DX 600(ACE2 Inhibitor)

  Cat. No.:  DC26232   Featured
Chemical Structure
478188-26-0
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More than 5000 active chemicals with high quality for research!
Field of application
DX600 is a potent and selective peptide inhibitor of angiotensin-converting enzyme 2 (ACE2; Kis = 2.8, 200, and 1,200 nM for recombinant, human, and murine ACE2, respectively).
Cas No.: 478188-26-0
Chemical Name: DX 600
Synonyms: ac-gly-asp-tyr-ser-his-cys-ser-pro-leu-arg-tyr-tyr-pro-trp-trp-lys-cys-thr-tyr-pro-asp-pro-glu-gly-gly-gly-nh2, (disulfide bond) trifluoroacetate;Ac-Gly-Asp-Tyr-Ser-His-Cys-Ser-Pro-Leu-Arg-Tyr-Tyr-Pro-Trp-Trp-Lys-Cys-Thr-Tyr-Pro-Asp-Pro-Glu-Gly-Gly-Gly-NH?;Ac-Gly-Asp-Tyr-Ser-His-Cys-Ser-Pro-Leu-Arg-Tyr-Tyr-Pro-Trp-Trp-Lys-Cys-Thr-Tyr-Pro-Asp-Pro-Glu-Gly-Gly-Gly-NH₂;DX-600;DX 600
SMILES: C([C@H]1C(N[C@H](C(N[C@H](C(N[C@@H](CSSC[C@@H](C(N[C@H](C(N2CCC[C@@]2([H])C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N2CCC[C@@]2([H])C(N1)=O)=O)CC1C=CC(=CC=1)O)=O)CC1C=CC(=CC=1)O)=O)CCCNC(N)=N)=O)CC(C)C)=O)=O)CO)=O)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)NC(=O)CNC(=O)C)CC1C=CC(=CC=1)O)CC1NC=NC=1)C(=O)N[C@@H]([C@H](O)C)C(=O)N[C@@H](CC1C=CC(=CC=1)O)C(N1CCC[C@H]1C(=O)N[C@@H](CC(=O)O)C(N1CCC[C@H]1C(=O)N[C@@H](CCC(=O)O)C(=O)NCC(=O)NCC(=O)NCC(=O)N)=O)=O)=O)CCCCN)=O)CC1=CNC2=CC=CC=C12)=O)C1=CNC2=CC=CC=C12
Formula: C141H185N35O40S2
M.Wt: 3074.32
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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