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Cat. No. Product name CAS No.
DC45944 Guanosine 5'-triphosphate-5'-adenosine Featured

Guanosine 5'-triphosphate-5'-adenosine, the 5′ cap analog, is a fluorescent substrate analog.

10527-47-6
DC45945 Guattegaumerine

Guattegaumerine is a bisbenzylisoquinoline alkaloid with antimitotic, cytotoxic and neuroprotective activities.

21446-35-5
DC45948 HBC

HBC is a green fluorescent protein (GFP) fluorophore-like synthetic dye, with a structurally rigid electron acceptor and a strong electron donor. HBC is used to detect RNA localization.

156840-13-0
DC45949 Heishuixiecaoline A

Heishuixiecaoline A is a germacrane-type sesquiterpenoid. Heishuixiecaoline A shows protective effect on the neurotoxicity of PC12 cells induced by Aβ25-35.

1469493-85-3
DC45950 Hellebrigenol

Hellebrigenol is a metabolite of bufadienolides with antitumor activity.

508-79-2
DC45952 Isorhamnetin 3-O-β-D-glucose-7-O-β-D-gentiobioside

Isorhamnetin 3-O-β-D-glucose-7-O-β-D-gentiobioside is a bioactive constituent that can be found in the seeds of Lepidium apetalum Willd. Isorhamnetin 3-O-β-D-glucose-7-O-β-D-gentiobioside exhibits significant triglyceride (TG)-lowering effects in HepG2 cells.

60778-00-9
DC45955 Loureiriol

Loureiriol is a homoisoflavonoid with weak anticancer effects.

479195-44-3
DC45957 L-Tyrosine D4

L-Tyrosine D4 is a deuterium labeled L-Tyrosine. L-Tyrosine is a non-essential amino acid which can inhibit citrate synthase activity in the posterior cortex.

62595-14-6
DC45958 Malvidin chloride

Malvidin (chloride) is a bioactive compound isolated from Oryza sativacv. Heugjinjubyeo. Malvidin shows cytotoxicity through the arrest of the G2/M phase of cell cycle and induction of apoptosis. Malvidin can be used for the research of cancer.

643-84-5
DC45961 Methyl (E)-cinnamate

Methyl (E)-cinnamate (EMC), a phytochemical constituent isolated from Alpinia katsumadai Hayata, is a natural flavor compound with anti-inflammatory properties. Methyl (E)-cinnamate is widely used in the food and commodity industry.

1754-62-7
DC45962 Mnm5s2U

Mnm5s2U, found in lysine and glutamate tRNA anticodon, has an wobble modification function in tRNA.

32860-54-1
DC45963 Neolancerin

Neolancerin is a natural product with weak cytotoxic activity against HL-60 cells.

117221-65-5
DC45966 Pal-Glu(OSu)-OH

Pal-Glu(OSu)-OH is a side chain of Liraglutide. Liraglutide is a glucagon-like peptide-1 (GLP-1) receptor agonist that can be used for type 2 diabetes mellitus research.

294855-91-7
DC45969 S-(4-Hydroxybenzyl)glutathione

S-(4-Hydroxybenzyl)glutathione is a glutathione derivative. S-(4-Hydroxybenzyl)glutathione inhibits the in vitro binding of kainic acid to brain glutamate receptors, with an IC50 of 2 μM.

129636-38-0
DC45971 SAR629

SAR629 is a potent monoglyceride lipase (MGL) covalent inhibitor. SAR629 also inhibits 2-Arachidonoylglycerol (2-AG) degradation.

1221418-42-3
DC45972 Tarasaponin IV

Tarasaponin IV, as an oleanane-type triterpene saponin, is isolated from the bark of Aralia elata. Tarasaponin IV can be used for the research of cancer.

156980-31-3
DC45973 Tetrahydroxymethoxychalcone

Tetrahydroxymethoxychalcone is a phenolic and flavonoid compound. Tetrahydroxymethoxychalcone is found to enhance myoblast proliferation and differentiation. Tetrahydroxymethoxychalcone plays important roles in myogenesis and muscle regeneration.

197227-39-7
DC45975 Tumulosic acid

Tumulosic acid, a triterpenoid, inhibits KLK5 protease activity (IC50= 14.84 μM). Tumulosic acid suppresses the proteolytic processing of LL-37 in keratinocytes at ≤10 μM.

508-24-7
DC45978 γ-Asarone

γ-Asarone, a phenylpropene, shows strong correlation with the biological activities (anti-oxidative, anti-inflammatory and neurotrophic effects).

5353-15-1
DC45982 Thymectacin

Thymectacin (NB1011) is an agent selectively targeting tumor cells that have a high expression of thymidylate synthase (TS). Thymectacin is an aryloxy phosphoramidate derivative of BVdU (brivudin).

232925-18-7
DC45985 Salvianolic acid Y

Salvianolic acid Y is a phenolic acid with the same planar structure as Salvianolic acid B. Salvianolic acid Y rescues cell injury by H2O2.

1638738-76-7
DC45987 Pelargonidin 3-galactoside chloride

Pelargonidin 3-galactoside chloride is a major anthocyanin with anticancer effects. Pelargonidin 3-galactoside chloride inhibits α-glucosidase.

34425-22-4
DC45988 Echinocystic acid 28-O-β-D-glucoside

Echinocystic acid 28-O-β-D-glucoside is a metabolite of Echinocystic acid by microbial oxidation and glucosidation. Echinocystic acid 28-O-β-D-glucoside is a tissue factor pathway inhibitor, with an IC50 of 10.61 nM.

99633-30-4
DC45991 Luteolin-7-O-α-L-arabinopyranosyl (1→6)-β-D-glucopyranoside

Luteolin-7-O-α-L-arabinopyranosyl (1→6)-β-D-glucopyranoside is a flavonoid with antiradical activity.

