Home > Inhibitors & Agonists
Cat. No. Product name CAS No.
DCC3193 Ly544344

Prodrug of LY354740, highly selective and potent agonist of group II mGlu receptors (mGluR2)

441765-98-6
DCC3194 Ly-580276

Novel inhibitor of the type I transforming growth factor beta receptor (TβRI)

476475-07-7
DCC3195 Lyc-31138

Novel F1F0-ATPase modulator, significantly decreasing M2 glutamate and increasing M4 glutamate

1381806-47-8
DCC3196 Ly-hn2am

Nove fluorescent probe for highly sensitive monitoring drug induced lysosomal pH value changes, exhibiting good biological compatibility, low cytotoxicity and high resistance to photobleaching

DCC3197 Lyngbyastatin 7

Natural Potent Marine-Derived Elastase Inhibitor

DCC3198 Lysine Orotate

Inhibitor of viral replication, especially useful in the treatment of the Herpes family of viruses which includes Herpes Simplex 1 and 2 , EBV , CMV and Varicella.

28003-86-3
DCC3199 Lyso-7

Inhibitor of cyclooxygenase (COX); Pan partial agonist of PPARγ, PPARα and PPARβ/δ

1244215-18-6
DCC3200 Lzz-02

Novel inhibitor of the transcriptional activity of β-catenin, degrading the expression of β-catenin by stabilizing axin 2 and diminishing downstream proteins levels, including c-Myc and cyclin D1, effectively shrinking tumor xenograft derived from colonic

5307-25-5
DCC3201 M-084 Hydrochloride

TRPC4/5 channel blocker, exhibiting antidepressant and anxiolytic effects

51314-51-3
DCC3202 M1-pam-a

Novel selective muscarinic M1 receptor positive allosteric modulator, significantly improved scopolamine-induced cognitive deficits without prominent signs of diarrhea at up to 1000 mg/kg in mice

DCC3203 M1-pam-b

Novel selective muscarinic M1 receptor positive allosteric modulator, showed both significant improvement of scopolamine-induced cognitive deficits and severe diarrhea

DCC3204 M4k2009 Featured

M4K2209 is a potent, selective BMP type I receptor ALK2 inhibitor with IC50 of 9 nM, >180-fold selective over ALK5 (IC50=2427 nM).

2600795-07-9
DCC3205 M4k2127

Novel potent and selective ALK2 inhibitor, showing high initial brain uptake, including in the region of interest (pons)

DCC3206 M4k2163

Novel CNS Penetrant ALK2 Inhibitor for the Treatment of Diffuse Intrinsic Pontine Glioma

DCC3207 M-5mpep

Partial antagonist of mGlu5

872428-47-2
DCC3208 M7594_0037

Novel Peptide Deformylase (PDF) Inhibitor, having inhibitory activity against HeLa, A549 and MCF-7

774551-07-4
DCC3209 Mac-0547630

Novel potent and selective inhibitor of UppS without off-target effects on membrane potential

950386-41-1
DCC3210 Mac13243

Novel inhibitor of the bacterial lipoprotein targeting chaperone, LolA

1071638-38-4
DCC3211 Macluraxanthone

Natural immunomodulator, significantly decreasing TNF-α and IL-10 cytokine production, regulating the NF-κB and MAPK signaling pathways, displaying the strongest antiproliferative effects with IC50 values of 2.84 and 0.95 μM against A431 and HeLa cancer c

5848-14-6
DCC3212 Madtp-372

Potent and selective inhibitor of the induction of cytopathic effect by CHIKV and VEEV

DCC3213 Madurmycin

Polyether ionophore antibiotic, inhibiting proliferation and induces apoptosis in myoblast cells

61991-54-6
DCC3214 Magl-2102

Novel reversible monoacylglycerol lipase (MAGL) inhibitor

DCC3215 Magnesium L-threonate

Inhibitor of TNF-α, preventing and restoring memory deficits associated with neuropathic pain

