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Cat. No. Product name CAS No.
DC23305 BM-1197

BM-1197 is a potent, specific dual inhibitor of Bcl-2 and Bcl-xL with Ki of <1 nM, shows >1,000-fold selectivity over Mcl-1.

1391107-89-3
DC20802 BM-635

BM-635 is a small molecule anti-mycobacterial compound acting by inhibiting the mycobacterial membrane protein Large 3 (MmpL3).

1073372-01-6
DC23304 BM-957

BM-957 is a highly potent, dual Bcl-2 and Bcl-xL inhibitor with Ki of <1 nM for both, IC50 of 5.4 and 6.0 nM, respectively.

1391107-54-2
DC20321 Bm-MPK1-IN-15b

Bm-MPK1-IN-15b is a potent, orally bioavailable inhibitor of B. malayi stress-activated kinase Bm-MPK1 with IC50 of 24 nM.

2222294-62-2
DC8452 BMN-673 8R,9S

BMN-673 (8R,9S) is the (8R,9S) enantiomer of BMN-673. BMN 673 is a novel PARP inhibitor with IC50 of 0.58 nM(PARP1). It does not inhibit PARG and is highly sensitive to PTEN mutation.

1207456-00-5
DC23833 SB 4 (Eticovo) Featured

BMP signaling agonist sb4 is a small molecule BMP signaling agonist with EC50 of 73.6 nM, enhances the efficacy of BMPs and activates endogenous BMP4 target genes.

100874-08-6
DC20812 BMS 695735

BMS 695735 is a potent, selective IGF-1R inhibitor with IC50 of 34 nM.

1054315-48-8
DC11761 BMS-816336

A novel potent, selective, orally active human 11β-HSD1 inhibitor with IC50 of 3.0 nM.

1009583-20-3
DC22988 BMS-189453 Featured

BMS-189453 (BMS189453, BMS453) is a synthetic retinoid that acts as an agonist of RARβ and an antagonist of RARα and RARγ.

166977-43-1
DC8515 BMS-2

BMS-2 is a potent MET kinase inhibitor with an IC50 value of 1.8nM. It also possesses potent inhibitory activity against Flt-3 and VEGFR-2 kinases, IC50 values of 4nM and 27nM respectively.

888719-03-7
DC22032 BMS-211

BMS-211 is a prodrug of the parent pan-CK2 inhibitor BMS-699..

DC11294 BMS-212

BMS-212 is a potent and selective stimulator of glucokinase (GK) (EC50 = 35 nM) that is promisingly used as an antidiabetic.

2173153-38-1
DC10200 BMS-214662

BMS-214662 is a potent and selective farnesyl transferase inhibitor with potent antitumor activity with an IC50 of 1.35 nM.

195987-41-8
DC8762 BMS-265246

BMS-265246 is a potent and selective CDK1/2 inhibitor for CDK1/cyclin B and CDK2/cyclin E with IC50 of 6 nM and 9 nM, respectively.

582315-72-8
DC20808 BMS-394136

BMS-394136 is a potent, selective IKur/Kv1.5inhibitor, increases atrial action potential duration (APD) and prolongs AERP but not VERP in both rabbits and beagles..

343246-73-1
DC20809 BMS433771

BMS433771 is a potent, orally active RSV fusion inhibitor, exhibits excellent potency against multiple laboratory and clinical isolates of both group A and B viruses with mean EC50 of 20 nM.

543700-68-1
DC23529 BMS-457

BMS-457 is a potent and selective CCR1 antagonist with binding IC50 of 0.8 nM, >1,000-fold selectivity against other CC family receptors.

946594-19-0
DC7007 BMS-538203

BMS-538203 is a highly efficient HIV integrase inhibitor and antiviral agent.

543730-41-2
DC23167 BMS-564929

BMS-564929 is a potent, selective androgen receptor modulator (SARM) that binds to AR with Ki of 2.11 nM.

627530-84-1
DC22033 BMS-595

BMS-595 (BMS595) is a novel potent, selective, ATP-competitive casein kinase 2 (CK2) inhibitor with IC50 of 1.3 nM (CKα).

DC24131 BMS-599626 hydrochloride

BMS-599626 (AC-480) is a potent, selective inhibitor of EGFR and HER2 with IC50 of 20 nM and 30 nM.

873837-23-1
DC20805 BMS-641988

BMS-641988 is a potent, selective, nonsteroidal androgen receptor antagonist with Ki of 1.7 nM, MDA-MB-453 cell IC50 of 16 nM.

573738-99-5
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