52714-82-6
DC45992 Quercetin 3-O-(6''-O-galloyl)-β-D-glucoside

Quercetin 3-O-(6''-O-galloyl)-β-D-glucoside (Tellimoside) is a flavonol glycoside with strong inhibitory activity against the growth of Microcystis aeruginosa.

56316-75-7
DC45993 ICG-amine Featured

ICG amine, as a near-infrared fluorescent probe, binds to amino acid residues without condensing agents. ICG is a tricarbocyanine dye.

1686147-55-6
DC45994 Eupalinolide H

Eupalinolide H, a sesquiterpene lactone, has the potential to be used as natural anti-inflammatory agent.

1402067-83-7
DC45996 Gingerglycolipid A

Gingerglycolipid A is a monoacyldigalactosyl glycerol.

145937-22-0
DC45997 Emodin-1-O-β-gentiobioside

Emodin-1-O-β-gentiobioside is an anthraquinone.

849789-95-3
DC45999 SG3199-Val-Ala-PAB

SG3199-Val-Ala-PAB is an intermediate of Tesirine synthesis. Tesirine is a drug-linker conjugate for ADC which can be used for the research of several cancers.

1595275-61-8
DC46001 BPK-25

BPK-25, an active acrylamide, promotes degradation of nucleosome remodeling and deacetylation (NuRD) complex proteins by a post-translational mechanism involving covalent protein engagement. BPK-25 inhibits TMEM173 activation by the cyclic dinucleotide ligand cGAMP.

2305052-86-0
DC46002 DMAPP

DMAPP (Dimethylallyl pyrophosphate) is an isoprenoid precursor. DMAPP, as an isomer of isopentenyl pyrophosphate (IPP), exists in virtually all life forms.

358-72-5
DC46004 Kaempferol-3-O-α-L-rhamnopyranosyl-(1→6)-β-D-glucopyranosyl-(1→2)-β-D-glucopyranoside

Kaempferol-3-O-α-L-rhamnopyranosyl-(1→6)-β-D-glucopyranosyl-(1→2)-β-D-glucopyranoside is an antioxidant with an IC50 of 26.6 μM (DPPH assay).

476617-49-9
DC46005 Matairesinol monoglucoside

Matairesinol monoglucoside, a lignan compound, exhibits low activity on IFN-γ/STAT1 and IL-6/STAT3 signaling pathways with inhibition ratio of 5.8% and 7.0%, respectively.

34446-06-5
DC46007 Regaloside H

Regaloside H, a phenylpropanoid glycerol glucoside, is a gluconeogenesis inhibitor. Regaloside H can reduce glucose production in Hepatocytes.

126239-77-8
DC46008 Rhaponticin 2′′-O-gallate

Rhaponticin 2''-O-gallate, as a stilbene glucoside gallate, inhibits NO production.

94356-24-8
DC46009 Rhaponticin 6′′-O-gallate

Rhaponticin 6′′-O-gallate is a stilbene glucoside gallate that can be found in rhizome of Rheum undulatum L. Rhaponticin 6′′-O-gallate inhibits nitric oxide production in lipopolysaccharide-activated macrophages.

94356-23-7
DC46011 Anticancer agent 9

Anticancer agent 9, a glycine derivative, is an anticancer agent. Anticancer agent 9 can inhibit tumor cells viability of myelogenous leukemia and human prostate cancer.

592542-61-5
DC46012 Modified MMAF

Modified MMAF, an ADC cytotoxin, can be used in the synthesis of Antibody-drug Conjugate (ADC). Modified MMAF can be used for the targeted treatment of cancer.

1352202-47-1
DC46013 BPK-21

BPK-21, an active acrylamide, suppresses T cell activation through blockade of ERCC3 function. BPK-21 specifically targets C342 in the helicase ERCC3.

2305052-77-9
DC46016 Curcumin-β-D-glucuronide

Curcumin-β-D-glucuronide is a major metabolite after oral intake of Curcumin in hepatic tissue and portal blood. Curcumin-β-D-glucuronide can be used for the research of colon cancer.

227466-72-0
DC46018 Mn(II) protoporphyrin IX

Mn(II) protoporphyrin IX is a potential intravenous paramagnetic magnetic resonance contrast agent. Mn(II) protoporphyrin IX maintains strong paramagnetic properties.

21393-64-6
DC46020 7-Acetyllycopsamine

7-Acetyllycopsamine, a pyrrolizidine alkaloid, is a mild hepatotoxin. 7-Acetyllycopsamine can induce liver inflammation in mice.

73544-48-6
DC46023 Corymbiferin

Corymbiferin is one of active constituents, responsible for anti-diabetic properties. Corymbiferin improves antioxidant capacity and carbohydrate metabolism in diabetic rats, along with the improvement of histopathology of livers and pancreatic β cells.

5042-09-1
DC46024 Isoflupredone

Isoflupredone belongs to the class of corticosteroids and exerts its effect by binding to glucocorticoid and mineralocorticoid receptors of animals, such as horses. Isoflupredone can be used in wide range of conditions, such as infection and inflammatory diseases.

338-95-4
DC46025 Isorhamnetin 3,7-di-O-β-D-glucopyranoside

Isorhamnetin 3,7-di-O-β-D-glucopyranoside, a major flavonoid compound, is metabolized in vivo by intestinal bacteria to isorhamnetin and that isorhamnetin plays an important role as an antioxidant.

6758-51-6
DC46028 Stachyose

Stachyose, a small alkaloid, act as a hypoglycemic agent.

470-55-3
DC46029 Yadanzioside L

Yadanzioside L is a quassinoid and shows anti-tobacco mosaic virus (TMV) activity (IC50=4.86 μM).