778571-57-6
DCC3216 Magnesium Oxaloacetate

Inhibitor of the amebicidal activity of activated murine macrophages, helping the parasite to survive within the mouse large intestine and increasing the survival of C. elegans exposed to H2O2

59866-21-6
DCC3217 Magreth-16a

Potent CB2 receptor inverse agonist

DCC3218 Malonganenone A

Selective modulator of plasmodial Hsp70s with antimalarial activity

882403-69-2
DCC3219 Malp-2

Toll-like receptor 2/6 (TLR-2/6) agonist, regulating Lcn2 gene, promoting collateral growth

250718-44-6
DCC3220 Malp-2s

TLR2/6 agonist, activating the MyD88 pathway, provoking natural killer (NK) cell activation, increasing co-stimulators CD80/86 and CD40

DCC3221 Mal-rp

Novel quantitative chemical probe for live cell labeling and imaging of proteins that are sensitive to redox modifications

1485456-25-4
DCC3222 Manassantin A

Natural anticancer, anti-inflammatory, neuroleptic agent, also having human acyl-CoA:cholesterol acyltransferase (ACAT) inhibitory activities

88497-87-4
DCC3223 Mao-b Inhibitor 58

Highly potent, selective, competitive, and reversible inhibitor of monoamine oxidase B (MAO-B).

1619884-75-1
DCC3224 Mao-b Inhibitor C3

Novel potent and highly selective MAO-B Inhibitor

DCC3225 Mao-b Inhibitor C5

Potent and selective MAO-B inhibitor

1230-77-9
DCC3226 Mao-b Inhibitor Cc1

Novel potent selective and competitive inhibitor of MAO-B (IC 50 : 0.69 μM)

140399-50-4
DCC3227 Mao-b Inhibitor Cc2

Novel potent and competitive inhibitor of MAO-B (IC 50 : 0.51 μM), also inhibiting BChE (IC 50 : 7.00 μM)

DCC3228 Mao-b Ligand-1

Novel selective MAO-B inhibitor

1010879-39-6
DCC3229 Ma-pabc-adc-linker-18

Novel stable antibody-drug conjugate (ADC) in mouse serum

DCC3230 Maprotiline

Inhibitor of neuronal norepinephrine reuptake, reducing symptoms of anxiety associated with depression.

10262-69-8
DCC3231 Marbotinib

Novel highly efficient dual type I/II FMS-like tyrosine kinase inhibitor, disrupting the growth of leukemic cells

DCC3232 Margatoxin

Inhibitor of voltage-gated K(+) (Kv) channels Kv1.3 and Kv1.5

145808-47-5
DCC3233 Maritinone

Novel, active, and less toxic anti-tuberculosis (anti-TB) agent

33927-59-2
DCC3234 Maropitant Citrate [359875-09-5] Featured

Neurokinin receptor antagonist with antiemetic activity

359875-09-5
DCC3235 Massiliamide

Novel potent tyrosinase inhibitor from the Gram-negative bacterium Massilia albidiflava DSM 17472T

DCC3236 May1-in-13a

Novel potent inhibitor of May1 with Ki = 12 ± 1 nM, also inhibiting wild-type HIV-1 protease with Ki = 32 ± 5 pM and three drug resistance-associated mutants with Ki values ranging from 24 to 320 pM

DCC3237 Maysin

Natural Anti-inflammation Agent, Attenuating Amyloid Plaques by Inducing Humoral Immune Response with Th2 Skewed Cytokine Response in the Tg (APPswe, PS1dE9) Alzheimer's Mouse Model

70255-49-1
DCC3238 Mb-001

Novel potent inhibitor of the membrane-bound retinoid isomerase RPE65

DCC3239 Mb06322

Prodrug of MB05032, acting as potent and selective inhibitor of fructose 1,6-bisphosphatase for controlling gluconeogenesis in type 2 diabetes

280782-97-0
DCC3240 Mb16695

Novel Inhibitor of Mycobacterium tuberculosis α-1,4-Glucan Branching Enzyme (GlgB)

