Cat. No. | Product name | CAS No. |
DCAPI1349 |
Simvastatin (Zocor)
Featured
Simvastatin (MK 733) is a competitive inhibitor of HMG-CoA reductase with a Ki of 0.2 nM. |
79902-63-9 |
DC4108 |
Sitaxentan sodium
Featured
Sitaxentan sodium (TBC-11251) is a selective endothelin receptor-A antagonist with IC50 and Ki of 1.4 nM and 0.43 nM, respectively. |
210421-74-2 |
DC10386 |
Tenapanor
Featured
Tenapanor is an inhibitor of the Na+/H+ exchanger NHE3 with IC50 values of 5 and 10 nM against human and Rat NHE3, respectively. |
1234423-95-0 |
DC9609 |
Terutroban
Featured
Terutroban is a thromboxane/prostaglandin endoperoxide receptor antagonist. |
165538-40-9 |
DC1101 |
Ticagrelor (Brilinta,AZD6140)
Featured
Ticagrelor is the first reversibly binding oral P2Y12 receptor antagonist, also inhibits CYP2C9 and 4-hydroxylation with IC50 of 10.5 μM and 8.2 μM respectively. |
274693-27-5 |
DC9489 |
Tirofiban (hydrochloride monohydrate)
Featured
Tirofiban hydrochloride monohydrate is a potent non-peptide, glycoprotein IIb/IIIa (integrins alphaIIbbetaIII) antagonist |
150915-40-5 |
DC7327 |
Tirofiban(L700462;MK383)
Featured
Tirofiban(L700462;MK383) is a potent non-peptide, glycoprotein IIb/IIIa (integrins alphaIIbbetaIII) antagonist. |
144494-65-5 |
DC7519 |
Torcetrapib
Featured
Torcetrapib is a CETP inhibitor with IC50 of 37 nM, elevates HDL-C and reduces nonHDL-C in plasma. Phase 3. |
262352-17-0 |
DCAPI1452 |
Valsartan
Valsartan is a nonpeptide angiotensin II AT1-receptor antagonist with an IC50 ranging from 39.5 to 116 μM. This in turn causes blood vessel dilation. |
137862-53-4 |
DC8916 |
Vanoxerine dihydrochloride
Featured
Vanoxerine 2 Hcl(GBR12909) is a potent and selective DRI (Dopamine reuptake inhibitor). |
67469-78-7 |
DC7699 |
VTP-27999
Featured
VTP-27999 is an alkyl amine Renin inhibitor; VTP-27999 is useful for Hypertension and End-Organ Diseases. |
942142-51-0 |
DC7040 |
WAY-362450 (XL335; Turofexorate isopropyl)
Featured
WAY-362450 (XL335; Turofexorate isopropyl) is a highly potent, selective, and orally active farnesoid X receptor (FXR) agonist with an EC50 of 4 nM.WAY-362450 is useful for dyslipidemia. |
629664-81-9 |
DC7753 |
Zatebradine hydrochloride
Zatebradine hydrochloride is a bradycardic agent that creates use-dependent inhibition of hyperpolarization-activated current (If) in sinoatrial node cells (EC50 = 480 nM) and Purkinje fibres. |
91940-87-3 |
DC9461 |
Zatebradine
Zatebradine(UL-FS49) is a potent HCN channels antagonist, which decreased the heartbeat in a reversible manner; 92% inhibition of the hHCN1-mediated current at 10 uM. |
85175-67-3 |
DC9113 | Ketanserin | 74050-98-9 |
DC9178 | Ketanserin Tartrate | 83846-83-7 |
DC8860 |
Vorapaxar
Featured
Vorapaxar (SCH 530348) is a potent and orally active thrombin receptor (PAR-1) antagonist with Ki of 8.1 nM. |
618385-01-6 |
DC8901 |
Azilsartan medoxomil
Featured
Azilsartan medoxomil(TAK 491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. |
863031-21-4 |