99132-97-5
DC46031 Lucidin primeveroside

Lucidin primeveroside (Lucidin 3-O-β-primeveroside) is an anthraquinone derivative present in madder root, which has been used as a coloring agent and food additive. Lucidin primeveroside can be metabolically converted to genotoxic compound Lucidin, which subsequently forms lucidin-specific DNA adducts.

29706-59-0
DC46034 ABR-238901

ABR-238901 is an orally active and potent S100A8/A9 blocker and inhibits S100A8/A9 interaction with its receptors RAGE (receptor for advanced glycation endproducts) and TLR4 (toll-like receptor 4). ABR-238901 has the potential for myocardial infarction (MI) research.

1638200-22-2
DC46035 Encainide

Encainide (MJ9067) is an antiarrhythmic drug with class ⅠC activity. Encainide has the potential for life-threatening ventricular arrhythmias, symptomatic ventricular arrhythmias and supraventricular arrhythmias research.

66778-36-7
DC46040 Avasopasem manganese

Avasopasem manganese (GC4419; M-40419) is a potent superoxide dismutase mimetic that rapidly and specifically converts O2*- to hydrogen peroxide (H2O2), arresting the initiation of this cascade. Avasopasem manganese can be used for the research of severe oral mucositis (SOM) and cancer.

435327-40-5
DC46046 (3S,4S)-A2-32-01

(3S,4S)-A2-32-01 is a less active S-enantiomer of (3R,4R)-A2-32-01. (3R,4R)-A2-32-01 is an anti-virulence agent and a specific caseinolytic protein proteases (ClpP) inhibitor.

DC46047 Mal-PEG8-Val-Ala-PABC

Mal-PEG8-Val-Ala-PABC is a cleavable Tesirine linker used in the synthesis of Tesirine, a drug-linker conjugate for ADC.

DC46048 Szechenyin A

Szechenyin A is a constituent from Tibetan medicine Gentianae Szechenyii Spray.

DC46053 Cd(II) protoporphyrin IX

Cd(II) protoporphyrin IX is a protoporphyrin IX. Protoporphyrin IX is a heterocyclic organic compound, which consists of four pyrrole rings, and is the final intermediate in the heme biosynthetic pathway.

80216-25-7
DC46054 Pt(II) protoporphyrin IX

Pt(II) protoporphyrin IX is a protoporphyrin IX. Protoporphyrin IX is a heterocyclic organic compound, which consists of four pyrrole rings, and is the final intermediate in the heme biosynthetic pathway.

98303-94-7
DC46055 Ni(II) protoporphyrin IX

Ni(II) protoporphyrin IX is a metalloporphyrin that has a low tendency toward axial ligation, becomes distorted when bound to ferrochelatase.

15415-30-2
DC46056 Cu(II) protoporphyrin IX

Cu (II) Protoporphyrin IX is used as a negative control for Zn (II) Protoporphyrin (an inihibitor of heme oxygenase). Heme oxygenase has been implicated in tumor cell resistance to chemotherapy, reduction of free radical formation and inflammation, and associated with vascular repair.

14494-37-2
DC46057 Mg(II) protoporphyrin IX

Mg(II) protoporphyrin IX is a precursor of chlorophyll in Chlorella. Mg(II) protoporphyrin IX is a negative effector of nuclear photosynthetic gene expression. Mg(II) protoporphyrin IX can be used for the research of signaling molecule implicated in plastid-to-nucleus communication.

14947-11-6
DC46058 L-Iduronic acid sodium salt

L-Iduronic acid sodium salt is an important monosaccharide component of glycosaminoglycans (GAGs) such as Heparin, Heparan sulfate and Dermatan sulfate.

61199-83-5
DC46059 Cr(III) protoporphyrin IX

Cr(III) protoporphyrin IX is a protoporphyrin IX. Protoporphyrin IX is a heterocyclic organic compound, which consists of four pyrrole rings, and is the final intermediate in the heme biosynthetic pathway.

84640-43-7
DC46060 Macarangioside D

Macarangioside D, a megastigmane glucoside, possesses radical-scavenging activity.

819870-23-0
DC46061 Antioxidant 1024 Featured

Antioxidant 1024 (MD 1024) is an antioxidant agent and metal deactivator.

32687-78-8
DC46064 Coumberol

Coumberol is a fluorescent substrate of AKR1C3 protein. Coumberol can be used for the research of AKR1C3.

878019-53-5
DC46068 Dalbergin

Dalbergin is a composition of the extract from the Dalbergia Sissoo Linn. knot wood. Dalbergin demonstrats notable antioxidant ability.

482-83-7
DC46070 Epigambogic acid

Epigambogic acid is a natural anti-tumor, antitussive, expectorant and anti-inflammatory compound.

887606-04-4
DC46071 FR901463 Featured

FR901463 is a potent anti-cancer agent and can be used for cancer research. FR901463 enhances the transcriptional activity of the promoter of SV40 DNA virus.

146478-74-2
DC46072 Gentianose

Gentianose is a predominant carbohydrate reserve found in the storage roots of perennial Gentiana lutea.

25954-44-3
DC46073 Gomisin S

Gomisin S is a dibenzocyclooctadiene lignan.

119239-49-5
DC46074 Gomisin U

Gomisin U is a lignan compound.

135095-46-4
DC46075 Hemiphloin

Hemiphloin is a natural flavonoid.

71963-94-5
DC46078 Indicine N-oxide

Indicine N-oxide (NSC 132319), a pyrrolizidine alkaloid, is an antitumor agent for pediatric cancer and solid tumors research.

41708-76-3
DC46079 Isoarundinin II

Isoarundinin II is a stilbenoid compound.

151538-56-6
DC46080 Isofutoquinol A

Isofutoquinol A is a neolignan that can be found in Piper futokadzura.

