Cat. No. | Product name | CAS No. |
DC11453 |
Bz-Nle-Lys-Arg-Arg-AMC
Featured
Bz-Nle-Lys-Arg-Arg-AMC is a substrate for dengue virus NS2B-NS3 and yellow fever virus NS3 protease. |
863975-32-0 |
DC10864 |
C188-9
Featured
C188-9 is a potent inhibitor of STAT3 that binds to STAT3 with high affinity (KD=4.7±0.4 nM). C188-9 is well tolerated in mice, shows good oral bioavailability, and is concentrated in tumors. |
432001-19-9 |
DC10937 |
C25-140
Featured
C25-140 is a specific, first-in-class small molecule inhibitor of the TRAF6-Ubc13 interaction, binds TRAF6, inhibits TRAF6-Ubc13 interaction and TRAF6 activity. |
1358099-18-9 |
DC10276 |
C29
Featured
C29 is a potential TLR2 inhibitor. |
363600-92-4 |
DC7658 |
C646
Featured
C646 is an inhibitor for histone acetyltransferase, and inhibits p300 with a Ki of 400 nM. Preferentially selective for p300 versus other acetyltransferases. |
328968-36-1 |
DC9528 |
C75 (trans)
Featured
C75 trans is the trans form of C75; C75 is a potent fatty-acid synthase(FASN) inhibitor with IC50 of 35.4 μM(LNCaP cell Proliferation inhibition). |
191282-48-1 |
DC7697 |
CA-074-Me
Featured
CA-074 Me is a selective and cell-permeable inhibitor of cathepsin B. |
147859-80-1 |
DC10330 |
PD-1-IN-17
Featured
PD-1-IN-17 has CAS#CAS:1673560-66-1, which is a programmed cell death-1 (PD-1) inhibitor. PD-1-IN-17 was first reported in patent WO2015033301A1, (Compound 4), inhibits 92% splenocyte proliferation at 100 nM. PD-1-IN-17 may be related to CA-170 (AUPM170), which is a potent PD-1 inhibitor and curreently under clinical trials. |
1673560-66-1 |
DC10648 |
CA4948-Analog
Featured
CA4948-Analog is an analog of Emavusertib. It has similar property to CA-4948, which is a potent, and orally active interleukin-1 receptor-associated kinase 4 (IRAK4) inhibitor. It was reported in patent WO 2015104688. Emavusertib, also known as CA-4948 i |
1801343-74-7 |
DC12044 |
CA-5f
Featured
CA-5f is a novel late-stage autophagy inhibitor with potent anti-tumor effect against non-small cell lung cancer. |
1370032-19-1 |
DC26013 |
Cabotegravir Sodium
Featured
Cabotegravir is a potent HIV integrase inhibitor as an oral lead-in tablet and long-acting injectable for the treatment and prevention of HIV infection. |
1051375-13-3 |
DC8180 |
Cabotegravir(GSK744)
Featured
Cabotegravir is a potent HIV integrase inhibitor as an oral lead-in tablet and long-acting injectable for the treatment and prevention of HIV infection. |
1051375-10-0 |
DC9266 |
Cabozantinib S-malate
Featured
Cabozantinib S-malate (XL184, BMS-907351) is a potent VEGFR2 inhibitor with IC50 of 0.035 nM and also inhibits c-Met, Ret, Kit, Flt-1/3/4, Tie2, and AXL with IC50 of 1.3 nM, 4 nM, 4.6 nM, 12 nM/11.3 nM/6 nM, 14.3 nM and 7 nM, respectively. |
1140909-48-3 |
DC10736 |
CaCC(inh)-A01
Featured
CaCC(inh)-A01 is a non-selective inhibitor of calcium-activated chloride channels (CaCCs) that blocks ATP-stimulated chloride conductance in human salivary gland, intestinal, and bronchial epithelium (mean IC50 = 10 µM). |
407587-33-1 |
DC20856 |
CAD-031
Featured
CAD-031 (CAD31) is a novel brain penetrant, J147-derivative that has enhanced neurogenic activity over J147 in human neural precursor cells (NPCs). |
2071209-49-7 |
DC10457 |
Cadazolid (ACT-179811)
Featured
Cadazolid (ACT-179811) is a novel fluoroquinolone-oxazolidinone antibiotic and a protein synthesis inhibitor. |
1025097-10-2 |
DC5068 |
Idelalisib (CAL-101,GS-1101)
Featured
CAL-101 is a selective p110δ inhibitor with IC50 of 2.5 nM; shown to have 40- to 300-fold greater selectivity for p110δ thanp110α/β/γ, and 400- to 4000-fold more selectivity to p110δ than C2β, hVPS34, DNA-PK and mTOR. |
870281-82-6 |
DCAPI1559 |
Calcifediol
Featured
Calcifediol is a major circulating metabolite of vitamin D3, acting as a competitive inhibitor with an apparent Ki of 3.9 μM, suppresses PTH secretion and mRNA (ED50=2 nM). |
19356-17-3 |
DCAPI1415 |
Calcipotriol(Calcipotriene)
Featured
Calcipotriol is a synthetic VitD3 analogue with a high affinity for the vitamin D receptor. |
112965-21-6 |
DC10327 |
Calcitonin salmon
Featured
Calcitonin, Salmon is a calcium regulating hormone secreted from mammalian thyroid parafollicular cells and in non-mammalian species from the ultimobranchial gland. |
47931-85-1 |
DCAPI1150 |
Calcitriol (Rocaltrol)
Featured
Calcitriol is the most active metabolite of vitamin D and also a vitamin D receptor (VDR) agonist. |
32222-06-3 |
DC20857 |
Calhex-231
Featured
Calhex-231 is a potent negative allosteric modulator of CaSR that blocks calcium-mediated activation with IC50 of 0.39 uM. |
652973-93-8 |