DCC3241 Mb-211

Novel inhibitor of dengue and West Nile virus NS2B-NS3 protease

DCC3242 Mbls-in-5

Novel non-hemolytic and low toxic inhibitor of metallo-β-lactamases (MBLs), restoring the activity of meropenem against Escherichia coli, Citrobacter freundii, Proteus mirabilis and Klebsiella pneumonia, which carried resistance genes of blaNDM-1

DCC3243 Mbp-c12

Novel detergent, showing enhanced stability to all tested proteins compared to a gold standard detergent (DDM)

DCC3244 Mbp-c9

Novel detergent, showing enhanced stability to all tested proteins compared to a gold standard detergent (DDM)

DCC3245 Mbri-001

Deuterium-substituted anticancer agent, plinabulin, exhibiting better pharmacokinetic characteristics than that of plinabulin

2054938-28-0
DCC3246 Mbt-fh Inhibitor-7

The first selective small molecule inhibitor of the Mycobacterium tuberculosis fumarate hydratase

DCC3247 Mbx-1066

Potent antibacterial agent against a wide range of Gram-positive and Gram-negative bacteria

868971-24-8
DCC3248 Mbx-1162

Novel antibacterial agent, remarkably potent against antibiotic-resistant bacterial strains such as MDR A. baumannii , ESBL-producing Klebsiella pneumoniae, VRE, and MRSA

1225332-95-5
DCC3249 Mbx-1887

Antibacterial agent, with a relatively narrow spectrum against bacteria and a very high CC 50 value

1429918-90-0
DCC3250 Mbx2546

Novel specific inhibitor of HA-mediated viral entry, inhibiting HPAI H5N1 virus strain A/Hong Kong/H5N1

695160-12-4
DCC3251 Mc1220

Topical nonnucleoside reverse transcriptase inhibitor, partially preventing vaginal RT-SHIV infection of macaques

391681-51-9
DCC3252 Mc-1353

Potent and HDAC class I-selective inhibitor

676599-90-9
DCC3253 Mc1420

Novel potent acetylcholinesterase (AChE) inhibitor

DCC3254 Mc-1-f2

The first inhibitor of forkhead Box Protein C2 (FOXC2)

2376894-10-7
DCC3255 Mc2050

Novel selective PARP1 inhibitor, inhibitng apoptosis and blocking poly ADP-ribosylation of histone H1 in hydrogen peroxide treated SH-SY5Y neuroblastoma cells

1301601-24-0
DCC3256 Mc2392

Novel hybrid retinoid-HDAC inhibitor

DCC3257 Mc-70 Hydrochloride

Potent P-gp inhibitor with good selectivity towards BCRP pump (EC50 values 0.05 μM, 0.69 μM, 9.3 μM, and 73 μM for Caco-2, MDR1, MRP1, and BCRP inhibition, respectively)

2108830-71-1
DCC3258 Mca-13

Novel neurotropic agent

DCC3259 Mca-yvadapk(dnp)-oh

Specific and highly fluorescent substrate for caspase-1, also acting as a substrate for caspase-4

DCC3260 Mcc1019

Novel selective inhibitor of the Polo-box domain of Polo-like kinase 1 (PLK1)

29115-34-2
DCC3261 Mcc1189

First-in-class inhibitor of MFS efflux pump CaMdr1p

1257542-38-3
DCC3262 Mcc-134

Novel inverse agonist for the pancreatic-type ATP-sensitive K channel as vascular relaxing agent

181238-67-5
DCC3263 MCC950 free acid Featured

Potent and selective inhibitor of NLRP3, reducing interleukin-1β (IL-1β) production in vivo and attenuating the severity of experimental autoimmune encephalomyelitis (EAE)

210826-40-7
DCC3264 Mc-doxhzn

Albumin-binding prodrug of Doxorubicin

151038-96-9
DCC3265 Mcg315

Novel potent F508del-CFTR corrector, modulating poly-ADP ribose polymerase 3 and poly-ADP ribose polymerase 16 activities

