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Cat. No. Product name CAS No.
DC7568 Z-DEVD-FMK Featured

Cell-permeable, irreversible inhibitor of caspase-3/CPP32; inhibits tumor cell apoptosis. Neuroprotective in rat hippocampus following seizures in vivo.

210344-95-9
DC9923 CeMMEC1 Featured

CeMMEC1 is a novel potent inhibitor of the second bromodomain of TAF1, binding neither the first nor the second bromodomain of BRD4.

440662-09-9
DC10316 Cenicriviroc Featured

Cenicriviroc is an orally active, dual CCR2/CCR5 antagonist, and displays potent anti-inflammatory and aninfective activity.

497223-25-3
DC10010 Centrinone Featured

Centrinone is a selective and reversible inhibitor of polo-like kinase 4 (Plk4), a serine-threonine protein kinase that initiates centriole/centrosome assembly.

1798871-30-3
DC8138 CEP-28122 Featured

CEP-28122 is a highly potent and selective orally active inhibitor of anaplastic lymphoma kinase with antitumor activity in experimental models of human cancers.

1022958-60-6
DC8196 CEP-32496 Featured

CEP-32496 is a highly potent inhibitor of BRAF(V600E/WT) and c-Raf with Kd of 14 nM/36 nM and 39 nM, also potent to Abl-1, c-Kit, Ret, PDGFRβ and VEGFR2, respectively; insignificant affinity for MEK-1, MEK-2, ERK-1 and ERK-2.

1188910-76-0
DC7099 CEP33779 Featured

CEP33779(< 3 μM) inhibits phosphorylation of downstream target signal transducer and activator of transcription 5(pSTAT5) of JAK2 in a concentration dependent manner in HEL92 cells.

1257704-57-6
DC8009 CEP-37440 Featured

CEP-37440 is a novel potent and selective Dual FAK/ALK inhibitor with IC50 s of 2.3 nM (FAK) and 120 nM(ALK cellular IC50 in 75% human plasma).

1391712-60-9
DC10337 CEP-40783 Featured

CEP-40783 is a potent, selective and orally available inhibitor of AXL and c-Met with IC50 values of 7 nM and 12 nM, respectively.

1437321-24-8
DC7347 Cephalosporin C Na salt Featured

Cephalosporin C Na salt is used to study the effect of transpeptidase expression, binding, and inhibition on bacterial cell wall mucopeptide synthesis.

74970-31-3
DC7346 Cephalosporin C zinc salt Featured

Cephalosporin C zinc salt is used to study the effect of transpeptidase expression, binding, and inhibition on bacterial cell wall mucopeptide synthesis.

59143-60-1
DC9649 Cephalotaxlen Featured

Cephalotaxine is an antiviral as well as antitumor agent.

24316-19-6
DC9765 CERC-501(LY-2456302,Aticaprant) Featured

CERC-501(LY-2456302) is a potent, selective antagonist of the kappa opioid receptor (KOR) (Ki = 0.81 nM vs. 24.0 nM and 155 nM for the μ-opioid receptor (MOR) and δ-opioid receptor (DOR), respectively.

1174130-61-0
DC7814 Cerdulatinib(PRT-062070; PRT2070) Featured

Cerdulatinib(PRT-062070; PRT2070) is an novel oral dual Syk/JAK inhibitor.

1198300-79-6
DC9500 Cevimeline (hydrochloride hemihydrate) Featured

Cevimeline hydrochloride hemihydrate, a novel muscarinic receptor agonist, is a candidate therapeutic drug for xerostomia in Sjogren's syndrome.

153504-70-2
DC10440 Namodenoson (CF-102) Featured

CF-102(2-Cl-IB-MECA) is a selective A3 adenosine receptor agonist (Ki = 0.33 nM). Displays 2500- and 1400-fold selectivity over A1 and A2A receptors respectively. target: A3 adenosine receptor agonist;

163042-96-4
DC10069 CFI-400437 Featured

CFI-400437 is potent against PLK4 (IC50 = 0.6 nM) and selective against other members of the PLK family (>10 uM).

1247000-76-5
DC22809 c-FMS-IN-8 Featured

c-FMS-IN-8 is a potent, selective c-FMS kinase inhibitor with IC50 of 0.8 nM, shows activity in collagen-induced model of arthritis in mice..

885704-21-2
DC7039 CFTR Inhibitor II Featured

CFTR Inhibitor II is a cell-permeable glycinyl hydrazone compound that acts as a potent, selective and reversible open-channel blocker of CFTR with intermediate speed (< 1 min; 95% inhibition at 50 µM; Ki = 4.3 µM in CFTR-expressing FRT cells.

328541-79-3
DC12580 CG-806 Featured

CG-806 (CG806, CG'806) is a novel potent, pan-FLT3/BTK multi-kinase inhibitor with impressive inhibition of leukemic cell proliferation with IC50 at sub-nanomolar or low nanomolar levels.

1370466-81-1
DC7380 CGI-1746 Featured

CGI1746 is a small-molecule Btk inhibitor chemotype with a new binding mode that stabilizes an inactive nonphosphorylated enzyme conformation.

910232-84-7
DC7101 CGK733 Featured

CGK 733 is a potent and selective inhibitor of ATM/ATR with IC50 of ~200 nM.

905973-89-9
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