PDE 3 inhibitor

Non-peptide angiotensin II receptor antagonist

Novel peptide endomorphin (EM) degradation blocker

Novel peptide endomorphin (EM) degradation blocker

Novel peptide endomorphin (EM) degradation blocker

Novel corticotropin-release factor 1 antagonist

5-FU derivative, with various anticancer agents against human cancer xenografts

Novel PRMT inhibitor, preventing arginine methylation of cellular proteins, being essentially inactive against the lysine methyltransferase SET7/9

Novel Potent and Selective Inhibitor of Protein Arginine Methyltransferase 4 (PRMT4)

Antioxidant, inhibiting free radical oxidation of biomembrane lipids, modulating the activity of membrane-bound enzymes and the receptor complexes of the brain membranes

Novel non-steroidal CYP17 inhibitor. reducing androgen synthesis for treatment of castration-resistant prostate cancer

Novel butyrylcholinesterase inhibitor against Alzheimer's disease

Novel Potentiator of α7 Receptor Signaling

Useful pharmceutical building block

Antimalarial

Natural vesicle trafficking inhibitor

Specific inhibitor of trafficking pathways, disrupting recycling at the PM via interference with ROP6/RIC1 signalling

Novel inhibitor of eukaryotic ARF-GEFs (ADP-ribosylation factor guanine nucleotide exchange factors)

Specific inhibitor for plant callose deposition during cytokinesis without affectting endomembrane trafficking during interphase or cytoskeletal organization

Novel modulator of the PIN1 accumulation, selectively modifying PIN1 basal plasma membrane targeting in Arabidopsis with minimal effects on apical plasma membrane proteins

Novel modulator of the PIN1 accumulation, selectively modifying PIN1 basal plasma membrane targeting in Arabidopsis with minimal effects on apical plasma membrane proteins

Sodium/hydrogen exchange inhibitor