DCC3266 Mci-225

Selective NA reuptake inhibitor with 5-HT3 receptor antagonism

135991-48-9
DCC3267 Mcl0527-3

Novel inhibitor of p53-MDM2 interaction

DCC3268 Mcl-1 Degrader C3

Novel potent and selective degrader of Mcl-1

2163793-38-0
DCC3269 Mcl-1 Inhibitor-11

Novel reversible covalent inhibitor for Mcl-1 with improved water solubility than Mcl-1 Inhibitor-5

2012563-34-5
DCC3270 Mcl-1 Inhibitor-39

Novel selective Mcl-1 inhibitor

690218-87-2
DCC3271 Mcl-1 Inhibitor-5

The first reversible covalent inhibitor for Mcl-1, a protein-protein interaction (PPI) target

DCC3272 Mcl1-in-1

Novel potent and selective inhibitor of the apoptosis regulating proteins Mcl-1

713492-66-1
DCC3273 Mcmmad Featured

Novel mc (maleimidocaproyl) linker plus MMAD (Monomethylauristatin D) to be used for prepare antibodies conjugates via cysteine-capped mechanism

1401963-15-2
DCC3274 Mct4-in-18n

Novel highly selective inhibitor of monocarboxylate transporter 4 (MCT4/SLC16A3), resulting in lactate efflux inhibition and reduction of cellular viability in MCT4 high expressing cells

DCC3275 Mcule-5948770040

Novel SARS-CoV-2 Main Protease (Mpro) inhibitor, binding to Subsites S1 and S2 (Kd=1.3 µM)

DCC3276 Md-222

First-in-class highly potent PROTAC degrader of MDM2

2136246-72-3
DCC3277 Md-39-am

Diuretic agent, impling an increase in the Na+ excretion and showing antihypertensive effect

72564-74-0
DCC3278 Mdc-1112

Novel valproic acid (VPA) derivative, as a potent STAT3 inhibitor

DCC3279 Mdcccl1636

Novel partial PPARgamma ligand, displaying partial agonist activity in biochemical and cell-based transactivation assays, and reversed insulin resistance

DCC3280 Mdctmp

Novel proteolysis-resistant self-localizing ligand (SL), sustaining PM localization of eDHFR-fusion proteins (over several hours to a day), inducing prolonged signal activation and cell differentiation

DCC3281 Mde 6-82-1c

Novel MC5R antagonist

DCC3282 Mde10-136rs

Novel potent and highly selective melanocortin-3 receptor (MC3R) agonist, showing greater than 140-fold selective for the mMC3R over the mMC4R, possessed 70 nM potency at the mMC3R, and partially stimulated the mMC4R at 100 μM concentrations without antag

DCC3283 Mde6-5-2c

Novel potent and nonselective MC3R and MC4R macrocyclic agonist. decreased food intake and respiratory exchange ratio (RER)

DCC3284 Mdg486

Novel Inhibitor of BAF, activating latent HIV-1

92071-89-1
DCC3285 mdg559

Novel peroxisome proliferator activated receptor

512825-01-3
DCC3286 mdg582

Novel peroxisome proliferator activated receptor γ (PPARγ) ligand

459197-34-3
DCC3287 Mdl100240

Dual inhibitor of angiotensin-converting enzyme and neutral endopeptidase

142695-08-7
DCC3288 Mdm2/x Pdi

Potent Peptide dual inhibitor of MDM2/X, inhibiting p53 interactions with MDM2 (IC50 = 10 nmol/L) and MDMX (IC50 = 100 nmol/L), inducing apoptosis and cell cycle arrest of cell lines with overexpressed MDM2/X

DCC3289 Mdm2/xiap-in-14

Novel potent dual MDM2/XIAP inhibitor

DCC3290 Mdm2-p53-in-1b

Novel inhibitor of the MDM2-p53 interaction

856435-40-0
DCC3291 Mdmb-chminaca

Potent ligand of the central CB1 receptor

1185888-32-7
DCC3292 Me1111

Novel selective inhibitor of succinate dehydrogenase (complex II) of dermatophyte species