62499-70-1
DC46081 Iso-oxypeucedanin

Iso-oxypeucedanin is a coumarin found in Angelica dahurica.

5058-15-1
DC46083 Lagotisoide D

Lagotisoide D is a lridoid glycoside from Lagotis yunnanensis.

834155-36-1
DC46084 Loureirin D

Loureirin D is a dihydrochalcone found in dragon’s blood.

119425-91-1
DC46085 Lucidin 3-O-glucoside

Lucidin 3-O-glucoside is an anthraquinone analogue.

22255-29-4
DC46086 MC-Ala-Ala-Asn-PAB

MC-Ala-Ala-Asn-PAB is a linker extracted from patent CN104147612A, page 14. MC-Ala-Ala-Asn-PAB can be used to synthesis the tumor microenvironment specific activated micromolecular targeted conjugate.

1638970-44-1
DC46090 Pasakbumin D

Pasakbumin D is a quassinoid and can be used for the research of cancer.

138874-44-9
DC46091 Poricoic acid AM

Poricoic acid AM is a triterpenoid with ant-tumor activities.

151200-92-9
DC46092 PTIO

PTIO is a specific scavenger of NO. PTIO reacts with •NO to form the corresponding imino nitroxides and •NO2.

18390-00-6
DC46093 Quercetin 3-O-neohesperidoside

Quercetin 3-O-neohesperidoside, a flavonoid glycoside, has anti-inflammatory activity.

32453-36-4
DC46094 Quercetin 3-O-sophoroside-7-O-rhamnoside

Quercetin 3-O-sophoroside-7-O-rhamnoside is a flavonoid found in sea buckthorn berries.

64828-40-6
DC46095 Rheumone B

Rheumone B possesses antioxidant activity.

2095596-67-9
DC46096 Rubiayannone A

Rubiayannone A is an anthraquinone glycoside with an antiplatelet aggregation activity.

517918-25-1
DC46097 Shancigusin I

Shancigusin I is a natural compound found in Cremastra appendiculata.

1435488-35-9
DC46098 Siaresinolic acid 28-O-β-D-glucopyranosyl ester

Siaresinolic acid 28-O-β-D-glucopyranosyl ester possesses anti-tumor and antidiabetic effect activity.

155653-86-4
DC46099 Sibiricose A1

Sibiricose A1is an oligosaccharide ester that can be found in Polygala tenuifolia.

139726-40-2
DC46100 Silyamandin

Silyamandin is a flavonolignan compound. Silydianin can form Silyamandin through oxidative degradation.

1009565-36-9
DC46101 Sterebin E

Sterebin E is a labdane diterpenoid that can be found in Stevia rebaudiana leaves.

114343-74-7
DC46102 Syringetin-3-O-glucoside

Syringetin-3-O-glucosid (Syringetin 3-O-β-D-glucoside), a flavonol glycoside, shows relatively weak DPPH and ABTS radical scavenging activity.

40039-49-4
DC46104 Wilfordinine D

Wilfordinine D is a natural sesquiterpene alkaloid.

256937-98-1
DC46105 Epipinoresinol-4'-O-β-D-glucoside

Epipinoresinol-4'-O-β-D-glucoside (Simplocosin) is a glucoside compound.

24404-49-7
DC46107 Yadanziolide C

Yadanziolide C is a quassinoid with antiproliferative and differentiation-inducing properties in promyelocytic HL-60 cells.

95258-12-1
DC46108 Yadanzioside I

Yadanzioside I is a potent anti-tobacco mosaic virus (TMV) quassinoid with an IC50 of 4.22 μM.

99132-95-3
DC46109 Yadanzioside F

Yadanzioside F is one of the toxic components found in Brucea javanica. Brucea javanica has demonstrated a variety of antitumoral, antimalarial, and anti-inflammatory properties.

95258-11-0
DC46110 Yadanzioside C

Yadanzioside C is a quassinoid glucoside found in seeds of Brucea amarissima.

95258-16-5
DC46111 Neokurarinol

Neokurarinol is a natural flavonoid compound.

52483-00-8
DC46113 Kushenol O

Kushenol O is a flavonoid compound.

102390-91-0
DC46114 Mudanpioside J

Mudanpioside J, a monoterpene glycoside, is a metabolite of cortex moutan.

262350-52-7
DC46116 Ginnol

Ginnol is a natural product found in Lonicera macranthoides.

2606-50-0
DC46117 Secologanic acid

Secologanic acid is a secoiridoid glycoside.

60077-46-5
DC46118 Crenulatin

Crenulatin is a gallotannin.

63026-02-8
DC46119 Isomitraphylline

Isomitraphylline, an oxindole alkaloid, has potent anti-cancer activity.

4963-01-3
DC46121 Isoscoparin-2′′O-glucoside

Isoscoparin-2′′O-glucoside is a flavonoid that can be found in yellow grain mutant of rice. Isoscoparin-2′′O-glucoside shows antioxidant activity.

97605-25-9
DC46122 Sutchuenmedin A

Sutchuenmedin A is a prenylflavonoid. Sutchuenmedin A is isolated from the 70% EtOH extract of Epimedium sutchuenense.

1197194-31-2
DC46123 L-Mannitol

L-mannitol is a compound can be used for  the compound sweetener synthesis.

643-01-6
DC46124 Dihydromollugin

Dihydromollugin is a natural naphthoic acid ester.

60657-93-4
DC46125 Euphorbia factor L8

Euphorbia factor L(8) is a diterpenoid from the seeds of Euphorbia lathyris.

218916-53-1
DC46128 Regaloside F

Regaloside F is a phenolic glycerol glucoside that can be found in Lily bulbs.

120601-65-2
DC46129 Euphorbia factor L7b

Euphorbia factor L7b is an isolathyrolditerpene compound.

