Cat. No. | Product name | CAS No. |
DC7508 |
SU 5402
Featured
SU5402(SU-5402; SU5402) is potent and selective vascular endothelial growth factor receptor (VEGFR) and fibroblast growth factor receptor (FGFR) inhibitor. (IC50 values are 0.02, 0.03, 0.51 and > 100 μM at VEGFR2, FGFR1, PDGFRβ and EGFR respectively). |
215543-92-3 |
DC9950 |
SU5614
Featured
SU5614 is a potent and selective FLT3 inhibitor. |
1055412-47-9 |
DC5079 |
Orantinib (TSU-68)
Featured
SU6668 has greatest potency against PDGFR autophosphorylation with Ki of 8 nM, but also strongly inhibits Flk-1 and FGFR1 trans-phosphorylation, little activity against IGF-1R, Met, Src, Lck, Zap70, Abl and CDK2; does not inhibit EGFR. |
252916-29-3 |
DC21710 |
SU-909
Featured
SU-909 (SU909, IKKα-IN-48) is a potent, selective IKKα inhibitor with Ki of 0.08±0.07 uM, 10-20-fold selectivity over IKKβ (IC50=1.0±0.28 uM); inhibits FCS-stimulated phosphorylation of p100 in U2OS cells with IC50 of 8.8 uM, inhibits the noncanonical NF-kB pathway without affecting IKKβ-dependent IKappa-Bα loss in the canonical pathway. |
2126749-48-0 |
DC7928 |
SU9516
Featured
SU-9516 is a selective CDK2 inhibtor with IC50 of 22 nM; less potent for CDK1/CDK4(IC50=40/200 nM), no inhibition on PKC, EGFR, p38MAPK etc. |
377090-84-1 |
DC6906 |
Aprepitant (MK-0869, L-754030)
Featured
Substance P antagonists (SPA). |
170729-80-3 |
DC10664 |
Substance P free acid
Featured
Substance P free acid is a Sensory neuropeptide and inflammatory mediator. Exerts excitatory effects on central and peripheral neurons, constricts bronchioles and is involved in pain transmission. |
71977-09-8 |
DC10663 |
Substance P
Featured
Substance P is a Sensory neuropeptide and inflammatory mediator. Exerts excitatory effects on central and peripheral neurons, constricts bronchioles and is involved in pain transmission. |
33507-63-0 |
DC11334 |
Suc-Ala-Ala-Pro-Abu-pNA trifluoroacetate salt
Featured
Suc-AAP-Abu-pNA is a chromogenic peptide substrate for pancreatic elastase.It is cleaved by elastase to release p-nitroalinide (p-NA), which can be quantified by colorimetric detection at 405 nm as a measure of enzyme activity. |
108392-27-4 |
DC10581 |
Succinobucol(AGI 1067)
Featured
Succinobucol is a phenolic antioxidant with anti-inflammatory and antiplatelet effects. |
216167-82-7 |
DC26055 |
Caspase-1/4 Chromogenic Substrate(Suc-YVAD-pNA)
Featured
Suc-YVAD-pNA is a colorimetric substrate for caspase-1/interleukin-1β-converting enzyme (ICE) and caspase-4. |
208264-84-0 |
DC9732 |
Sufugolix(TAK-013)
Featured
Sufugolix(TAK-013) is a non-peptide, orally-active, selective antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (IC50 = 0.1 and 0.06 nM for affinity and in vitro inhibition, respectively). |
308831-61-0 |
DC22567 |
Sulfatinib
Featured
Sulfatinib (HMPL-012) is a potent, multi-targeted tyrosine kinase inhibitor of VEGFR-1/2/3, FGFR1, CSF1R with IC50 of 2/24/1 nM, 15 nM, 4 nM, respectively. |
1308672-74-3 |
DC10349 |
Sumanirole maleate
Featured
Sumanirole maleate(PNU 95666E; U95666E) is a highly selective D2 receptor full agonist with an ED50 of about 46 nM. |
179386-44-8 |
DC10271 |
SUN11602
Featured
SUN11602 is a novel aniline compound, which mimics the neuroprotective mechanisms of basic fibroblast growth factor. |
704869-38-5 |
DC3145 |
Sunitinib base
Featured
Sunitinib Malate (Sutent, SU11248) is a multi-targeted RTK inhibitor targeting VEGFR2 (Flk-1) and PDGFRβ with IC50 of 80 nM and 2 nM, and also inhibits c-Kit. |
557795-19-4 |
DC3146 |
Sunitinib malate
Featured
Sunitinib Malate (Sutent, SU11248) is a multi-targeted RTK inhibitor targeting VEGFR2 (Flk-1) and PDGFRβ with IC50 of 80 nM and 2 nM, and also inhibits c-Kit. |
341031-54-7 |
DC20205 |
Super-TDU
Featured
Super-TDU is an inhibitory peptide targeting YAP-TEADs interaction. |
1599441-71-0 |
DC10733 |
Sutezolid (PNU-100480)
Featured
Sutezolid (PNU-100480) is an oxazolidinone antimicrobial being developed for the treatment of tuberculosis. |
168828-58-8 |
DC22238 |
SUVN-G3031
Featured
SUVN-G3031 (SUVN-G 3031) is a potent, selective, orally active histamine H3 receptor (H3R) inverse agonist with Ki of 8.73 nM (hH3R). |
1394808-82-2 |
DC5017 |
Suvorexant
Featured
Suvorexant (MK-4305) is a potent, selective, and orally bioavailable antagonist of OX1R and OX2R currently under clinical investigation as a novel therapy for insomnia.Suvorexant is an analytical reference standard categorized as a diazepane sedative.Formulations containing suvorexant show abuse potential similar to zolpidem in recreational polydrug users with a history of sedative and psychedelic drug use.2 Suvorexant is regulated as a Schedule IV compound in the United States. This product is intended for use in analytical forensic applications. |
1030377-33-3 |
DC8267 |
SW033291
Featured
SW033291 is a potent inhibitor of 15-PGDH enzyme with IC50 value of 1.5 nM and dissociation constant Ki app value of 0.1 nM. |
459147-39-8 |