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Cat. No.	Product Name	Field of Application
DC24206	KN-93 HCl Featured	Potent, cell permeable inhibitor of CaM kinase II (IC50 = 0.37 μM).
DC7251	AM 281 Featured	Potent, selective CB1 cannabinoid receptor antagonist/inverse agonist (Ki values are 12 and 4200 nM for CB1 and CB2 receptors respectively). Increases locomotor activity following systemic administration in vivo. Analog of SR141716A (Ki = 14 nM).
DC7704	Poziotinib Featured	Poziotinib, is an orally bioavailable, quinazoline-based pan epidermal growth factor receptor (EGFR or HER) inhibitor with potential antineoplastic activity.
DC12421	PP1 inhibitor C31	PP1 inhibitor C31 is a 1E7-03 analog and protein phosphatase 1 (PP1) targeting small molecule with Kd of 1.88 uM, inhibits Ebola virus (EBOV) transcription and replication.
DC5007	pp1 Featured	PP1 is a potent and selective Src inhibitor for Lck/Fyn with IC50 of 5 nM/ 6 nM.
DC8742	PP121	PP-121 is a multi-targeted inhibitor of PDGFR, Hck, mTOR, VEGFR2, Src and Abl with IC50 of 2 nM, 8 nM, 10 nM, 12 nM, 14 nM and 18 nM, also inhibits DNA-PK with IC50 of 60 nM.
DC9931	PP2 analog Featured	PP2 analog is the analog of PP2,a Src family kinase inhibitor.
DC5008	PP2(AGL 1879) Featured	PP2 is Src family kinase inhibitor, potently inhibits Lck/Fyn with IC50 of 4 nM/5 nM, ~100-fold less potent to EGFR, inactive for ZAP-70, JAK2 and PKA.
DC7482	Torkinib (PP242) Featured	PP242 is a selective mTOR inhibitor with IC50 of 8 nM; targets both mTOR complexes with >10- and 100-fold selectivity for mTOR than PI3Kδ or PI3Kα/β/γ, respectively; also showed slightly weaker activity against BRD4 (Kd= 1.7 uM).
DC23712	PPARα activator compound 3	PPARα activator compound 3 is a specific PPAR activator that selectively up-regulates PPARα transcriptional activity, leading to PPARα target gene expression both in vitro and in vivo.
DC23517	PPBI	PPBI is a novel potent, selective, full M1 muscarinic agonist with EC50 of 5, 8, and 21 nM for human, rat, and mouse M1 receptors, respectively.
DC21525	PPI-2458	PPI-2458 is potent, specific, irreversible methionine aminopeptidase-2 (MetAP-2) inhibitor with IC50 of 0.2 nM, inhibits growth inhibition of HFLS-RA and HUVEC with IC50 of 0.04 nM.
DC7483	PPQ-102 Featured	PPQ-102 is a potent CFTR inhibitor which can completely inhibited CFTR chloride current with IC 50approximately 90 nM.
DC21943	PPTN trifluoroacetate salt	PPTN is a potent, highly specific amtagonist of P2Y14 receptor with Ki of 0.4 nM in functional assays.
DC21942	PPTN	PPTN is a potent, highly specific amtagonist of P2Y14 receptor with Ki of 0.4 nM in functional assays.
DC22059	PptT inhibitor 8918	PptT inhibitor 8918 (Compound 8918) is a mycobactericidal amidino-urea compound that targets phosphopantetheinyl transferase (PptT, IC50=2.5 uM), shows an MIC90 of 3.1 uM against Mtb H37Rv.
DC2083	PQ401 Featured	PQ 401 is an IGF-1R inhibitor with IC50 of <1 μM.
DC23868	PQC 083	PQC 083 is a novel nerve growth factor (NGF) antagonist with IC50 of 7.0 uM, functionally inhibits NGF's effects on PC12 cell differentiation.
DC10767	PQR530 Featured	PQR530 is a selective, orally bioavailable, potent dual PI3K/mTORC1/2 inhibitor.
DC20221	PQR620 Featured	PQR620 is a novel potent and selective brain penetrant inhibitor of mTORC1/2.
DC20510	PR5-LL-CM01	PR5-LL-CM01 is a novel selective, small-molecule inhibitor of PRMT5 methyltransferase with IC50 of 7.5 uM.
DC7252	PR-619 Featured	PR-619 is a broad-range DUB inhibitor with potential for further development as a chemotherapeutic agent in cancer therapy.
DC7280	Pracinostat(SB939) Featured	Pracinostat(SB939) is a potent pan-HDAC inhibitor with IC50 of 40-140 nM with exception for HDAC6; has no activity against the class III isoenzyme SIRT I.
DC12202	Pradefovir mesylate (Remofovir mesylate) Featured	Pradefovir mesylate is a good substrate for liver CYP3A4. Pradefovir is converted to 9-(2-phosphonylmethoxyethyl)adenine (PMEA) in human liver microsomes with a Km of 60 μM.
DC9359	Pralatrexate Featured	Pralatrexate(Folotyn) is an antifolate, and structurally a folate analog.
DC11526	Praliciguat Featured	Praliciguat (IW-1973, IW1973) is a potent, orally available sGC stimulator that concentration-dependently increases the production of cGMP with EC50 of 267 nM.
DC10263	Pralidoxime (chloride)	Pralidoxime is an antidote to organophosphate pesticides and chemicals.
DC8970	Pramipexole Base	Pramipexole is a dopamine agonist of the non-ergoline class indicated for treating Parkinson's disease (PD) and restless legs syndrome (RLS).
DC3151	Pramipexole dihydrochloride	Pramipexole is a partial/full D2S, D2L, D3, D4, receptor agonist with a Ki of 3.9, 2.2, 0.5, 5.1 nM.
DCAPI1305	Pramiracetam	Pramiracetam

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