93550-95-9
DC46130 Lucidone B

Lucidone B is a nortriterpenoid found in fruiting bodies of Ganoderma resinaceum.

97653-93-5
DC46134 DGK-IN-1

DGK-IN-1 is a T cell activator extracted from patent WO2020006018A1, example 25. DGK-IN-1 can be used for tumor immunity.

2407892-34-4
DC46135 Euphorbia factor L7a

Euphorbia factor L7a, as a natural product, is a diterpenoid from the seeds of Euphorbia lathyris.

93550-94-8
DC46136 Gardoside

Gardoside is an iridoid glycoside that can be found in the roots of L. alba.

54835-76-6
DC46137 Hythiemoside B

Hythiemoside B is isolated as a white amorphous powder. Hythiemoside B is an ent-pimarane glucoside isolated from the aerial part of Siegesbecikia orientalis L. (Asteraceae).

853267-90-0
DC46138 Isoanthricin

Isoanthricin ((Rac)-Deoxypodophyllotoxin) is the racemate of Deoxypodophyllotoxin. Deoxypodophyllotoxin is a potent antitumor and anti-inflammatory agent.

69222-20-4
DC46139 Kaempferol 3-O-rutinoside 7-O-glucoside

Kaempferol 3-O-rutinoside 7-O-glucoside is a flavonoid glycoside from red tomato.

34336-18-0
DC46140 Kizuta saponin K11

Kizuta saponin K11 is a saponin found in the leaves of Kalopanax pictum var. maximowiczii, a Korean medicinal plant.

97240-03-4
DC46141 Leonloside D

Leonloside D is a Hederagenin-derived saponin, composed of a molecule of Hederagenin and 1-3 molecules of rhamnose, glucose, or arabinose.

20830-84-6
DC46142 Methoxyeugenol 4-O-rutinoside

Methoxyeugenol 4-O-rutinoside (compound 9) is a phenyl glucoside that can be found in the bark of Daphniphyllum angustifolium.

903519-86-8
DC46143 Odoriflavene

Odoriflavene is a phenolic compound found in the root heartwood of Dalbergia odorifera T. Chen (Leguminosae).

101153-41-7
DC46144 Oxocrebanine

Oxocrebanine, an aporphine alkaloid, can be found in Fissistigma poilanei (Annonaceae).

38826-42-5
DC46146 Pratensein-7-O-β-D-glucopyranoside

Pratensein-7-O-β-D-glucopyranoside is a new isoflavone.

36191-03-4
DC46147 Rutarensin

Rutarensin is a phenolic compound found in Ruta chalepensis cell culture.

119179-04-3
DC46148 Sterebin A

Sterebin A is a bisnorditerpenoid that can be found in Blumea aromatic.

107647-14-3
DC46149 Volvalerenic acid A

Volvalerenic acid A is a germacrane-type sesquiterpenoid that can be found in the roots of Valeriana officinalis var. latifolia.

1247014-34-1
DC46151 Methyl 1,4-bisglucosyloxy-3-prenyl-2-naphthoate

Methyl 1,4-bisglucosyloxy-3-prenyl-2-naphthoate is a natural product.

90685-26-0
DC46152 rel-(1S,2S,3R,4S)-1,2-Epoxy-3-methoxyfuranogermacr-10(15)-en-6-one

rel-(1S,2S,3R,4S)-1,2-Epoxy-3-methoxyfuranogermacr-10(15)-en-6-one is a sesquiterpene.

75412-95-2
DC46153 (±)-ErSO Featured

(±)-ErSO is the racemate of ErSO. ErSO is a selective anticipatory unfolded protein response (a-UPR) activator.

2407860-40-4
DC46157 Beta-D-Glucopyranosyl nitromethane

Beta-D-Glucopyranosyl nitromethane, as a salt of a strongly basic anion exchanger in the OH cycle, is a glycosyl derivative of nitromethane.

81846-60-8
DC46159 (R)-PF-06256142

(R)-PF-06256142 is the R enantiomer of PF-06256142 with low active. PF-06256142 is a potent and selective orthosteric D1 receptor agonist that can reduce receptor desensitization relative to dopamine and other catechol-containing agonists.

1609583-15-4
DC46160 LIN28 inhibitor LI71 enantiomer

LIN28 inhibitor LI71 enantiomer is the enantiomer of LIN28 inhibitor LI71 with less active. LIN28 inhibitor LI71 is a potent and cell-permeable LIN28 inhibitor, which abolishes LIN28-mediated oligouridylation with an IC50 of 7 uM.

956189-58-5
DC46164 MG-2119

MG-2119 is a potent monomeric tau and α-syn aggregation inhibitor. MG-2119 is a potential agent for neurological disorders research.

1065500-40-4
DC46168 (3S,4S)-PF-06459988

(3S, 4S)-PF-06459988 is the S enantiomer of PF-06459988 with less active. PF-06459988 is a potent irreversible inhibitor of T790M mutant epidermal growth factor receptor (EGFR). PF-06459988 has excellent selectivity against EGFR wild-type while possessing a minimally reactive electrophile that reduces the propensity of off-target labeling.

1858291-14-1
DC46176 BGSN3

BGSN3 is a good substrate for the SNAP-tag® and H5 enzymes. The activities of SNAP-tag® and H5 enzymes on BGSN3 are reasonable (IC50=17.8 and 10 μM, respectively).

DC46181 ECBN hydrochloride Featured

A-30912A nucleus hydrochloride is the product of the reaction catalyzed by Echinocandin B (ECB) deacylase.

1029890-89-8
DC46182 Didemnin B Featured

Didemnin B is a depsipeptide extracted from the marine tunicate Trididemnin cyanophorum. Didemnin B can be used for the research of cancer.

