Cat. No. | Product name | CAS No. |
DC7731 |
Emapunil(AC-5216)
Featured
Emapunil(AC-5216;XBD-173) is a translocator protein |
226954-04-7 |
DC9620 |
EMD638683
Featured
EMD638683 is a potent SGK1 inhibitor with an IC50 of 3 uM. |
1181770-72-8 |
DC8885 |
EMICORON
Featured
EMICORON is a novel G-quadruplex (G4) ligand showing high selectivity for G4 structures over the duplex DNA, causing telomere damage and inhibition of cell proliferation in transformed and tumor cells. |
1422423-23-1 |
DC9771 |
ACU4429,ACU 4429,ACU-4429
Featured
Emixustat hydrochloride strongly inhibits 11-cis-retinol production with IC50 values of 232 ± 3 nM. |
1141934-97-5 |
DC10301 |
Emodepside
Featured
Emodepside (PF 1022-221) is a cyclooctadepsipeptide with broad-spectrum anthelmintic activity. |
155030-63-0 |
DC5018 |
Empagliflozin (BI-10773)
Featured
Empagliflozin is a potent, selective sodium glucose co-transporter-2 inhibitor that is in development for the treatment of type 2 diabetes. Empagliflozin is an inhibitor of the sodium glucose co-transporter-2 (SGLT-2), which is found almost exclusively in |
864070-44-0 |
DC23171 |
Empesertib(BAY 1161909)
Featured
Empesertib (BAY-1161909, BAY1161909) is a potent, selective Monopolar spindle 1 (Mps1/TTK) inhibitor with IC50 of 0.34 nM. |
1443763-60-7 |
DC9762 |
Emricasan
Featured
Emricasan (IDN-6556, PF-03491390) is a potent irreversible pan-caspase inhibitor. |
254750-02-2 |
DC5902 |
Emtricitabine
Featured
Emtricitabine is a nucleoside analogue which inhibits the reverse nucleoside transcriptase enzyme. Structurally this antiviral agent is similar to Lamivudine. This agent is effective at targeting HIV and HBV viruses since these viruses replicate in a reve |
143491-57-0 |
DC23108 |
EN460
Featured
EN460 is a specific mall molecule inhibitor of endoplasmic reticulum oxidation 1 (ERO1), interacts selectively with the reduced, active form of ERO1α and prevents its reoxidation (IC50=1.9 uM). |
496807-64-8 |
DC24204 |
EN6
Featured
EN6 is a small-molecule in vivo activator of autophagy that covalently targets cysteine 277 in the ATP6V1A subunit of the lysosomal v-ATPase, which activates mTORC1 via the Rag guanosine triphosphatases. |
1808714-73-9 |
DC8177 |
Enclomiphene citrate
Featured
Enclomiphene is a non-steroidal estrogen receptor antagonist that promotes gonadotropin-dependent testosterone secretion by the testes. |
7599-79-3 |
DC9959 |
Endoxifen (E-isomer)
Featured
Endoxifen (E-isomer hydrochloride) is a tamoxifen metabolite and potent Selective Estrogen Response Modifier (SERM). |
1197194-61-8 |
DC8403 |
Endoxifen (Z-isomer hydrochloride)
Featured
Endoxifen HCl, the active metabolite of Tamoxifen, ia a potent and selective estrogen receptor antagonist. Phase 2. |
1032008-74-4 |
DC8265 |
Endoxifen
Featured
Endoxifen is a Estrogen receptor α (ERα) ligand; potent antiestrogen,an active metabolite of the cancer drug tamoxifen. |
112093-28-4 |
DC7589 |
Eniporide(EMD96785)
Featured
Eniporide is a The Na(+)/H(+) exchange inhibitor. |
176644-21-6 |
DC20993 |
ENMD-1068
Featured
ENMD-1068 is a novel selective PAR2 antagonist without inhibitory activity against thrombin-mediated PAR3 and PAR4 signaling. |
789488-77-3 |
DC7118 |
ENMD-2076
Featured
ENMD-2076 has selective activity against Aurora A and Flt3 with IC50 of 14 nM and 1.86 nM, 25-fold selective for Aurora A than over Aurora B and less potent to VEGFR2/KDR and VEGFR3, FGFR1 and FGFR2 and PDGFRα. |
934353-76-1 |
DC9247 |
AP-III-a4 hydrochloride
Featured
ENOblock Hcl(AP-III-a4 Hcl) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasis in vivo. |
2070014-95-6 |
DC7119 |
ENO block(AP-III-a4)
Featured
ENOblock(AP-III-a4) is a novel small molecule which is the first, nonsubstrate analogue that directly binds to enolase and inhibits its activity (IC50=0.576 uM); inhibit cancer cell metastasis in vivo. |
1177827-73-4 |
DC20018 |
Enocyanin
Featured
Enocyanin is an anthocyanin extracted from grapes. Enocyanin shows inhibitory effect on the leucine aminopeptidase, acid phosphatase, γ-glutamyl transpeptidase and esterase activity. |
11029-12-2 |
DC10547 |
Ensartinib
Featured
Ensartinib is a potent inhibitor of ALK, which is used to treat non-small-cell lung cancer. |
1365267-27-1 |