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Cat. No. Product name CAS No.
DC22446 CE-224535

CE-224535 (PF-04905428) is a potent and selective P2X7 receptor antagonist with IC50 of 1.4 nM (inhibition of the release of lL-1b from monocytes stimulated by ATP).

724424-43-5
DC20881 CE-245677

CE-245677 is a potent, selective, orally active, dual Tie2/Trk kinase inhibitor with IC50 of 4.7 nM, 1 nM for Tie2 and TrkA/B, respectively.

717899-97-3
DC20336 CE3F4 Featured

CE3F4 is a potent, noncompetitive EPAC1 inhibitor that blocks EPAC1-induced Rap1 activation both in cell-free systems and in intact cells and did not influence protein kinase A holoenzyme activity.

143703-25-7
DC23912 Cecropin B

Cecropin B is an antimicrobial peptide with MICs(0.5 to 16 ug/ml) against Gramnegative strains.

80451-05-4
DC20987 Cedazuridine Featured

Cedazuridine (E7727) is a novel cytidine deaminase inhibitor, and a componet of ASTX727 for treatment of hematologic malignancies..

1141397-80-9
DC8686 Cefetamet pivoxil hydrochloride

Cefetamet pivoxil hydrochloride is an oral third generation cephalosporin antibiotic.

111696-23-2
DC9358 Cefmenoxime (hydrochloride)

Cefmenoxime hydrochloride is a third-generation cephalosporin antibiotic.

75738-58-8
DC20190 Cefoxitin

Cefoxitin is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.

35607-66-0
DC9356 Cefpiramide (sodium)

Cefpiramide sodium (SM-1652; Wy-44635) is a new Pseudomonas-active cephalosporin with a broad spectrum of antibacterial activity.

74849-93-7
DC8687 Cefpirome sulfate

Cefpirome Sulfate is a fourth generation cephalosporin antibiotic.

98753-19-6
DC9355 Ceftibuten (dihydrate)

Ceftibuten dihydrate is a third-generation cephalosporin antibiotic.

118081-34-8
DC12245 Ceftizoxime

Ceftizoxime is a bacterial inhibitor which acts by interfering with bacterial cell wall synthesis and inhibiting cross-linking of the peptidoglycan.

68401-81-0
DC7569 Z-LEHD-FMK

Cell permeable fluoromethyl ketone (FMK)-derivatized peptides act as effective irreversible Caspase inhibitors with no cytotoxic effects and, therefore, are useful tools for studying Caspase activity.

210345-04-3
DC7568 Z-DEVD-FMK Featured

Cell-permeable, irreversible inhibitor of caspase-3/CPP32; inhibits tumor cell apoptosis. Neuroprotective in rat hippocampus following seizures in vivo.

210344-95-9
DC23359 CeMMEC2

CeMMEC2 is a novel potent BRD4 inhibitor with IC50 of 0.9 uM, binds to both bromodomains of BRD4, comparably to (S)-JQ1..

902955-25-3
DC10357 Cenerimod

Cenerimod (ACT-334441) is a potent and orally available sphingosine 1-phosphate 1 receptor (S1P1) agonist extracted from patent WO 2016184939 A1 and WO 2011007324 A1, example 1, with an EC50 of 2.7 nM.

1262414-04-9
DC10316 Cenicriviroc Featured

Cenicriviroc is an orally active, dual CCR2/CCR5 antagonist, and displays potent anti-inflammatory and aninfective activity.

497223-25-3
DC21554 AS 703569

Cenisertib (AS 703569;R763) is a novel potent, orally available inhibitor of Aurora kinases, exhibits signifficant anti-proliferative activity against a wide range of tumor cells both in vitro and in vivo (A549 EC50=9 nM).

871357-89-0
DC12318 Centanafadine hydrochloride (EB-1020 (hydrochloride))

Centanafadine (hydrochloride) is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively.

923981-14-0
DC12319 Centanafadine (EB-1020)

Centanafadine is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively.

924012-43-1
DC10010 Centrinone Featured

Centrinone is a selective and reversible inhibitor of polo-like kinase 4 (Plk4), a serine-threonine protein kinase that initiates centriole/centrosome assembly.

1798871-30-3
DC22796 CEP-1347

CEP-1347 (KT-7515) is a potent and selective MLK inhibitor that completely rescues motoneurons and inhibits JNK1 activation with IC50 of 20 nM.

156177-65-0
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