Cat. No. | Product name | CAS No. |
DC7568 |
Z-DEVD-FMK
Featured
Cell-permeable, irreversible inhibitor of caspase-3/CPP32; inhibits tumor cell apoptosis. Neuroprotective in rat hippocampus following seizures in vivo. |
210344-95-9 |
DC9923 |
CeMMEC1
Featured
CeMMEC1 is a novel potent inhibitor of the second bromodomain of TAF1, binding neither the first nor the second bromodomain of BRD4. |
440662-09-9 |
DC10316 |
Cenicriviroc
Featured
Cenicriviroc is an orally active, dual CCR2/CCR5 antagonist, and displays potent anti-inflammatory and aninfective activity. |
497223-25-3 |
DC10010 |
Centrinone
Featured
Centrinone is a selective and reversible inhibitor of polo-like kinase 4 (Plk4), a serine-threonine protein kinase that initiates centriole/centrosome assembly. |
1798871-30-3 |
DC8138 |
CEP-28122
Featured
CEP-28122 is a highly potent and selective orally active inhibitor of anaplastic lymphoma kinase with antitumor activity in experimental models of human cancers. |
1022958-60-6 |
DC8196 |
CEP-32496
Featured
CEP-32496 is a highly potent inhibitor of BRAF(V600E/WT) and c-Raf with Kd of 14 nM/36 nM and 39 nM, also potent to Abl-1, c-Kit, Ret, PDGFRβ and VEGFR2, respectively; insignificant affinity for MEK-1, MEK-2, ERK-1 and ERK-2. |
1188910-76-0 |
DC7099 |
CEP33779
Featured
CEP33779(< 3 μM) inhibits phosphorylation of downstream target signal transducer and activator of transcription 5(pSTAT5) of JAK2 in a concentration dependent manner in HEL92 cells. |
1257704-57-6 |
DC8009 |
CEP-37440
Featured
CEP-37440 is a novel potent and selective Dual FAK/ALK inhibitor with IC50 s of 2.3 nM (FAK) and 120 nM(ALK cellular IC50 in 75% human plasma). |
1391712-60-9 |
DC10337 |
CEP-40783
Featured
CEP-40783 is a potent, selective and orally available inhibitor of AXL and c-Met with IC50 values of 7 nM and 12 nM, respectively. |
1437321-24-8 |
DC7347 |
Cephalosporin C Na salt
Featured
Cephalosporin C Na salt is used to study the effect of transpeptidase expression, binding, and inhibition on bacterial cell wall mucopeptide synthesis. |
74970-31-3 |
DC7346 |
Cephalosporin C zinc salt
Featured
Cephalosporin C zinc salt is used to study the effect of transpeptidase expression, binding, and inhibition on bacterial cell wall mucopeptide synthesis. |
59143-60-1 |
DC9649 |
Cephalotaxlen
Featured
Cephalotaxine is an antiviral as well as antitumor agent. |
24316-19-6 |
DC9765 |
CERC-501(LY-2456302,Aticaprant)
Featured
CERC-501(LY-2456302) is a potent, selective antagonist of the kappa opioid receptor (KOR) (Ki = 0.81 nM vs. 24.0 nM and 155 nM for the μ-opioid receptor (MOR) and δ-opioid receptor (DOR), respectively. |
1174130-61-0 |
DC7814 |
Cerdulatinib(PRT-062070; PRT2070)
Featured
Cerdulatinib(PRT-062070; PRT2070) is an novel oral dual Syk/JAK inhibitor. |
1198300-79-6 |
DC9500 |
Cevimeline (hydrochloride hemihydrate)
Featured
Cevimeline hydrochloride hemihydrate, a novel muscarinic receptor agonist, is a candidate therapeutic drug for xerostomia in Sjogren's syndrome. |
153504-70-2 |
DC10440 |
Namodenoson (CF-102)
Featured
CF-102(2-Cl-IB-MECA) is a selective A3 adenosine receptor agonist (Ki = 0.33 nM). Displays 2500- and 1400-fold selectivity over A1 and A2A receptors respectively. target: A3 adenosine receptor agonist; |
163042-96-4 |
DC10069 |
CFI-400437
Featured
CFI-400437 is potent against PLK4 (IC50 = 0.6 nM) and selective against other members of the PLK family (>10 uM). |
1247000-76-5 |
DC22809 |
c-FMS-IN-8
Featured
c-FMS-IN-8 is a potent, selective c-FMS kinase inhibitor with IC50 of 0.8 nM, shows activity in collagen-induced model of arthritis in mice.. |
885704-21-2 |
DC7039 |
CFTR Inhibitor II
Featured
CFTR Inhibitor II is a cell-permeable glycinyl hydrazone compound that acts as a potent, selective and reversible open-channel blocker of CFTR with intermediate speed (< 1 min; 95% inhibition at 50 µM; Ki = 4.3 µM in CFTR-expressing FRT cells. |
328541-79-3 |
DC12580 |
CG-806
Featured
CG-806 (CG806, CG'806) is a novel potent, pan-FLT3/BTK multi-kinase inhibitor with impressive inhibition of leukemic cell proliferation with IC50 at sub-nanomolar or low nanomolar levels. |
1370466-81-1 |
DC7380 |
CGI-1746
Featured
CGI1746 is a small-molecule Btk inhibitor chemotype with a new binding mode that stabilizes an inactive nonphosphorylated enzyme conformation. |
910232-84-7 |
DC7101 |
CGK733
Featured
CGK 733 is a potent and selective inhibitor of ATM/ATR with IC50 of ~200 nM. |
905973-89-9 |