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Cat. No.	Product Name	Field of Application
DC7206	R1530 Featured	R1530 is the multikinase inhibitor with potential antiangiogenesis and antineoplastic activities.
DC11138	Guanabenz acetate	R15A inhibitor.
DC10692	R162 Featured	R162 is an inhibitor of GDH activity and represses glioma cell growth.
DC22205	R191	R191 (R-191) is a potent, small molecule IRAK1/4 kinase inhibitor (IRAK4 IC50=3 nM), exhibits good selectivity against a broad panel of kinases.
DC22670	R243 Featured	R243 is a potent, small molecule CCR8 antagonist that inhibits CCR8 signaling and chemotaxis, inhibits CCL1-induced Ca2+ flux and CCL1-driven peritoneal macrophages aggregation at 0.2 uM.
DC7037	R306465(JNJ-16241199) Featured	R306465, also known as JNJ-16241199, is a novel hydroxamate-based histone deacetylase (HDAC) inhibitor with broad-spectrum antitumour activity against solid and haematological malignancies in preclinical models.
DC21551	R-360163	R-360163 is a small molecule inhibitor that effectively inhibits the β-catenin/Tcf4 interaction with Ki of 16 uM in FP assay.
DC1014	R406 free base Featured	R406 is a potent Syk inhibitor with IC50 of 41 nM and also potently inhibits Flt3.
DC8733	R406 Featured	R406 is a potent Syk inhibitor with IC50 of 41 nM and also potently inhibits Flt3.
DC7258	Bemcentinib（R428，BGB324) Featured	R428 is a potent and selective small-molecule inhibitor(IC50=14 nM), blocks the activities of Axl.
DC2068	R547	R547 is a potent and selective CDK inhibitor with Ki and IC50 of 1-3 nM and 80 nM respectively.
DC10897	R-7050 Featured	R-7050 is a tumor necrosis factor receptor (TNFR) antagonist with greater selectivity toward TNFα.
DC9462	R-7128(Mericitabine) Featured	R-7128(Mericitabine) is a selective nucleoside analog inhibitor of the hepatitis C virus (HCV) NS5B RNA-dependent RNA polymerase, with activity across all HCV genotypes.
DC9841	Fostamatinib(R788) Featured	R788 (Fostamatinib), a prodrug of the active metabolite R406, is a potent Syk inhibitor with IC50 of 41 nM.
DC10995	R916562	R916562 (R562) is a potent, dual Axl/VEGF-R2 inhibitor with celluar IC50 of 136 nM for Axl.
DC1013	R788 disodium (Fostamatinib) Featured	R935788 (Fostamatinib disodium, R788) is a Syk inhibitor with IC50 of 41 nM.
DC21555	R-999636	R-999636 is a small molecule inhibitor that effectively inhibits the β-catenin/Tcf4 interaction with Ki of 8.8 uM in FP assay.
DC10304	RA190 Featured	RA190, a bis-benzylidine piperidon, inhibits proteasome function by covalently binding to cysteine 88 of ubiquitin receptor RPN13.
DC9103	Rebeprazole sodium	Rabeprazole sodium(LY307640 sodium) is an antiulcer drug in the class of proton pump inhibitors.
DC10578	rac BHFF Featured	Rac BHFF is a potent and selective GABAB receptor positive allosteric modulator that increases the efficacy and potency of GABA ( > 149% and > 15-fold respectively). Orally active and exhibits anxiolytic activity in vivo.
DC21544	rac Pterosin B	rac Pterosin B is a potent and specific SIK3 signaling inhibitor that suppresses SIK3 downstream cascades by up-regulating the phosphorylation levels in the SIK3 C-terminal regulatory domain.
DC9107	Racecadotril Featured	Racecadotril (acetorphan), a potent enkephalinase inhibitor (IC50= 4.5 uM), protects endogenous enkephalins from degradation.
DC9657	RAD140 Featured	RAD140 is a potent, orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM).
DC20528	RAD51-IN-1 Featured	RAD51-IN-17 is a quinazolinone derivative that inhibts homologous recombinase RAD51, effectively inhibits both RAD51 foci formation in response to DNA damage, and proliferation of TNBC cell lines.
DC9513	Radafaxine (hydrochloride) Featured	Radafaxine Hcl(BW-306U; GW-353162A) is a potent metabolite of bupropion; selective for inhibiting the reuptake of norepinephrine over dopamine; DAT (dopamine transporter) and NET(norepinephrine transporter) transporters inhibitor, and nAChR family modulat
DC21069	Radalbuvir	Radalbuvir (GS-9669) is a highly optimized thumb site II nonnucleoside inhibitor of HCV NS5B polymerase with binding affinity of 1.35 nM for genotype 1b.
DC9351	Radezolid Featured	Radezolid (RX-1741) is a novel oxazolidinone antibiotic agent.
DC12701	Radiprodil Featured	Radiprodil is an orally active and selective NMDA NR2B antagonist; a potential therapeutic agent in treatment of neuropathic pain and possibly other chronic pain conditions.
DC8011	Radotinib (IY-5511) Featured	Radotinib(IY-5511) is a novel and selective BCR-ABL1 tyrosine kinase inhibitor with IC50 of 34 nM for wild-type BCR-ABL1 kinase.
DC5049	RAF265 (CHIR-265) Featured	RAF265 (CHIR-265) is a highly selective B-Raf and VEGFR2 inhibitor with IC50 of 3-60 nM and EC50 of 30 nM, including B-Raf, C-Raf and mutant B-Raf.

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