DC7825 |
Canagliflozin hemihydrate |
Canagliflozin 0.5 H2O(JNJ 28431754; TA 7284) is a highly potent and selective SGLT2 inhibitor for hSGLT2 with IC50 of 2.2 nM, exhibits 413-fold selectivity over hSGLT1. |
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DC22425 |
Cangrelor sodium
Featured
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Cangrelor (AR-C69931MX) is a potent, selective P2T/P2Y12 receptor antagonist with IC50 of 0.4 nM against ADP-induced aggregation of human platelets. |
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DC4154 |
Capecitabine
Featured
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Capecitabine is a tumor-selective fluoropyrimidine carbamate which achieves higher intratumoral 5-FU level with lower toxicity than 5-FU. |
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DC7615 |
Capromorelin
Featured
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Capromorelin tartrate is a potent ghrelin receptor agonist/growth hormone secretagogue (Ki = 7 nM). |
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DC26044 |
Caprooyl-Tetrapeptide-3 |
Caprooyl tetrapeptide-3 is a derivative of tetrapeptide-3 that is linked to caproic acid. |
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DC7952 |
Capasazepine
Featured
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Capsazepine is a synthetic analogue of the sensory neurone excitotoxin, capsaicin; potent TRPV1 receptor antagonist with IC50 of 562 nM. |
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DC20331 |
Capstafin |
Capstafin is a phosphorylation of capsaicinoid derivative that acts as a highly potent, selective inhibitor of STAT5b with Ki of 0.34 uM. |
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DC21586 |
Capzimin |
Capzimin (Rpn11 inhibitor 3027) is a derivative of 8TQ, and potent and specific inhibitor of proteasome isopeptidase Rpn11 with IC50 of 0.34 uM, >7-fold improved potency over 8TQ (quinoline-8-thiol). |
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DCAPI1210 |
Carbazochrome sodium sulfonate |
Carbazochrome sodium sulfonate |
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DC9173 |
Carbetapentane citrate |
Carbetapentane citrate is a selective inhibitor of the cough, with mild atropine-like effect and local anesthesia effect. |
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DC12087 |
Carboxy pyridostatin trifluoroacetate salt |
Carboxy pyridostatin trifluoroacetate salt has the peculiarity to exhibit high molecular specificity for RNA over DNA G4s. |
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DC6502 |
cardamonin
Featured
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Cardamonin, isolated from the fruits of Alpinia species, is a chalconoid with anti-inflammatory and anti-tumor activity. |
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DC8456 |
Cardiogenol C (hydrochloride)
Featured
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Cardiogenol C is a diaminopyrimidine that induces cardiomyogenesis in mouse embryonic stem cells. |
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DC24127 |
Cardiogenol C hydrochloride |
Cardiogenol C is a small cell-permeable molecule that selectively and efficiently induce mouse embryonic stem cells (ESCs) to differentiate into cardiomyocytes with EC50 of 0.1 uM. |
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DC23875 |
Cardionogen 1 |
Cardionogen 1 (CDNG1) is a small molecule that promotes cardiomyocyte generation by modulating Wnt signaling. |
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DC23881 |
Cardionogen 2 |
Cardionogen 2 (CDNG2) is a small molecule that promotes cardiomyocyte generation by modulating Wnt signaling. |
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DC9012 |
Carisoprodol |
Carisoprodol is a centrally acting skeletal muscle relaxant of the carbamate class and produces all the effects associated with barbiturate receptor ligands. |
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DC21875 |
CARM1 inhibitor 9 |
CARM1 inhibitor 9 is a potent, selective inhibitor of arginine methyltransferase 1 (CARM1, PRMT4) with IC50 of 94 nM. |
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DC24110 |
CARM1-IN-1
Featured
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CARM1-IN-7g is a potent, selective coactivator-associated arginine methyltransferase 1 (CARM1) with IC50 of 8.6 uM, exhibits lower or no activity against a panel of different PRMTs or HKMTs (>80-fold over PRMT1 and SET7). |
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DC8972 |
Carmustine
Featured
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Carmustine is a cell-cycle phase nonspecific alkylating antineoplastic agent. |
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DC20119 |
Carnostatine (SAN9812) |
Carnostatine (SAN9812) is a specific and highly selective carnosinase (CN1) inhibitor with a Ki of 11 nM. |
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DC9119 |
Carvedilol |
Carvedilol(BM14190) is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation. |
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DC10539 |
POL1 inhibitor(POL1-IN-1)
Featured
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CAS 1822358-25-7 |
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DC8013 |
CASIN
Featured
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CASIN is a Cdc42 GTPase inhibitor (IC50 = 2 μM). |
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DC22402 |
Casopitant |
Casopitant (GW679769) is a potent, centrally-acting neurokinin 1 (NK1) receptor antagonist (pKi=9.48) with antidepressant and antiemetic activities. |
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DC22403 |
Casopitant mesylate
Featured
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Casopitant (GW679769) is a potent, centrally-acting neurokinin 1 (NK1) receptor antagonist (pKi=9.48) with antidepressant and antiemetic activities. |
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DC22047 |
CAT639 |
CAT639 is an improved analog of ATV399 that exhibits improved β-cell viability and insulin secretion in the rat insulin-producing INS1E cells and primary rat dispersed islet cells, inhibits dimerization of iNOS. |
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DCAPI1130 |
Catharanthine |
Catharanthine inhibits nicotinic receptor mediated diaphragm contractions with IC50 of 59.6 µM. |
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DC22206 |
Cathepsin B inhibitor RC1 |
Cathepsin B inhibitor RC1 is a small-molecule that blocks the process of anthrax lethal toxin (LT) cytotoxicity, inhibits enzymatic activity of host cathepsin B that mediates the escape of toxins into the cytoplasm from late endosomes. |
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DC10903 |
CAY10465
Featured
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CAY10465 is an analog of resveratrol acting as a potent and selective aryl hydrocarbon receptor agonist, with a Ki of 0.2 nM. |
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