1391758-52-3
DCC3293 me6tren Tetrahydrochloride

Potent and efficacious mobilizing agent of hematopoietic stem and progenitor cells (HSPCs), activating MMP-9 expression and disrupting the SDF-1α/CXCR4 axis, exhibiting more significant mobilizing effects than G-CSF or AMD3100

859322-03-5
DCC3294 Mebeverine Hydrochloride Featured

Second generation papaverine analog, acting as an anticholinergic agent

2753-45-9
DCC3295 Mebhydrolin

Selective FXR antagonist, ameliorates glucose homeostasis in type 2 diabetic mice

524-81-2
DCC3296 Medermycin

Polyketide antibiotic, acting as a AKT selective kinase inhibitor, alkylating a regulatory loop cysteine

60227-09-0
DCC3297 Medrogestone

Progestational hormone, for the treatment of menstrual irregularities, prostatic hypertrophy, and endometrial carcinoma

977-79-7
DCC3298 Me-indoxam

Potent sPLA2 inhibitor, having no effect on arachidonic acid release and platelet activating factor synthesis

172732-62-6
DCC3299 mel_s3

Inducer of Megakaryocyte Differentiation in Erythroleukemia Cells, Impairing Bcr-Abl Signaling Cascades

1505462-80-5
DCC3300 Melafolone

Natural dual inhibitor of COX-2 and EGFR, improving program death 1 (PD-1) checkpoint blockade therapy through normalizing tumor vasculature and PD-L1 downregulation

129724-42-1
DCC3301 Melarsoprol

Prodrug of melarsen oxide (Mel Ox), irreversibly binding to vicinal sulfhydryl groups on pyruvate kinase, disrupting energy production in the parasite

494-79-1
DCC3302 Melinamide

Inhibitor of cholesterol esterification

14417-88-0
DCC3303 Melk-in-c1

Novel Multi-Kinase Inhibitor, Triggering Mitotic Catastrophe of Glioma Stem Cells Mainly through MELK Kinase Inhibition

DCC3304 Melogliptin

Potent, selective and orally bioavailable inhibitor of dipeptidyl peptidase 4 (DPP-4)

868771-57-7
DCC3305 Melperone Hydrochloride

5-HT2A/D2 receptor antagonist

1622-79-3
DCC3306 Men16132

Novel potent and selective nonpeptide kinin B2 receptor antagonist

1157852-02-2
DCC3307 meridianin A

Novel Cell Death-Inducing Kinase Inhibitor with Enhanced Selectivity for Cyclin-Dependent Kinases; Antimalarial

213472-98-1
DCC3308 Meriolin 3

Potent cell-permeable, ATP site-targeting inhibitor of CDKs

954143-48-7
DCC3309 Meriolin 5

Potent cell-permeable, ATP site-targeting inhibitor of CDKs

1011711-76-4
DCC3310 Merodantoin

Apoptosis inducer, triggering ROS dependent autophagy-associated apoptosis in a variety of human cancer cell lines and against mutant KRAS expressing cancer cells involving AKT-dependent ROS production

143413-73-4
DCC3311 Meso-dihydroguaiaretic Acid

LXR-α antagonist, inhibiting hepatic lipid accumulation by activating AMP-activated protein kinase in human HepG2 cells

36469-60-0
DCC3312 Mesterolone

Anabolic and androgenic agent

1424-00-6
DCC3313 Mesyl Salvinorin B

Novel selective and potent full KOP receptor agonist with fewer side effects (e.g., sedation or anhedonia) than classic KOP receptor

862073-79-8
DCC3314 Metabolex-36

Novel selective GPR120 agonist

1224102-50-4
DCC3315 Metamizole

Cyclooxygenase 3 (COX3) inhibitor, acting as a potent inductor of cytochrome P450 isoenzymes CYP2B6 and CYP3A4

50567-35-6
DCC3316 Methocinnamox

Potent, long-lasting, and selective antagonist of morphine-mediated antinociception

