CCG-4986|CCG 4986;CCG4986

Cas No.:	7134-19-2
Chemical Name:	Methyl-N-[(4-chlorophenyl)sulfonyl]-4-nitrobenzenesulfinimidoate
Synonyms:	CCG 4986;CCG4986
SMILES:	C(S(=NS(C1=CC=C(Cl)C=C1)(=O)=O)OC)1=CC=C([N+]([O-])=O)C=C1
Formula:	C₁₃H₁₁ClN₂O₅S₂
M.Wt:	374.81
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

A non-peptide, selective RGS4 inhibitor that inhibits RGS4/Gα(o) binding with 3 to 5 uM potency; shows selectivity for RGS4 and does not inhibit RGS8; binds to RGS4, inhibits RGS4 stimulation of Galpha(o) GTPase activity in vitro, and prevents RGS4 regulation of mu-opioid-inhibited adenylyl cyclase activity in permeabilized cells.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

Cat. No.	Product name	Field of application
DC9613	CCG-63808	CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins.
DC9612	CCG-63802	CCG-63802 is a reversible inhibitor of regulator of G-protein signaling (RGS) protein; with greatest potency at RGS4. IC50 value: Target: RGS CCG-63802 is selective amongst RGS proteins, with greatest potency at RGS4.
DC11662	CCG-4986	A non-peptide, selective RGS4 inhibitor that inhibits RGS4/Gα(o) binding with 3 to 5 uM potency.