| Cat. No. | Product Name | Field of Application | Chemical Structure |
|---|---|---|---|
| DC12273 | EMT inhibitor-1 | EMT inhibitor-1 is an inhibitor of of Hippo, TGF-β, and Wnt signaling pathways with antitumor activities. |
|
| DC23108 | EN460 Featured | EN460 is a specific mall molecule inhibitor of endoplasmic reticulum oxidation 1 (ERO1), interacts selectively with the reduced, active form of ERO1α and prevents its reoxidation (IC50=1.9 uM). |
|
| DC20892 | Enadoline | Enadoline (CI 977. |
|
| DC20993 | ENMD-1068 Featured | ENMD-1068 is a novel selective PAR2 antagonist without inhibitory activity against thrombin-mediated PAR3 and PAR4 signaling. |
|
| DC8778 | Enocitabine | Enocitabine is an anti-tumor agent and an antineoplastic. A derivative of Cytarabine. |
|
| DC20018 | Enocyanin Featured | Enocyanin is an anthocyanin extracted from grapes. Enocyanin shows inhibitory effect on the leucine aminopeptidase, acid phosphatase, γ-glutamyl transpeptidase and esterase activity. |
|
| DC4208 | Entecavir Monohydrate Featured | Entecavir hydrate belongs to the family of medicines called antivirals. |
|
| DC8881 | Entecavir | Entecavir is a deoxyguanosine nucleoside analogue with antiviral activity against the hepatitis B virus (HBV). |
|
| DC6909 | Entinostat (MS-275) Featured | Entinostat (MS-275) strongly inhibits HDAC1 and HDAC3 with IC50 of 0.51 μM and 1.7 μM, compared with HDACs 4, 6, 8, and 10. Phase 1/2. |
|
| DC21856 | Enviroxime | Enviroxime (Zinviroxime. |
|
| DC20848 | Enzaplatovir | Enzaplatovir (BTA-585, BTA-C585) is an orally bioavailable RSV fusion protein inhibitor for the treatment of respiratory syncytial virus infections.. |
|
| DC20950 | EOAI3402143 | EOAI3402143 (Deubiquitinase inhibitor G9, EOAI 3402143) is a novel covalent deubiquitinase Usp9x/Usp24 inhibitor with increased aqueous solubility and greater cellular Usp9x inhibitory activity than WP1130. |
|
| DC21601 | Epertinib | Epertinib (S-222611) is a novel potent, orally active, reversible EGFR and HER2 inhibitor with IC50 of 1.48, 7.15 and 2.49 nM for EGFR, HER2 and HER4, respectively. |
|
| DC20374 | EphB3-IN-1 | EphB3-IN-1 is the first potent, selective inhibitor of EphB3 that exhibits inhibiting EphB3 autophosphorylation in cells with IC50 of 3 nM. |
|
| DC11433 | Vatiquinone | EPI-743 (Vatiquinone,EPI-589) is an orally bioavailable para-benzoquinone for treatment of inherited mitochondrial diseases, an analogue of the antioxidant ubidecarenone. |
|
| DC9363 | Epibrassinolide | Epibrassinolide (EBR; B1105; 24-Epibrassinolide) is a biologically active compound of the brassinosteroids, steroid-derived plant growth regulator family; was shown as a potential apoptotic inducer in various cancer cells without affecting the non-tumor c |
|
| DC9467 | Epinastine Featured | Epinastine(WAL801) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis. |
|
| DC23786 | Epolactaene | Epolactaene is a neuritogenic fungal isolate that arrests the cell cycle at the G0/G1 phase and induces the outgrowth of neurites in human neuroblastoma SH-SY5Y cells. |
|
| DC7120 | Epothilone A | Epothilone A is a Taxol-like microtubule-stabilizing agent that induces tubulin polymerization, leading to cell cycle arrest at the G2-M transition, cytotoxicity, and apoptosis. |
|
| DC4198 | Epothilone B Featured | Epothilone B is a Taxol-like microtubule-stabilizing agent with EC0.01 of 1.8 μM. |
|
| DC7012 | Epothilone D | Epothilone D(Desoxyepothilone B; KOS 862) is a natural polyketide compound isolated from the myxobacterium Sorangium cellulosum. |
|
| DC8030 | Epoxomicin Featured | Epoxomicin is a selective and irreversible inhibitor of 20S proteasome with an IC50 value of 4 nM. |
|
| DC12311 | Eprobemide (LIS 630) Featured | Eprobemide is a non-competitive reversible inhibitor of monoamine oxidase A. |
|
| DC12529 | EPZ020411 dihydrochloride | EPZ020411 is a potent, selective PRMT6 inhibitor with IC50 of 10 nM, displays 10-fold and 20-fold selectivity over PRMT1/8, and >100-fold over other histone methyltransferases (PRMT3/4/5/7). |
|
| DC23134 | EPZ020411 hydrochloride | EPZ020411 is a potent, selective PRMT6 inhibitor with IC50 of 10 nM, displays 10-fold and 20-fold selectivity over PRMT1/8, and >100-fold over other histone methyltransferases (PRMT3/4/5/7). |
|
| DC20996 | EPZ 025654 | EPZ025654 (GSK 35336023) is a potent, selective arginine methyltransferase CARM1 inhibitor with IC50 of 3 nM. |
|
| DC22657 | EPZ-030456 | EPZ-030456 (EPZ030456) is a potent, selective SMYD3 inhibitor with biochem IC50 of 4 nM. |
|
| DC8595 | Equisetin | Equisetin is an N-methylserine-derived acyl tetramic acid produced by a number of Fusarium species with antibiotic and cytotoxic activity. |
|
| DC20997 | ER000444793 Featured | ER-000444793 is a potent, cyclophilin D-independent inhibitor of mitochondrial permeability transition pore (mPTP) with with IC50 of 2.8 uM. |
|
| DC22468 | ER-27319 maleate | ER-27319 maleate is a potent, selective inhibitor of antigen or anti-IgE-mediated degranulation of rodent and human mast cells by selective inhibition of FcɛRI-mediated activation of Syk. |
|