117332-69-1
DCC3317 Methoxybrassinin

Natural potent anti-proliferative agent, inducing apoptotic cell death

105748-60-5
DCC3318 Methoxyluteolin

Inhibitor of pro-inflammatory mediator release from mast cells

855-97-0
DCC3319 Methyl 6-bromo-1h-indazole-4-carboxylate

Useful pharmaceutical building block

885518-49-0
DCC3320 Methyl Meso-(meta-pyridinium) Bodipy

Novel photosensitizer as a photodynamic antimicrobial agent against Staphylococcus aureus, Escherichia coli, Candida albicans, and Methicillin-resistant S. aureus (MRSA)

DCC3321 Methyl Streptonigrin

Novel inhibitor of ABCG2 transporter function

3398-48-9
DCC3322 Methylaervine Featured

Natural antifungal agent, significantly inducing lipid peroxidation, activating the antioxidant enzymes, and exhibiting effective activity against F. solani (EC50 = 10.56 µM)

86293-40-5
DCC3323 Methylene Quinuclidinone

Metablite of PRIMA-1 and APR-246, covalently binding to cysteine residues in mutant p53 and wild type p53, and being increased in unfolded p53, inducing massive apoptosis in p53 null tumor cells

5291-26-9
DCC3324 Methylhonokiol

Novel Class of Cannabinoid CB2 Receptor Inverse Agonist

68592-15-4
DCC3325 Methylnaltrexone Iodide

Peripherally restricted μ-opioid antagonist

1360001-83-7
DCC3326 Met-in-3s

Highly Selective Class II MET Inhibitor

DCC3327 Metoclopramide Hydrochloride

Dopamine D2 antagonist, antiemetic

7232-21-5
DCC3328 Metocurine

Non-depolarizing muscle relaxant

5152-30-7
DCC3329 Metrizoate Calcium

Radiographic Contrast Agent

20828-80-2
DCC3330 Mfn103

Novel Dual Fluorescent and Magnetic Resonance False Neurotransmitter

DCC3331 Mg2-1812

Novel potent negative allosteric modulator (NAM) of mGlu2

DCC3332 Mg-277

Novel potent inhibitor of the p53-MDM2 interaction with an IC50 value of 67.5 nmol/L, against acute leukemia cell lines with different p53 status and was much less effective in inducing MDM2 degradation

2411085-89-5
DC3333 mG2N001 Featured

mG2N001 is a potent negative allosteric modulator (NAM) of metabotropic glutamate receptor 2 (mGluR2) with IC50 of 93 nM.

DCC3334 Mgcd516

Novel, multi-targeted kinase inhibitor, demonstrating potent inhibition of Trk, RET and DDR, in addition to Met, Axl and VEGFRs

1123837-88-6
DCC3335 Mgs-0028

Selective metabotropic glutamate 2/3 receptor agonist

260353-67-1
DCC3336 Mgs-0039

Potent and orally active group II mGluR antagonist with antidepressant-like potential

569686-87-9
DCC3337 Mhi-148

Near-infrared cyanine dye, acting as an optical imaging agent

DCC3338 Mhi-i2

Novel photodynamic antitumor agent

DCC3339 mhy1556

Novel tyrosinase inhibitor, showing concentration-dependent inhibitory effects with no significant cytotoxicity in cell viability assay

1446352-58-4
DCC3340 mhy218

Novel potent HDAC inhibitor, possessing potent anticancer activities

1326750-59-7
DCC3341 Mhy219

Novel potent histone deacetylase (HDAC) inhibitor, inducing apoptosis via up-regulation of androgen receptor expression in human prostate cancer cells

1326750-61-1
DCC3342 mhy336

Novel topoisomerase II inhibitor, markedly inducing apoptotic cell death via the mitochondria-mediated intrinsic pathway in LNCaP cells

84858-42-4
DCC3343 mhy384

Novel tyrosinase inhibitor, down-regulating of MITF and tyrosinase through direct tyrosinase inhibition

