DCC5399 |
Ver-246608 |
Novel pan-isoform ATP competitive inhibitor of pyruvate dehydrogenase kinase, disrupting Warburg metabolism and inducing context-dependent cytostasis in cancer cells |
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DCC5400 |
veratramine Hydrochloride |
Antitumor agent |
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DCC5401 |
Veratridine |
Natural Janus-Faced Modulator of Voltage-Gated Sodium Ion Channels, acting on the channel as either an agonist or antagonist depending on the nature of the electrophysiological stimulation protocol |
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DCC5402 |
Verminoside |
Natural anti-inflammatory and antioxidant agent, inhibiting both iNOS expression and NO release in the LPS-induced J774.A1 macrophage cell line, enhancing protein expression levels of PARP-1 and p53, and attenuating intracellular ROS and stress (oxidative |
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DCC5403 |
Vernakalant |
Novel blocker of atrial potassium channels |
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DCC5404 |
Vernolepin |
Natural Reversible Plant Growth Inhibitor |
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DCC5405 |
Verticilide |
Natural insect ryanodine receptor (RyR) antagonist |
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DCC5406 |
Verticillin A |
Apoptosis inducer, inhibiting Leiomyosarcoma and Malignant peripheral nerve sheath tumor growth |
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DCC5407 |
Vesamicol Hydrochloride |
Potent inhibitor of acetylcholine transport |
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DCC5408 |
Vesiculopolin B |
Novel anti-vesiculoviral agent, inhibiting transcription initiation of vesiculoviruses |
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DCC5409 |
Vezf1-in-t4 |
Novel Inhibitor of the Pro-Angiogenic Activity of the Zinc Finger Transcription Factor Vezf1 |
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DCC5410 |
Vhl-hif1α Inhibitor-tg0 |
The first sub-micromolar inhibitor of the VHL-HIF1α interaction |
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DCC5411 |
Vibsanin A |
Natural protein kinase C (PKC) activator and HSP90 inhibitor, sensitizing human acute myeloid leukemia cells to tyrosine kinase inhibitor-induced myeloid differentiation via activation of PKC and upregulation of Lyn |
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DCC5412 |
Vicagrel |
Clopidogrel analog as an antiplatelet agent |
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DCC5413 |
Vidarabine Monohydrate |
Broad spectrum antibiotic, inhibiting adenylyl cyclase type 5 (AC5) and protecting against chronic coronary artery occlusion (CAO) |
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DCC5414 |
Vilanterol |
Selective long-acting beta2-adrenergic agonist (LABA) with inherent 24-hour activity for once daily treatment of COPD and asthma |
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DCC5415 |
Vincamine V2a |
Novel antagonist against hypocretin (orexin) receptor 2, significantly preventing acute morphine-conditioned place preference (CPP) and stress-induced reinstatement of extinguished morphine-CPP in mouse models of opioid reward and relapse |
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DCC5416 |
Vincapusine |
Natural inhibitor of 3C-like protease (3CLpro), targeting SARS-CoV-2 3CLpro, SARS-CoV 3CLpro and MERS-CoV 3CLpro |
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DCC5417 |
Vincetoxicoside A |
Natural antimicrobial, antioxidant, and anti-inflammator agent |
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DCC5418 |
Virodhamine Trifluoroacetate |
Endogenous cannabinoid receptor mixed agonist/antagonist, being a full agonist at GPR55 and CB2 and partial agonist/antagonist at CB1 |
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DCC5419 |
Vitexin 4"-o-glucoside |
Natural inhibitor of ST2 (IL1RL1) |
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DCC5420 |
Viviren |
Coelenterazine analog for bioluminescence imaging (BLI) |
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DCC5421 |
Vmy-1-101 |
Fluorescent cyclin-dependent kinase inhibitor, blocking the proliferation of human breast cancer cells |
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DCC5422 |
vmy-2-95 |
Novel and selective desensitizer of |
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DCC5423 |
Setmelanotide Tfa Salt
Featured
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Novel highly-selective melanocortin-4 receptor (MC4R) agonist, increasing resting energy expenditure in obese individuals |
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DCC5424 |
Voa Analog 19 |
Novel potent VEGFR2 modulator, exhibiting increased antiangiogenic potency than voacangine against VEGF-induced VEGFR2 phosphorylation without cytotoxic effects, resulting in significant tumor cell death in a mouse xenograft model |
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DCC5425 |
Voclosporin |
Novel calcineurin inhibitor and immunosuppressive agent |
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DCC5426 |
Vonoprazan Fumurate |
Novel potassium-competitive acid blocker |
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DCC5427 |
Vpc-00628 |
Novel potent and highly selective type-II inhibitor of p38α/β, targeting an inactive state of the kinases induced by a unique folded P-loop conformation |
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DCC5428 |
Vpc-13163 |
Potent Antiandrogen, Targeting the BF3 Site of the Androgen Receptor and Inhibiting Enzalutamide-Resistant Prostate Cancer |
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