β receptor (LTβR, IC50=0.169 uM), and TNF receptor superfamily member 12A (FN14)-dependent nuclear translocation of p52 (IC50=0.167 uM) via inhibiting CDK12/CCNK, does not inhibit the TNF-α-mediated nuclear translocation of p65 (RelA). |
|
| DC21345 | Contezolid | Contezolid (MRX I) is an orally active oxazolidinone agent with antibacterial activity Gram-positive pathogens, including MRSA, penicillin-PRSP, PISP, and vancomycin-resistant enterococci (VRE) with MIC of 0.25-4 ug/mL. |
|
| DC11048 | Contilisant | Contilisant is a neuroprotective, non-toxic, antioxidant, permeable ligand, showing in vitro pharmacological properties on the selected biological targets (hAChE IC50=0.53 uM. |
|
| DC12098 | Corin Featured | Corin is a dual inhibitor of histone lysine specific demethylase (LSD1) and histone deacetylase (HDAC), with a Ki(inact) of 110 nM for LSD1 and an IC50 of 147 nM for HDAC1. |
|
| DC11104 | Tildacerfont Featured | corticotropin releasing factor (CRF) antagonist. |
|
| DC22488 | Corticotropin-releasing factor (human) Featured | Corticotropin-releasing hormone (CRH) is a peptide hormone involved in the stress response.. |
|
| DC22479 | Cortisone acetate | Cortisone acetate (Cortisone 21-acetate) is a synthetic glucocorticoid corticosteroid and corticosteroid ester. |
|
| DC23908 | Cortisone Featured | Cortisone is a pregnane (21-carbon) steroid hormone, one of the main hormones released by the adrenal gland in response to stress. |
|
| DC8694 | Cortodoxone | Cortodoxone is a glucocorticoid steroid hormone that can be oxygenated to cortisol (Hydrocortisone). |
|
| DC9554 | Cot inhibitor-1 | Cot inhibitor-1 is a COT/Tpl2 inhibitor. |
|
| DC9555 | Cot inhibitor-2 | Cot inhibitor-2 is a COT/Tpl2 inhibitor. |
|
| DC20933 | Cotylimide-VI | Cotylimide-VI (CTL-VI) is a small molecule that perturbs plant hormone strigolactone accumulation and inhibits hypocotyl growth.. |
|
| DC10363 | Coumestrol Featured | Coumestrol, a phytoestrogen present in soybean products, exhibits activities against cancers, neurological disorders, and autoimmune diseases. It suppresses proliferation of ES2 cells with an IC50 of 50 μM. |
|
| DC21413 | Cowanin | Cowanin is a novel natural product from Garcinia speciosa that inhibits the Notch signaling pathway with IC50 of 2.4 uM. |
|
| DC8543 | CP465022 HCl | CP 465022 hydrochloride is a selective GluR (AMPA) antagonist which is non-competitive. |
|
| DC23320 | CP 31398 dihydrochloride Featured | CP-31398 is a small molecule p53 reactivator that protects p53 from thermal denaturation, not only reactivates mutant p53 but also induces stabilization of wild type p53. |
|
| DC23610 | CP-339818 hydrochloride Featured | CP-339818 is a potent, selective, non-peptide KV1.3 channel antagonist with IC50 of 200 nM. |
|
| DC23415 | CP-481715 | CP-481715 is a potent and selective CCR1 antagonist with Ki of 9.2 nM and IC50 of 74 nM, lacks intrinsic agonist activity and . |
|
| DC4132 | CP-547632 Featured | CP-547632 is as a potent inhibitor of the VEGFR-2 and basic fibroblast growth factor (FGF) kinases (IC50 11 and 9 nM, respectively). |
|
| DC8251 | CP-724,714 | CP-724,714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >640-fold selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc. Phase 2. |
|
| DC8892 | CP724714 | CP-724714 is a potent, selective inhibitor of HER2/ErbB2 with IC50 of 10 nM, >640-fold selectivity against EGFR, InsR, IRG-1R, PDGFR, VEGFR2, Abl, Src, c-Met etc in cell-free assays. Phase 2. |
|
| DC9317 | CP-809101 (hydrochloride) | CP-809101 Hcl is a potent and selective 5-HT2C receptor agonist with pEC50 of 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors respectively. |
|
| DC9385 | CPA inhibitor | CPA inhibitor is a potent inhibitor for carboxypeptidase A (CPA). |
|
| DC23544 | CPG-52364 | CPG-52364 (CPG52364) is an orally available, small molecule TLR7/8/9 antagonist for the treatment of systemic lupus erythematosus and other autoimmune disorders.. |
|
| DC7564 | CPI 0610(Pelabresib) Featured | CPI 0610 is a potent, selective, and cell-active BET bromodomain inhibitor with IC50 of 39 nM for BRD4-BD1 in TR-FRET assay. |
|
| DC8002 | CPI-360 (R) Featured | CPI-360 is a compound in design and preparation of wew palladium precatalysts for C-C and C-N cross-coupling reactions. |
|