77327-05-0
DC46185 4-Vinylcyclohexene dioxide

4-Vinylcyclohexene dioxide (Vinylcyclohexene dioxide, VCD) is a chemical used to induce menopause and decrease estrogen production. 4-Vinylcyclohexene dioxide is used as a crosslinking agent for the production of epoxy resins.

106-87-6
DC46186 Gadoteridol

Gadoteridol (ProHance, SQ-32692, Gd-HP-DO3A) is a nonionic contrast agent for magnetic resonance imaging (MRI).

120066-54-8
DC46187 Triheptanoin

Triheptanoin (API, IND106011, UX007, Glycerol trienanthate) is a synthetic, medium-chain triglyceride consisting of three odd-chain 7-carbon (heptanoate) fatty acids on a glycerol backbone. Triheptanoin is used for treatment of fatty acid oxidation disorders and GLUT1.

620-67-7
DC46188 NSC622608

NSC622608 is a first small-molecule ligand for V-domain Ig Suppressor of T-cell Activation (VISTA) with an IC50 of 4.8 μM in TR-FRET assay.

2593254-90-9
DC46191 Compound W

Compound W (3,5-Bis(4-nitrophenoxy)benzoic acid) is an inhibitor of γ-secretase. Compound W causes a decrease in the released levels of Aβ42 and notch-1 Aβ-like peptide 25 (Nβ25).

173550-33-9
DC46193 BRM/BRG1 ATP Inhibitor-1 Featured

BRM/BRG1 ATP Inhibitor-1 is an orally active inhibitors of Brahma Homolog (BRM)/SMARCA2 with IC50 below 0.005 µM.

2270879-17-7
DC46194 Abz-FRLKGGAPIKGV-EDDNP TFA

Abz-FRLKGGAPIKGV-EDDNP TFA is a fluorogenic substrate used to measure the enzymatic activities of protease forms, such as papain-like protease 2 (PLP2) from severe acute respiratory syndrome coronavirus (SARS-CoV). Abz-FRLKGGAPIKGV-EDDNP TFA has the potential for study 2019-nCoV (COVID-19) infection.

DC46196 AgAuSe QDs

AgAuSe QDs (AgAuSe) is a near infrared (NIR) fluorescent quantum dots (QDs), with a bright emission from 820 to 1170 nm. AgAuSe QDs can be used for the research in biomedical imaging and NIR devices.

DC46197 PbS/CdS QDs

PbS/CdS QDs (PbS/CdSe QD) is a fluorescent probe that can be used for in vivo fluorescence imaging in the second near-infrared window.

DC46221 AZ-PFKFB3-67 quarterhydrate

AZ-PFKFB3-67 quarterhydrate is potent and selective metabolic kinase PFKFB3 inhibitor, with IC50s of 11, 159 and 1130 nM for PFKFB3, PFKFB2 and PFKFB1 respectively.

DC46236 4-Methylumbelliferyl β-D-Glucopyranoside

4-Methylumbelliferyl β-D-Glucopyranoside, a β-D-glucoside, is a fluorogenic substrate for β-glucosidase, utilizes to assay β-glucosidase activity. 4-Methylumbelliferyl β-D-Glucopyranoside releases the highly fluorescent 4-methylumbelliferyl (4-MU), which has an emission maximum at 445-454 nm. The excitation maximum for 4-MU is pH-dependent: 330, 370, and 385 nm at pH 4.6, 7.4, and 10.4, respectively.

18997-57-4
DC46237 THK-5470(THK5470) Featured

THK-5470(THK 5470), a monoamine oxidase-B (MAO-B) imaging probe, could be used for neurological diseases study. THK-5470 shows remarkably high binding affinity against MAO-B with an IC50 value of 4.2 nM, low binding affinity against tau with an IC50 value of 4462 nM. THK-5470 has high selective binding property and high affinity (from patent EP2019-846498).

2410554-04-8
DC46245 FAPI-34

FAPI-34 is a fibroblast-activating protein (FAP) inhibitor with favorable pharmacokinetic and biochemical properties. (patent WO2019154886A1).

2374782-07-5
DC46246 Ilexoside XLVIII

Ilexoside XLVIII is an acyl CoA cholesteryl acyl transferase (ACAT) inhibitor. Ilexoside XLVIII is a triterpene saponin isolated from an aqueous extract of the leaves of Ilex kudincha.

129095-76-7
DC46270 WRW4 TFA

WRW4 TFA, a specific formyl peptide receptor-like 1 (FPRL1) antagonist, inhibits WKYMVm binding to FPRL1 with an IC50 of 0.23 μM. WRW4 TFA specifically inhibits the increase in intracellular calcium by the FPRL1 agonists MMK-1, amyloid beta42 (Abeta42) peptide, and F peptide.

DC46272 MAIT-203

MAIT-203, a cyclopentyalanin-derived peptidomimetic, potently inhibits the interaction of adenomatous polyposis coli (APC) and Asef (RhoGEF4), but not APC-Sam68 or APC-striatin interactions. MAIT-203 binds APC-ARM with a Ki of 0.015 μM and a Kd of 0.036 μM. MAIT-203 significantly represses the migration and invasion of colorectal cancer cells.

DC46284 L-Leucine-7-amido-4-methylcoumarin hydrochloride

L-Leucine-7-amido-4-methylcoumarin (Leu-AMC) hydrochloride is a bright blue fluorogenic peptidyl substrate for LAP3 (leucine aminopeptidase). L-Leucine-7-amido-4-methylcoumarin hydrochloride can be used for leucine aminopeptidase inhibition assays in vitro.

62480-44-8
DC46302 Hexidium iodide

Hexidium iodide, a fluorescent nucleic binding acid stain (excitation/emission ~ 518/600 nm), permeants to mammalian cells and selectively stains almost all gram-positive bacteria. Hexidium iodide can bind to the DNA of all bacteria after permeabilization by EDTA.

