Cat. No. | Product name | CAS No. |
DC21393 |
nNOS-IN-25
A potent, selective cell permeable neuronal nitric oxide synthase (nNOS) inhibitor with Ki of 30 nM. |
1895092-16-6 |
DC20633 |
ACG-548B
A potent, selective choline kinase α (ChoKα) inhibitor with IC50 of 0.12 uM, >400-fold selectivity over ChoKβ. |
795316-16-4 |
DC20632 |
ACG-416B
A potent, selective choline kinase α (ChoKα) inhibitor with IC50 of 0.13 uM, >385-fold selectivity over ChoKβ. |
95316-15-3 |
DC21741 |
RSM-932A
A potent, selective choline kinase α (ChoKα) inhibitor with IC50 of 1.0 uM, 33-fold selectivity over ChoKβ. |
850807-63-5 |
DC22917 |
SCH 79797 dihydrochloride
Featured
A potent, selective competitive and nonpeptide PAR-1 antagonist with IC50 of 70 nM. |
1216720-69-2 |
DC20580 |
Vitacoxib
A potent, selective COX-2 inhibitor with IC50 of 0.34 ug/mL, >50-fold selectivity over COX-1 (IC50=19.4 ug/mL). |
1374128-90-1 |
DC22418 |
CCX-771
A potent, selective CXCR7 antagonist with IC50 of 4.1 nM. |
|
DC22912 |
SCH39166
A potent, selective D1 dopamine receptor antagonist with Ki of 3.6 nM, >300-fold selectivity over D2 and 5-HT2 receptors. |
1227675-51-5 |
DC22910 |
ABT-724
A potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors. |
70006-24-5 |
DC22909 |
ABT-724 trihydrochloride
A potent, selective dopamine D4 receptor agonist that activates human dopamine D4 receptors with EC50 of 12.4 nM, with no effect on dopamine D1, D2, D3, or D5 receptors. |
587870-77-7 |
DC22586 |
AZD9496 maleate
A potent, selective estrogen receptor downregulator (SERD) with ER downregulation pIC50 of 9.68. |
1639042-28-6 |
DC20378 |
FABP4 inhibitor 1
A potent, selective FABP4 inhibitor with Ki of 30 nM.. |
1526928-21-1 |
DC11956 |
CCG 258748
A potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM. |
|
DC22881 |
GLP1-agonist-1
A potent, selective GLP-1 agonist. |
281208-76-2 |
DC20392 |
GLUT4-IN-17
A potent, selective glucose transporter 4 (GLUT4) inhibitor with IC450 of 10.8 uM, inhibits MM cell proliferation. |
1061081-61-5 |
DC22747 |
AICP
A potent, selective GluN2C-selective NMDA receptor glycine site superagonist with EC50 of 1.7 nM at GluN1/2C. |
861213-66-3 |
DC23558 |
(+)-NFPS
A potent, selective GlyT1 inhibitor that demonstrates >10-fold greater activity in in vitro functional glycine reuptake assay than racemic (±)-NFPS. |
571147-18-7 |
DC20400 |
HDAC1,2-IN-2
A potent, selective HDAC1 and HDAC2 inhibitor with IC50 of 6 nM and 45 nM, respectively. |
937727-03-2 |
DC21373 |
HDAC6 inhibitor NCT-14b
A potent, selective HDAC6 inhibitor with IC50 of 84 nM, with IC50s of >3.5 uM for the other HDAC isoforms.. |
|
DC21461 |
PD-118057
A potent, selective hERG potassium channel (Kv11.1) activator that increases peak tail hERG current of 111.1% at 10 uM in HEK293 cells. |
313674-97-4 |
DC22946 |
ML-T531
Featured
ML-T531 is a potent, selective hERG potassium channel (Kv11.1) activator with EC50 of 3.13 uM. |
791127-70-3 |
DC22990 |
HIF1-IN-2
A potent, selective HIF-1 inhibitor with IC50 of 1.9 nM, with no signigicant inhibition on HSF and NF-κB. |
159915-87-4 |