Cat. No. | Product name | CAS No. |
DC12456 |
BTT-266
Featured
BTT-266 (BTT266) is a voltage-gated CaV2.2 calcium channel inhibitor that disrupts the CaVα·CaVβ3 protein-protein interaction, directly binds to CaVβ3 with Kd of 3.6 uM. |
2413939-89-4 |
DC23703 |
BTYNB
Featured
BTYNB is a potent and selective inhibitor of IMP1 binding to c-Myc mRNA with IC50 of 5 uM. |
304456-62-0 |
DC9704 |
Unii-G55ZH52P57
Featured
BTZ043 is a inhibitor of decaprenyl-phosphoribose-epimerase (DprE1), It can display nanomolar bactericidal activity against Mycobacterium tuberculosis in vitro. |
1161233-85-7 |
DCAPI1392 |
BTZ043 racemate
Featured
BTZ043 racemate is a decaprenylphosphoryl-β-D-ribose 2-epimerase (DprE1) inhibitor acting as a new antimycobacterial agent that kill Mycobacterium tuberculosis. |
957217-65-1 |
DC22041 |
BTZO-1
Featured
BTZO-1 is a cardioprotective agent and Macrophage migration inhibitory factor (MIF) activator, binds to MIF with Kd of 68.6 nM, regulates ARE-mediated gene expression. |
99420-15-2 |
DC6501 |
Bufalin
Featured
Bufalin inhibits steroid receptor coactivator 1 (SRC-1) and SRC-3 at doses as low as 5 nM, promotes the degradation of SRC-3 protein, and inhibits cancer cell growth both in vitro and in vivo. |
465-21-4 |
DCAPI1140 |
Bumetanide
Featured
Bumetanide |
28395-03-1 |
DC11381 |
Butabindide (oxalate)
Featured
Butabindide is a potent inhibitor of cholecystokinin-inactivating peptidase/tripeptidyl peptidase 2 (CCK-inactivating peptidase/TPP-2; Ki = 7 nM).1 It is selective for CCK-inactivating peptidase/TPP-2 over a panel of serine proteases (Kis = >1 μM) as well as CCK receptors (Kis = >0.1 mM). |
185213-03-0 |
DC10693 |
O-Butyryl timolol
Featured
Butyryltimolol is a lipophilic ester prodrug of timolol, a beta adrenergic blocer with antihypertensive and hemodynamic properties. |
106351-79-5 |
DC7563 |
BV6
Featured
BV6 induced apoptotic and necrotic cell death in monocytes while T-cells, dendritic cells and macrophages were largely protected against BV6-induced cell death. |
1001600-56-1 |
DC8089 |
BVT 2733(BVT.2733)
Featured
BVT 2733 is a selective 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor,protecting osteoblasts against endogenous glucocorticoid induced dysfunction. |
376640-41-4 |
DC8278 |
BVT-14225
Featured
BVT 14225 is a new selective 11b-HSD1 inhibitor, it belongs to a class of arylsulfonamidothiazoles with in vitro and in vivo antidiabetic effects |
376638-65-2 |
DC21685 |
BVT-948
Featured
BVT-948 (SPS8I-3) is a noncompetitive, cell-permeable inhibitor of protein tyrosine phosphatases (PTPs) with IC50 of 0.09-1.7 uM. Results show that the effect of BVT948 (BVT.948) is to strengthen the insulin signal and has no effects on the duration of th |
39674-97-0 |
DC12041 |
BW-A 78U
Featured
BW-A 78U is a PDE4 inhibitor with an IC50 of 3 μM. |
101155-02-6 |
DC7675 |
BX-471(ZK 811752)
Featured
BX471 is a potent, selective non-peptide CCR1 antagonist (Ki = 1 nM for human CCR1); exhibits 250-fold selectivity for CCR1 over CCR2, CCR5 and CXCR4. |
217645-70-0 |
DC8808 |
BX-513 hydrochloride
Featured
BX-513 hydrochloride inhibits MIP-1α-induced intracellular calcium mobilization (IC50 = 2.5 μM). |
193542-65-3 |
DC8062 |
BX517
Featured
BX517 is a novel phosphoinositide-dependent kinase-1 (PDK1) inhibitor. |
850717-64-5 |
DC7092 |
BX795
Featured
BX795 is a potent and selective dual inhibitor of TBK1/PDK1 with IC50s of 2 nM/6 nM respectively; > 50 fold selectivity over PKA, PKC, c-Kit, GSK3β etc. |
702675-74-9 |
DC7093 |
BX912
Featured
BX-912 is a selective inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1) with IC50 of 12 nM; >10 fold selectivity over PKA, PKC, C-Kit, EGFR etc. |
702674-56-4 |
DC11219 |
BXI-72
Featured
BXI-72 (NSC334072) is a potent, selective small molecule Bcl-XL inhibitor that targets the BH3 domain of Bcl-XL (Kd=0.9 nM). |
23491-45-4 |
DC7094 |
Alpelisib(BYL-719)
Featured
BYL719 is a potent and selective PI3Kα inhibitor with IC50 of 5 nM, ;liitle or no effect on PI3Kβ/γ/δ. |
1217486-61-7 |
DC26049 |
Bz-IEGR-pNA (acetate)
Featured
Bz-IEGR-pNA is a colorimetric substrate for Factor Xa. |
1325307-57-0 |