211566-66-4
DC46303 PFB-FDGlu

PFB-FDGlu is a selective lysosomal Glucocerebrosidase (GCase) substrate, which is metabolised by GCase to yield fluorescein. PFB-FDGlu is cell permeable and can be used with a flow cytometer to measure GCase activity in living cells on a single-cell basis.

209540-62-5
DC46304 Trimethylolpropane ethoxylate triacrylate

Trimethylolpropane ethoxylate triacrylate (ETPTA) is a plasticizer that can be used synthesize nanocomposites.

28961-43-5
DC46305 4-Hydroxymephenytoin D3

4-Hydroxymephenytoin D3 is the deuterium labeled 4-Hydroxymephenytoin. 4-Hydroxymephenytoin is a metabolism of an antiepileptic drug mephenytoin, which is used as a CYP2C19 substrate.

1173022-56-4
DC46306 Ganciclovir mono-O-acetate

Ganciclovir mono-O-acetate is a derivative of Ganciclovir. Ganciclovir, a nucleoside analogue, is an orally active antiviral agent with activity against CMV.

88110-89-8
DC46312 Adipokinetic Hormone (AKH) (24-32), locust TFA

Adipokinetic Hormone (AKH) (24-32), locust (TFA), isolated from locust corpora cardiaca, is a neurohormone that regulates lipid utilisation during flight.

DC46313 Photo-lysine hydrochloride

Photo-lysine hydrochloride, a new lysine-based photo-reactive amino acid, captures proteins that bind lysine post-translational modifications.

DC46315 trans,trans-2,4-Decadienal

trans,trans-2,4-Decadienal is a lipid peroxidation product of linolieic acid.

25152-84-5
DC46316 1-Methyl-2-[(Z)-6-undecenyl]-4(1H)-quinolone

1-Methyl-2-[(Z)-6-undecenyl]-4(1H)-quinolone, as a colorless oil, is a quinolone alkaloid isolated from the fruit of Evodia rutaecarpa BENTHAM (Rutaceae).

120693-49-4
DC46320 HBC599

HBC599 is a HBC analog. HBC is nonfluorescent in solution, but emits strong fluorescence upon forming tight complex with Pepper RNA aptamer. HBC-Pepper complex can be used to visualize RNA dynamics in live cells.

2530162-00-4
DC46321 SiR-COOH

SiR-COOH could be used to follow the intracellular location of the model therapeutic drug in GFP cells (Abs, 645 nm; Em, 676 nm).

1418275-26-9
DC46326 (±)-H3RESCA-TFP

(±)-H3RESCA-TFP ((±)-H3L28) is a tetrafluorophenyl ester derivative of restrained complexing agent (RESCA). (±)-H3RESCA-TFP can be used to conjugate the chelator with a biomolecule via amine coupling (e.g., N terminus and/or the ε-amino groups of lysine).

1919794-40-3
DC46327 Methyl 5-hydroxypyridine-2-carboxylate

Methyl 5-hydroxypyridine-2-carboxylate is a phenolic acid that can found in the stems of Mahonia fortune. Methyl 5-hydroxypyridine-2-carboxylate exhibits NO inhibitory effects in vitro.

30766-12-2
DC46328 NHS-MMAF

NHS-MMAF is a modified MMAF extracted from patent WO2012143499, intermediat 219. MMAF is a potent tubulin polymerization inhibitor and is used as a antitumor agent

1404073-19-3
DC46329 Phoyunnanin E

Phoyunnanin E, isolated from Dendrobium venustum, possesses anti-migration activity. Phoyunnanin E can be used for the research of cancer.

886747-60-0
DC46330 pNP-ADPr

pNP-ADPr is a colorimetric substrate that used for the first continuous Poly(ADP-ribose) glycohydrolase (PARG) and ADP-ribosyl hydrolase 3 (ARH3) activity assays. pNP-ADPr can be used for the research of poly(ADP-ribose)polymerase (PARP) enzymes.

939028-75-8
DC46331 Sodium dodecyl sulfate D25

Sodium dodecyl sulfate D25 is a deuterium labeled Sodium dodecyl sulfate. Sodium dodecyl sulfate is the most widely used of the anionic alkyl sulfate surfactants.

110863-24-6
DC46332 tert-OMe-byakangelicin

tert-OMe-byakangelicin is a coumarin that can enhances the adrenaline-induced lipolytic effect and inhibits insulin-stimulated triglyceride synthesis from glucose in fat cells.

79638-04-3
DC46333 Tris-NTA

Tris-NTA is a His-tagged protein ligand, which can be used to bind His-tagged proteins.

1146592-99-5
DC46334 Gyrophoric acid

Gyrophoric acid is a good ultraviolet filter in lichen populations. Gyrophoric acid shows DPPH radical scavenging activity with an IC50 value of 105.75 µg/ml.

548-89-0
DC46335 Isobyakangelicol

Isobyakangelicol is a coumarin that can be found in the roots of Angelica dahurica. Isobyakangelicol inhibits the growth of HeLa and HepG2 cells, with IC50s of 70.04 μM and 17.97 μM.

35214-81-4
DC46337 3X FLAG peptide

3X FLAG Peptide is a synthetic peptide with a 3-time repeated DYKXXD motif.

402750-12-3
DC46342 Protein E7(43-62) TFA

Protein E7(43-62) TFA is an E7-derived peptide with anti-tumor effects (short peptide spanning the 43th to 62th amino acid residues in the E7 protein).

DC46343 PSEM 308 hydrochloride

PSEM 308 hydrochloride is a pharmacologically selective actuator module (PSAM) agonist. PSEM 308 Activates PSAML141F-GlyR chimeric ion channels.

