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EST73502

  Cat. No.:  DC42314   Featured
Chemical Structure
1838622-25-5
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Field of application
EST73502 is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 has antinociceptive activity.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1838622-25-5
Chemical Name: (2R)-9-[2-(2,5-Difluorophenyl)ethyl]-4-ethyl-2-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
Synonyms: EST73502;FC1=C(CCN2CCC3(CN(C([C@H](O3)C)=O)CC)CC2)C=C(C=C1)F;(2R)-9-[2-(2,5-Difluorophenyl)ethyl]-4-ethyl-2-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
SMILES: FC1C([H])=C([H])C(=C([H])C=1C([H])([H])C([H])([H])N1C([H])([H])C([H])([H])C2(C([H])([H])N(C([H])([H])C([H])([H])[H])C([C@@]([H])(C([H])([H])[H])O2)=O)C([H])([H])C1([H])[H])F
Formula: C19H26F2N2O2
M.Wt: 352.4188
Purity: >98%
Sotrage: Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS
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MSDS_25921_DC42314_1838622-25-5
COA
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Cat. No. Product name Field of application
DC48169 DS34942424 DS34942424 is an orally potent analgesic without mu opioid receptor agonist activity.
DC42314 EST73502 EST73502 is a selective, orally active and blood-brain barrier (BBB) penetrant dual μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, with Kis of 64 nM and 118 nM for MOR and σ1R, respectively. EST73502 has antinociceptive activity.
DC8626 Eluxadoline Eluxadoline is an orally active mixed μ opioid receptor (μOR) agonist δ opioid receptor (δOR) antagonist.
DC9765 CERC-501(LY-2456302,Aticaprant) CERC-501(LY-2456302) is a potent, selective antagonist of the kappa opioid receptor (KOR) (Ki = 0.81 nM vs. 24.0 nM and 155 nM for the μ-opioid receptor (MOR) and δ-opioid receptor (DOR), respectively.
DC7097 Cebranopadol(GRT-6005) branopadol(GRT-6005) is a novel first in class compounds with potent agonist activity on ORL-1 (opioid receptor like -1) and the well established mu opioid receptor.
DC8298 BAN ORL 24 BAN ORL 24 is a potent, selective, competitive ORL1 non-peptide agonist. Displays 1000-fold selectivity over classical opioid receptors.
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