1367664-23-0
DCC3344 mhy407

Novel sensitizer of cancer cells, significantly increasing DNA damage as determined by DNA breakage, levels of damage-responsive proteins, and DNA foci

1453811-70-5
DCC3345 Mhy-449

Novel inducer of G2/M phase arrest in the cell cycle progression, resulting in growth inhibition and induction of apoptosis in a concentration-dependent manner, and inhibition of proliferation in a time-dependent manner

DCC3346 mhy498

Novel inhibitor of nitric oxide-induced melanogenesis, targeting the NO-induced cGMP signaling pathway

1208535-06-1
DCC3347 mhy-794

Novel tyrosinase inhibitor, directly inhibiting mushroom tyrosinase

1393371-29-3
DCC3348 Mhy884

Novel tyrosinase inhibitor, suppressing UVB-induced activation of NF-κB signaling pathway through the downregulation of oxidative stress

1393371-35-1
DCC3349 Mi-1061

Novel Chemically Stable, Potent, and Efficacious MDM2 Inhibitor

1410737-34-6
DCC3350 Mi-1900

Novel inhibitor of TMPRSS2, also strongly preventing SARS-CoV-2 multiplication and CPE in Calu-3 cells in a dose-dependent manner. causing strong inhibition of SARS-CoV-2 replication

DCC3351 Mi-319

Novel MDM2 antagonist, restoring p53 functions and increases the life span of orally treated follicular lymphoma bearing animals

DCC3352 Mi-432

Novel matriptase-1/matriptase-2 (MT-1/2) inhibitor, also inhibiting TMPRSS2, proteolytic activation and multiplication of influenza A virus in Calu-3 cells

DCC3353 mi-888 Tfa Salt

Highly Potent and Efficacious MDM2 Inhibitor

1303609-30-4
DCC3354 Microtubule Inhibitor 185322

Novel inhibitor of microtubule assembly, inducung mitotic arrest and apoptosis of MM cells

1027308-36-6
DCC3355 Mif Degrader Md13

Novel Potent MIF Degrader

DCC3356 Mifamurtide

Immunomodulator, regulating the activation of monocytes and macrophages, upregulating the secretion of pro-inflammatory cytokines such as TNF-alpha, IL-1, IL-8, nitric oxide and prostaglandins E2 and D2

83461-56-7
DCC3357 Mig-7 Inhibitor D-39

Novel inhibitor of Migration-Inducting Gene 7 (MIG-7) expression, suppressing EOC cell growth and VEGFA expression

DCC3358 Miglustat

Product Description:

72599-27-0
DCC3359 Milacemide Hydrochloride

MAO-B inhibitor and glycine prodrug, being studied for treatment for the symptoms of Alzheimer's disease

76990-85-7
DCC3360 Miliusol

Natural anti-tumor agent, demonstrating with tumor inhibitory efficacy comparable or even superior to the mainstay chemotherapeutics paclitaxel or fluorouracil

663892-51-1
DCC3361 Mina53-in-10

First-in-class inhibitor of MYC-induced nuclear antigen (MINA53) with selectivity over NO66 and other JmjC oxygenases

DCC3362 Minigastrin I (human)

Inhibitor of cholecystokinin B receptors (CCK2)

54405-27-5
DCC3363 Mip-1072

Novel inhibitor of the prostate-specific membrane antigen (PSMA)

949575-20-6
DCC3364 Mip-1095

Novel inhibitor of the prostate-specific membrane antigen (PSMA)

949575-22-8
DCC3365 Mipe-1686

Novel long-lasting myostatin inhibitor, significantly increasing muscle mass and hindlimb grip strength in Duchenne muscular dystrophic model mice

DCC3366 Mips1455

Novel photoactivatable allosteric ligand for the M1 muscarinic acetylcholine receptor

1627580-82-8
DCC3367 Mips1780

Novel selective positive allosteric modulator (PAM) at the M1 muscarinic acetylcholine receptor

