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Cat. No.	Product Name	Field of Application
DC22988	BMS-189453 Featured	BMS-189453 (BMS189453, BMS453) is a synthetic retinoid that acts as an agonist of RARβ and an antagonist of RARα and RARγ.
DC8513	BMS-3 Featured	BMS-3 is a potent inhibitor of the LIM kinase. It has IC50's of 5nM and 6 nM for LIMK1 and LIMK2 respectively.
DC7375	BMS-303141 Featured	BMS-303141 is a potent ATP-citrate lyase (ACL) inhibitor with IC50 value of 0.13 uM (human recombinant ACL).
DC8457	BMS-309403 Featured	BMS309403 is orally active, reducing atherosclerosis in mice lacking apoplipoprotein E.
DC5037	BMS-536924 Featured	BMS-536924 is an ATP-competitive IGF-1R inhibitor with IC50 of 100 nM, modest activity for Mek, Fak, and Lck with very little activity for Akt1, MAPK1/2.
DC7897	BMS-582949 HCl Featured	BMS-582949 is a dual action p38 Kinase Inhibitor.
DC3105	BMS-599626 (AC480) Featured	BMS-599626 (AC480) is a selective and efficacious inhibitor of HER1 and HER2 with IC50 of 20 nM and 30 nM, respectively.
DC7730	Temsavir（BMS-626529） Featured	BMS-626529 is a novel small-molecule attachment inhibitor that targets HIV-1 gp120 and prevents its binding to CD4+ T-cells.
DC9252	BMS-687453 Featured	BMS687453 is a potent and selective peroxisome proliferator activated receptor (PPAR) α agonist, with an EC50 of 10 nM for human PPARα and ∼410-fold selectivity vs human PPARγ in PPAR-GAL4 transactivation assays.
DC9700	BMS-707035 Featured	BMS-707035 is a potent, specific, and reversible HIV-I integrase (IN) inhibitor that blocks HIV IN strand transfer activity.
DC3114	Avagacestat (BMS-708163) Featured	BMS-708163 is a potent, selective γ-secretase inhibitor of Aβ40 and Aβ42 with IC50 of 0.3 nM and 0.27 nM, respectively.
DC3126	BMS754807 Featured	BMS-754807 is a potent and reversible inhibitor of IGF-1R/IR family kinases, inhibits IGF-1R, IR, Met, TrkA and TrkB with IC50 of 1.8 nM, 1.7 nM, 5.6 nM, 7.4 nM and 4.1 nM, respectively.
DC9861	BMS-779788(XL-652) Featured	BMS-779788(XL652) is a novel small-molecule modulator of the Liver X Receptor (LXR), a nuclear hormone receptor implicated in a variety of cardiovascular and metabolic disorders.
DC10494	BMS813160 Featured	BMS-813160 is a dual CCR2/CCR5 chemokine antagonist.
DC12670	BMS-817378 free base Featured	BMS-817378 is a prodrug of the dual Met/VEGFR-2 inhibitor BMS-794833.
DC20815	BMS-823778 Featured	BMS-823778 (BMS823778) is an orally available, potent and selective inhibitor of 11βHSD-1 with IC50 of 2.3 nM, displays >10,000-fold selectivity over 11βHSD-2.
DC7154	BMS-833923 (XL-139) Featured	BMS 833923 is an orally bioavailable inhibitor of Smo. It blocks binding of BODIPY cyclopamine (IC50 = 21 nM) and inhibits Gli activation in cell lines that express wild-type Smo or activated mutant forms of Smo (IC50s = 6-35 nM). BMS 833923 robustly inhi
DC7090	BMS-863233 (XL-413) Featured	BMS-863233, also known as XL-413, is an orally bioavailable cell division cycle 7 homolog (CDC7) kinase inhibitor with potential antineoplastic activity.
DC4175	BMS-911543 Featured	BMS-911543 is a potent and selective inhibitor of JAK2 with IC50 of 1.1 nM, approximately 350-, 75- and 65-fold selective to JAK1, JAK3 and TYK2, respectively.
DC23872	BMS-932481(BMS932481;BMS 932481) Featured	BMS-932481 (BMS932481) is a potent, selective, orraly active γ-secretase modulator (GSM), shows selectivity for Aβ40 and Aβ42 reduction (IC50=6.6 nM) while sparing total Aβ levels both in vitro and in vivo.
DC21092	BMS-955176 Featured	BMS-955176 (GSK-3532795) is a second-generation HIV-1 maturation inhibitor that exhibits potent activity (EC50=3.9±3.4 nM) against a library (n=87) of gag/pr recombinant viruses.
DC20821	BMS-962212 Featured	BMS-962212 is a potent, highly selective and reversible small molecule coagulation Factor XIa (FXIa) inhibitor with Ki of 0.7 nM.
DC10459	BMS-986020 Featured	BMS-986020 is an LPA1 antagonist.
DC11923	BMS-986120 Featured	BMS-986120 (BMS986120) is a potent, selective, orally bioavailable, and reversible PAR4 antagonist with Kd of 0.098 nM for human PAR4.
DC26073	BMS-986122 Featured	BMS-986122 is a potent positive allosteric modulator of μ-opioid receptor, significantly increases the inhibition of forskolin-stimulated adenylyl cyclase activity produced by an EC10 (30 pM) concentration of endomorphin-I in CHO-μ cells..
DC11819	BMS-986142 Featured	BMS-986142 is a potent, selective, and reversible BTK (Bruton’s tyrosine kinase) inhibitor (BTK IC₅₀ = 0.5nM; human WB IC₅₀ = 90 nM).
DC10609	BMS-986158 Featured	BMS-986158 is an inhibitor of the bromodomain and extra-terminal (BET) proteins.
DC12174	Deucravacitinib(BMS986165) Featured	BMS-986165 is a selective, potent, allosteric inhibitor of tyrosine kinase 2 (Tyk2).
DC23532	BMS-986166 Featured	BMS-986166 (BMS986166) is a potent, selective S1P receptor modulator for the treatment of ulcerative colitis..
DC23460	BMS986187 Featured	BMS-986187 is a novel potent, positive allosteric modulator of δ-opioid receptor with EC50 of 30 nM, 100-fold selectivity over μ-opioid receptor..

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