| DC23182 |
ABX464
Featured
|
ABX464 (ABX-464, ABX 464) is a novel class of anti-HIV small molecule targeting Rev-mediated viral RNA biogenesis, shows dose dependent inhibition of HIV-1 replication in stimulated PBMCs with IC50 of 0.1-0.5 uM. |
|
| DC7698 |
AC 55541
Featured
|
AC 55541 is a potent and selective protease-activated receptor 2 (PAR2) agonist (pEC50 = 6.7) that displays no activity at other PAR subtypes or at over 30 other receptors involved in nociception and inflammation. |
|
| DC12577 |
AC-263093
Featured
|
AC-263093 (AC263093) is a potent, functionally selective neuropeptide FF receptor type 2 (NPFFR2) agonist with pKi of 6.9. |
|
| DC20300 |
AC-4-130 |
AC-4-130 is a novel, potent STAT5 SH2 domain inhibitor, binds to and efficiently blocks STAT5 activation and subsequent transcriptional activity, shows high selectivity for STAT5 over STAT1 and STAT3. |
|
| DC21863 |
AC5 inhibitor C90 |
AC5 inhibitor C90 is a novel potent, selective adenylyl cyclase type 5 (AC5) inhibitor with IC50 of 30 nM, >5-fold selectivity over AC2 and AC6 subtypes. |
|
| DC12086 |
AC-55649
Featured
|
AC-55649 is a potent, highly isoform-selective agonist of human RARβ2 receptor, with a pEC50 of 6.9. |
|
| DC7700 |
AC710
Featured
|
AC710, is a potent Globally Selective Inhibitor of Platelet-Derived Growth Factor Receptor-Family Kinases. |
|
| DC12492 |
N-(p-Amylcinnamoyl) anthranilic Acid (ACA)
Featured
|
ACA is a cell permeable inhibitor of PLA2,reported to inhibit α-ketoisocaproic acid and glyceraldehyde-induced insulin secretion, as well as glucose-induced insulin secretion. |
|
| DC9917 |
Acacetin
Featured
|
Acacetin is an O-methylated flavone found in Robinia pseudoacacia (black locust), Turnera diffusa (damiana),Betula pendula (silver birch),and in the fern Asplenium normale. |
|
| DC22280 |
Acarbose
Featured
|
Acarbose is the first identified α-glucosidase inhibitor. |
|
| DC11458 |
Ac-DEVD-pNA(Caspase-3 Substrate)
Featured
|
Ac-DEVD-pNA is a colorimetric substrate for caspase-3 (CPP32) (Km=9.7μM) and related cysteine proteases. |
|
| DC11359 |
Caspase-3 Substrate |
Ac-DNLD-AMC is a fluorogenic caspase-3 substrate. |
|
| DC9986 |
Acebilustat(ZK322)
Featured
|
Acebilustat(ZK322) is a potent and selective leukotriene A4 hydrolase inhibitor. |
|
| DC10592 |
ASL 601(Acecainide)
Featured
|
Acecainide, also known as N-acetylprocainamide and ASL 601, is the N-acetylated metabolite of procainamide. |
|
| DC9127 |
Acemetacin |
Acemetacin is a non-steroidal anti-inflammatory drug and a glycolic acid ester of indometacin that is a cyclooxygenase inhibitor. |
|
| DCAPI1009 |
Acetanilide (Antifebrin) |
Acetanilide (Antifebrin) |
|
| DC8978 |
Acetazolamide |
Acetazolamide is a potent carbonic anhydrase (CA) inhibitor; best-studied agent for the amelioration of acute mountain sickness (AMS). |
|
| DC20115 |
Acetoacetic acid sodium salt |
Acetoacetic acid sodium salt is a metabolite of non-esterified fatty acids, involved in the development of human diabetes. Acetoacetic acid sodium salt induces oxidative stress to inhibit the assembly of very low density lipoprotein in bovine hepatocytes. |
|
| DC10248 |
Acetohydroxamic acid |
Acetohydroxamic acid is an Urease Inhibitor. In the urine, it acts as an antagonist of the bacterial enzyme urease. |
|
| DC20151 |
Acetosyringone
Featured
|
Acetosyringone is a phenolic compound from wounded plant cells, enables virA gene which encodes a membrane-bound kinase to phosphorylate itself and activate the virG gene product, which stimulates the transcription of other vir genes and itself. Acetosyri |
|
| DC12151 |
Acetyl Perisesaccharide C |
Acetyl Perisesaccharide C is an oligosaccharide, which is isolated from the root barks of Periploca sepium. |
|
| DC9894 |
Acetylcholine iodide |
Acetylcholine iodide is a neurotransmitter found at neuromuscular junctions, autonomic ganglia, parasympathetic effector junctions, a subset of sympathetic effector junctions, and at many sites in the central nervous system. |
|
| DC10637 |
Acetylspiramycin (ASPM) |
Acetylspiramycin (ASPM) is a macrolide antimicrobial agent. |
|
| DC21985 |
Ac-IEPD-CHO |
Ac-IEPD-CHO is a potent, reversible inhibitor of serine protease Granzyme B (GzmB) with Ki of 80 nM, also inhibits caspase-7 (Ki=550 nM) and induces apoptosis.. |
|
| DC11350 |
Caspase-8 Chromogenic Substrate I |
Ac-IETD-pNA is a substrate for caspase-8. |
|
| DCAPI1205 |
Acipimox |
Acipimox |
|
| DC1092 |
Acitazanolast (WP-871,Zepelin) |
Acitazanolast is an active metabolite of tazanolast and anti-allergic drug. |
|
| DCAPI1244 |
Acitretin |
Acitretin |
|
| DC22805 |
(R)-9b |
Ack1 inhibitor (R)-9b is a potent and selective ACK1 (TNK2) inhibitor with IC50 of 48 nM. |
|
| DC21864 |
Ack1 inhibitor 37 |
Ack1 inhibitor 37 is a potent and selective Ack1 (TNK2) inhibitor with Ki of 0.3 nM, displays high selectivity over related kinases LCK, JAK3, KDR and TIE2 (Ki= 138, 6.5, 380 and 200 nM). |
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