DCC3368 Mipsagargin

Novel thapsigargin-based PSMA-activated prodrug, inhibiting the sarcoplasmic/endoplasmic reticulum calcium adenosine triphosphatase (SERCA) pump protein

1245732-48-2
DCC3369 Mir-21 Inhibitor

Novel specific and efficient inhibitor of miR-21 expression, inducing a 485% increase in the luciferase reporter signal at 10 μM

DCC3370 Mir-21 Inhibitor-1

Novel inhibitor of microRNA-21 (miR-21)

304880-74-8
DCC3371 Miro1 Reducer

Novel Miro1 degrader, rescuing dopaminergic neurodegeneration and promoting Miro1 degradation in Parkinson’s Disease fibroblasts

DCC3372 Miro1 Reducer 3

Novel degrader of Miro1 (mitochondrial Rho GTPase 1), reducing Miro1 levels in fibroblasts and stress-induced degeneration of dopaminergic neurons derived from Parkinson's disease (PD) patients, as well as age-dependent neuronal loss and prolongs lifespan

DCC3373 miroistonil

Novel inhibitor of AMA1-RON2 interaction, blocking merozoite invasion from schizont-infected RBCs; Antidepressant; Acetylcholinesterase inhibitor

33299-81-9
DCC3374 mitf-in-17

The first small molecule inhibitor of Mitf-E-box DNA binding with depigmenting activity

313984-78-0
DCC3375 Mitobady

Sensitive and specific Raman probe for live cell imaging of mitochondria

1644119-76-5
DCC3376 Mitodpp-2

Fluorescent probe for measuring the activity levels of erasers of S-palmitoylation, acyl-protein thioesterases (APTs), within mitochondria of live cells

DCC3377 Mitoebselen-2

Radiation Mitigator, reducing lipid hydroperoxides and preventing apoptotic cell death

DCC3378 Mitofp

Novel mitochondrial-targeted pan-APT inhibitor

DCC3379 Mito-peg5-ato

Novel potent antiproliferative mitochondria-targeted OXPHOS inhibitor (IC50=38 nM) in MiaPaCa-2 cells, being more effective than other inhibitors of OXPHOS in MiaPaCa-2 and U87MG cells

DCC3380 mitopy1

Novel selective fluorescent H2O2 probe, tracking the mitochondria of live biological specimens and responds to local fluxes of hydrogen peroxide (H2O2) by a turn-on fluorescence enhancement

1041634-69-8
DCC3381 Mitozolomide

Antineoplastic DNA alkylating agent

85622-95-3
DCC3382 Mizoribine Mono-phosphate

Specific inhibitor of the cellular inosine-5-monophosphate dehydrogenase (IMPDH); Immunosuppressive agent

62025-48-3
DCC3383 Mk0359

Potent and selective PDE4 inhibitor

346629-30-9
DCC3384 Mk-0493

Novel potent, orally active and selective agonist of the melanocortin receptor 4 (MC4R)

455956-93-1
DCC3385 mk-0499

The class III antiarrhythmic agent, blocking HERG, a human cardiac delayed rectifier K+ channel

156619-48-6
DCC3386 Mk-0626

Novel Dipeptidyl peptidase IV (DPP-4) inhibitor, improving neovascularization by increasing both the number of circulating endothelial progenitor cells and endothelial nitric oxide synthetase expression

DCC3387 Mk-0633 Tosylate

Potent and Selective 5-Lipoxygenase Inhibitor

1137737-87-1
DCC3388 Mk-0736

Selective 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor

719272-79-4
DCC3389 Mk-0916

Selective 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) inhibitor

633317-53-0
DCC3390 Mk-1220

Novel Macrocyclic Inhibitor of Hepatitis C Virus NS3/4A Protease with Improved Preclinical Plasma Exposure

924270-31-5
DCC3391 Mk-1597

Novel renin inhibitor

1007392-69-9
DCC3392 Mk-2295

Potent TRPV1 antagonist

878811-00-8
<Prev1...168169170171172...191Next>