DC46344 FATP1-IN-1

FATP1-IN-1 is a fatty acid transport protein 1 (FATP1) inhibitor. FATP1-IN-1 is an inhibition of recombinant human or mouse acyl-CoA synthetase activity of FATP1, with the IC50 values of 0.046 μM or 0.60 μM, respectively.

1431945-95-7
DC46349 ALS-I Featured

ALS-I, an acid-Liable surfactant, is adopted for in-solution enzymatic digestions, can help to solubilize hydrophobic proteins. ALS-I is significantly enhanced peptide recovery for mass spectrometry (MS) mapping in the study of the proteomes of regenerating rat retina and mouse brain.

308818-13-5
DC46351 Ac2-12 TFA

Ac2-12 TFA, an annexin/lipocortin 1 (LC1)-mimetic peptide, inhibit neutrophil extravasation. Ac2-12 TFA has antimigratory action and inhibits recruitment of neutrophils in experimental inflammation models.

DC46352 Encainide hydrochloride

Encainide (MJ9067) hydrochloride is an antiarrhythmic drug with class IC activity. Encainide has the potential for life-threatening ventricular arrhythmias, symptomatic ventricular arrhythmias and supraventricular arrhythmias research.

66794-74-9
DC46353 PEG-8 laurate

PEG-8 laurate is a single chain surfactant. PEG-8 laurate reduces the skin barrier, and acts as a penetration enhancer. PEG-8 laurate can be used to synthesize elastic vesicles.

35179-86-3
DC46354 Neopanaxadiol

Neopanaxadiol, an aglycone of protopanaxadiol type ginsenosides, has the potential for Alzheimer's disease research.

1203590-03-7
DC46355 γ-Terpinene

γ-Terpinene, a monoterpene, is an orally active antioxidant compound which can scavenge radicals directly. γ-Terpinene has potent antinociception activity.

99-85-4
DC46360 A 71915

A 71915 is a highly potent and competitive natriuretic peptide receptor A (ANP, NPRA) antagonist (pKi= 9.18). A 71915 displaces [125I]ANP dose dependently, with a Ki of 0.65 nM. A71915( pA2= 9.48) against rat ANP-induced cGMP production in NB-OK-1 cells.

132956-87-7
DC46368 Carnostatine

Carnostatine (SAN9812) is a potent and selective carnosinase 1 (CN1) inhibitor with a Ki of 11 nM for human recombinant CN1. Carnostatine (SAN9812) can be used for the treatment of diabetic nephropathy (DN).

DC46370 VGSC blocker-1

VGSC blocker-1 is a potent and small molecule blocker of neonatal isoform of the VGSC subtype, Nav1.5 (nNav1.5). VGSC blocker-1 blocks INa peak currents 34.9% at 1 μM and inhibits cell invasion 0.3% at 1 μM in human breast cancer cell line MDA-MB-231, without affecting the cell viability.

2230472-55-4
DC46383 Mycalolide B

Mycalolide-B is a specific inhibitor of actomyosin ATPase isolated from marine sponge. Mycalolide-B inhibits ATP-induced contraction and Mg2+-ATPase activity in the absence of Ca2+.

122752-21-0
DC46394 MK-8262 Featured

MK-8262 is an orally active and potent cholesteryl ester transfer protein (CETP) inhibitor with an IC50 of 53 nM and a log D of 5.3. MK-8262, a bistrifluoromethyl analogue, has the potential for coronary heart disease (CHD) correlated high-density lipoprotein (HDL) and low-density lipoprotein (LDL) research.

1432054-03-9
DC46396 PRGL493

PRGL493 is a potent and selective long-chain acyl-CoA synthetase 4 (ACSL4) inhibitor. PRGL493 blocks cell proliferation and tumor growth in both breast and prostate cellular and animal models. PRGL493 is used for cancer research.

2479378-45-3
DC46403 Ethaselen

Ethaselen (BBSKE) is an orally active, selective thioredoxin reductase (TrxR) inhibitor with IC50s of 0.5 and 0.35 μM for the wild-type human TrxR1 and rat TrxR1, respectively. Ethaselen specifically binds to the unique selenocysteine-cysteine redox pair in the C-terminal active site of mammalian TrxR1. Ethaselen, an organoselenium compound, is a potent antitumor candidate that exerts potent inhibition on non-small cell lung cancer (NSCLC) by targeting TrxR.

217798-39-5
DC46404 Posizolid

Posizolid (AZD2563), an oxazolidinone antibiotic, is developed by AstraZeneca for the study of bacterial infections. Posizolid shows very good anti-mycobacterial activity.

252260-02-9
DC46411 AB-680 ammonium

AB-680 ammonium is a highly potent, reversible and selective inhibitor of CD73 (an ecto-nucleotidase), with a Ki of 4.9 pM for hCD73, displays >10,000-fold selectivity over related ecto-nucleotidases CD39. Anti-tumor activity.

DC46416 FTO-IN-1 TFA

FTO-IN-1 TFA is a fat mass and obesity-associated enzyme (FTO) inhibitor extracted from patent WO2018157843A1, compound 32, with an IC50 of <1 μM. FTO-IN-1 TFA can be used for the research of cancer.

DC46419 11R-VIVIT TFA Featured

11R-VIVIT TFA is a cell-permeable nuclear factor of activated T cells (NFAT) inhibitor. 11R-VIVIT TFA can be used for the research of podocyte and diabetic nephropathy.

DC46422 GSK9027

GSK9027, as a non-steroidal glucocorticoid receptor (GR) agonist, behaves as a partial agonist on the 2×glucocorticoid response element (GRE) reporter system, and achieves intrinsic activities relative to dexamethasone.

1229096-88-1
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