DC9595 |
E-4031
Featured
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E-4031 is a benzenesulfonamide antiarrhythmic agent; blocks the ATP-sensitive potassium channel.
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DC9378 |
Efonidipine (hydrochloride monoethanolate)
Featured
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Efonidipine(NZ-105) Hcl monoethanolate is a dual T-type and L-type calcium channel blocker (CCB).
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DC8301 |
Elacridar
Featured
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Elacridar is an orally selectly potent P-glycoprotein (P-gp/ABCG1) inhibitor. |
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DC8268 |
Eliprodil
Featured
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Eliprodil is a non-competitive NMDA receptor antagonist that acts at the polyamine modulatory site. |
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DC8706 |
Emamectin Benzoate |
Emamectin Benzoate works as a chloride channel activator by binding gamma aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods. |
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DC4171 |
Escitalopram oxalate
Featured
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Escitalopram Oxalate is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM. |
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DC8821 |
Etifoxine Hydrochloride
Featured
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Etifoxine Hydrochloride is a psychotropic agent with anxiolytic and anticonvulsant activity. Etifoxine Hydrochloride is an activator of GABAA R β2 and GABAA R β3. |
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DC9893 |
Evans Blue |
Evans Blue is a potent inhibitor of the uptake of L-glutamate into synaptic vesicles, also an AMPA/kainate receptor antagonist |
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DC7987 |
Encenicline hydrochloride (EVP-6124)
Featured
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Encenicline hydrochloride (EVP-6124 hydrochloride) is a novel partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs). |
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DC10382 |
Farampator
Featured
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Farampator (CX-691;Org24448) is an AMPA receptor positive modulator. |
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DC11309 |
Fipronil |
Fipronil is an insecticide that acts as a selective antagonist of insect GABA receptors (IC50s = 30 and 1,600 nM for cockroach and rat receptors, respectively). |
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DC9623 |
Flecainide (acetate)
Featured
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Flecainide(Tambocor) is a class 1C antiarrhythmic drug especially used for the management of supraventricular arrhythmia; works by blocking the Nav1.5 sodium channel in the heart, causing prolongation of the cardiac action potential.
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DC9451 |
Flumazenil |
Flumazenil(Ro 15-1788) is a benzodiazepine antagonist, non-selective for α1, α2, α3 or α5-containing GABAA receptors. |
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DC9078 |
Fluoxetine Hydrochloride
Featured
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Fluoxetine HCl is an antidepressant of the selective serotonin reuptake inhibitor (SSRI) class. |
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DC4239 |
Flupirtine maleate |
Flupirtine maleateis a non-opioid, centrally acting analgesia, muscle relaxation and neuroprotection. Currently under a clinical trial (recruiting phase) as a treatment for Multiple Sclerosis and has been used as an analgesic. |
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DC10158 |
Fluralaner
Featured
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Fluralaner (INN) is a systemic insecticide and acaricide Fluralaner through potent blockage of GABA and L-glutamate gated chloride channels. |
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DC6917 |
Vonoprazan
Featured
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For the detailed information of Vonoprazan, the solubility of Vonoprazan in water, the solubility of Vonoprazan in DMSO, the solubility of Vonoprazan in PBS buffer, the animal experiment (test) of Vonoprazan, the cell expriment (test) of Vonoprazan, the in vivo, in vitro and clinical trial test of Vonoprazan, the EC50, IC50,and affinity,of Vonoprazan, For the detailed information of Vonoprazan, the solubility of Vonoprazan in water, the solubility of Vonoprazan in DMSO, the solubility of Vonoprazan in PBS buffer, the animal experiment (test) of Vonoprazan, the cell expriment (test) of Vonoprazan, the in vivo, in vitro and clinical trial test of Vonoprazan, the EC50, IC50,and affinity,of Vonoprazan, Please contact DC Chemicals.. |
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DC10947 |
FPL64176
Featured
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FPL64176 is a potent L-type Ca++ channel activator with EC50 of 16 nM. |
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DC9381 |
Gabapentin (hydrochloride) |
Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog. |
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DC8954 |
Gabapentin
Featured
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Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog. It was originally developed to treat epilepsy, and currently is also used to relieve neuropathic pain. |
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DC9859 |
GAL-021
Featured
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GAL-021 is a new intravenous BKCa-channel blocker. |
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DC7130 |
GBR 12935 dihydrochloride
Featured
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GBR 12935 is a potent and selective inhibitor of dopamine uptake (KD = 5.5 nM in rat striatal membranes). |
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DC10721 |
Gefapixant(AF-219,MK-7264)
Featured
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Gefapixant(AF-219,MK-7264) is novel P2X3 receptor antagonist. |
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DC10753 |
GLPG-1837(ABBV-974)
Featured
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GLPG-1837(ABBV-974) is a novel cystic fibrosis transmembrane conductance regulator CFTR potentiator. |
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DC11678 |
GLPG-2222 |
GLPG-2222 (ABBV-2222, Galicaftor) is a novel potent and efficacious CFTR corrector with EC50 of 5 nM. |
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DC11035 |
GlyT1 inhibitor 46 |
GlyT1 inhibitor 46 is a novel potent, selective, orally available inhibitor of glycine transporter-1 (GlyT1) with IC50 of 38 and 21 nM for rat and human GlyT1, respectively. |
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DC10874 |
GlyT2-IN-1(YODA 1)
Featured
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GlyT2-IN-1(YODA 1) is a glycine transporters GLYT2 inhibitor. |
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DC10907 |
GNE-131
Featured
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GNE-131 is a novel NaV1.7 inhibitor with IC50 0.003uM,improving metabolic stability,efficacy in mouse IEM model at C-plasma <2.8uM. |
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DC11090 |
GR3027
Featured
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GR3027 (Golexanolone) is a GABA-A receptor modulating steroid antagonist that selectively antagonizes the enhanced activation of GABAA receptors by neurosteroids such as allopregnanolone and THDOC. |
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DC8006 |
GS967(GS-458967)
Featured
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GS967 is a novel, potent, and selective inhibitor of cardiac late sodium current(late INa). |
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