DCC5429 |
Vpc-16606 |
Novel potent and selective inhibitor of ERα-dependent cell growth and gene expression, preventing the interaction between ERα-LBD and SRC-3 fusion proteins in a dose-dependent manner |
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DCC5430 |
Vpc24191 |
S1P1/S1P3 receptor agonist |
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DCC5431 |
Vpc-3033 |
Novel Androgen Receptor Antagonist, inhibiting the LNCaP cell line as well as cell lines with wild-type androgen receptor |
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DCC5432 |
Vpc44116 |
Competitive S1P1/3 antagonist, increasing capillary permeability as measured by Evans blue dye leakage in mouse lung tissue |
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DCC5433 |
Vrt-325 |
Corrector of F508del-cystic fibrosis transmembrane conductance regulator (CFTR) mutant |
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DCC5434 |
Vrv-pl-viiia Inhibitor 5m |
Inhibitor of the catalytic activity of VRV-PL-VIIIa, strongly inhibiting the hemolysis of red blood cells and VRV-PL-VIIIa-induced myotoxicity and lung hemorrhage in mice |
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DCC5435 |
Vrx-480773 |
Novel Potent HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI) |
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DCC5436 |
Vsw1198 |
Novel inhibitor of geranylgeranyl diphosphate synthase (GGDPS) |
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DCC5437 |
Vswrapta |
Novel Promoter of Neuronal Branching Via Transcellular Activation of the Focal Adhesion Kinase (FAK) and the ERK1/2 Signaling Pathway In Vitro |
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DCC5438 |
Vt-me6 |
Sphingosine kinase (SphK) inhibitor, having modest SphK2-selectivity |
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DCC5439 |
Vtx-2337 Analog-1 |
Novel selective agonist of TLR8 |
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DCC5440 |
Vu0034403 |
Novel non-MPEP site metabotropic glutamate receptor 5 (mGlu5) positive allosteric modulators (PAMs) |
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DCC5441 |
Vu0160573 |
Selective modulator of G protein-coupled inward rectifier K (GIRK) |
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DCC5442 |
Vu0184670 |
Allosteric modulator of the M1 muscarinic receptor |
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DCC5443 |
vu0360173 |
Novel Positive Allosteric Modulator (PAM) of the Metabotropic Glutamate Receptor 5 (mGlu5) |
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DCC5444 |
Vu0361747 |
Novel Allosteric Modulator of Metabotropic Glutamate Receptor Subtype 5, Revealing Chemical and Functional Diversity and In Vivo Activity in Rat Behavioral Models of Anxiolytic and Antipsychotic Activity |
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DCC5445 |
Vu0364289 |
Potent and specific PAM for the rat mGluR5 receptor |
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DCC5446 |
Vu0366058 |
Potent noncompetitive antagonist of Metabotropic_glutamate_receptor_5>metabotropic glutamate receptor 5 (mGlu5) |
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DCC5447 |
Vu0366248
Featured
|
VU0366248 is a mGlu5 negative allosteric modulator. |
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DCC5448 |
vu0403602 |
Novel Positive Allosteric Modulator (PAM) of the Metabotropic Glutamate Receptor 5 (mGlu5) |
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DCC5449 |
Vu0404251 |
Highly potent non-MPEP site metabotropic glutamate receptor 5 (mGlu5) positive allosteric modulator (PAM) |
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DCC5450 |
Vu0409775 |
Muscarinic antagonist; inhibiting ACh-induced Ca(2+) responses at rat M(1-5) receptor subtypes |
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DCC5451 |
Vu0410150 |
Novel positive allosteric modulator (PAM) of mGlu4 |
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DCC5452 |
Vu0413144 |
Allosteric modulator of the M2/5 muscarinic acetylcholine receptor |
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DCC5453 |
vu0415248 |
Highly M1-selective antagonist |
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DCC5454 |
Vu0415371 |
Novel M4 muscarinic acetylcholine receptor modulator |
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DCC5455 |
Vu0415374 |
Novel mGlu4 positive allosteric modulator (PAM) |
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DCC5456 |
Vu0431316 |
Novel negative allosteric modulator of mGlu5 with activity in a mouse model of anxiety |
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DCC5457 |
vu0448350-1 |
Highly selective muscarinic M1 PAM |
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DCC5458 |
vu0452865 |
Selective orthosteric M1 antagonist |
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