DC9130 |
Azelastine HCl |
Azelastine HCl is a potent, second-generation, selective, histamine antagonist. |
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DC8338 |
Azeliragon(PF-04494700,TTP488)
Featured
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Azeliragon is an oral, small-molecule inhibitor of RAGE. |
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DCAPI1590 |
Azelnidipine |
Azelnidipine is an L-type calcium channel protein inhibitor |
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DC20156 |
Azetidine-2-carboxylic acid
Featured
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Azetidine-2-carboxylic acid is a non proteinogenic amino acid homologue of proline. Found in common beets. Azetidine-2-carboxylic acid can be misincorporated into proteins in place of proline in many species, including humans. Toxic and teratogenic agent. |
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DC4210 |
Azilsartan kamedoxomil
Featured
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Azilsartan medoxomil is an angiotensin II receptor antagonist indicated for the treatment of mild to moderate essential hypertension. |
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DCAPI1469 |
azilsartan
Featured
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Azilsartan(TAK-536) is a specific and potent angiotensin II type 1 receptor antagonist with IC50 of 2.6 nM. |
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DC9596 |
Azimilide (Dihydrochloride) |
Azimilide 2Hcl(NE-10064 2Hcl) is a class III antiarrhythmic compound, inhibits I(Ks) and I(Kr) in guinea-pig cardiac myocytes and I(Ks) (minK) channels expressed in Xenopus oocytes.
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DCAPI1362 |
Azithromycin (Zithromax) |
Azithromycin (Zithromax) |
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DC4141 |
Azocosterol 2HCL |
Azocosterol is a potential avian reproductive inhibitor. |
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DCAPI1225 |
Azomycin (2-Nitroimidazole) |
Azomycin (2-Nitroimidazole) |
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DC9818 |
Azoramide
Featured
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Azoramide is a small-molecule modulator of the unfolded protein response with antidiabetic activity. |
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DC10992 |
Azosemide |
Azosemide (Azosemidum) is a potent Na-K-Cl Cotransporter NKCC1 with IC50 of 0.246 and 0.197 uM for hNKCC1A and NKCC1B, being about 4-times more potent than bumetanide. |
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DC12497 |
(Z)-Azoxystrobin
Featured
|
Azoxystrobin is a systemic, broad-spectrum fungicide belonging to the class of methoxyacrylates,which are derived from the naturally-occurring strobilurins. |
|
DC22953 |
AZSMO-23 |
AZSMO-23 (AZSMO 23, AZSMO23) is a potent hERG potassium channel (Kv11.1) activator that activates WT hERG pre-pulse and tail current with EC50 of 28.6 and 11.2 μM respectively. |
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DCAPI1341 |
Aztreonam (Azactam, Cayston) |
Aztreonam (Azactam, Cayston) |
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DC21570 |
Azvudine
Featured
|
Azvudine (RO 0622) is a potent HCV NS5B RNA polymerase inhibitor, inhibits HCV replication in the replicon system with IC50 of 24 nM; inhibits RNA synthesis by HCV polymerases from either HCV genotypes 1a and 1b or containing S96T or S282T point mutations (IC50=10-100 nM). |
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DC23756 |
Aβ polymerization stimulator O4 |
Aβ polymerization stimulator O4 is an orcein-related small molecule can drive polymerization of amyloid-β (Aβ). |
|
DC12114 |
B I09 |
B I09 is an IRE-1 RNase inhibitor, with an IC50 of 1230 nM. |
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DC10026 |
B02
Featured
|
B02 is a cell-permeable pyridinylvinyl-quinazolinone compound that is shown to specifically inhibit human RAD51 (IC50 = 27.4 µM). |
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DC22010 |
B591 |
B591 (B-591) is a potent, specific pan-PI3K inhibitor with IC50 of 1.3/0.36/1.1/1.58 uM for PI3Kα/β/γ/δ, respectively. |
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DC12033 |
(S)-B-973B
Featured
|
B-973 (B973) is a potent, selective α7 nAChR ago-PAM, denonstrates analgesic effect with attenuating pain behavior and decreasing paw edema in vivo. |
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DC22011 |
BAA473 |
BAA473 (BAA-473) is a bile acid analogue that functions as the first small molecule activator of the Pyrin inflammasome, induces secretion of IL18 in LPS-primed PBMCs. |
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DC10859 |
Baccatin III
Featured
|
Baccatin III is the precursor to paclitaxel/ taxol. Antileukaemic and antitumor agent isolated from the bark of the Pacific yew tree (Taxus breviofolia). |
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DC20063 |
BACE1-IN-2 |
BACE1-IN-2 is a 1,4-Oxazine β-Secretase 1 (BACE1) inhibitor with an IC50 of 22 nM. |
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DCAPI1066 |
Bacitracin zinc |
Bacitracin zinc |
|
DC8971 |
Baclofen |
Baclofen is a gamma-amino-butyric acid (GABA) derivative used as a skeletal muscle relaxant. |
|
DC2013 |
Bafetinib (INNO-406)
Featured
|
Bafetinib (INNO-406) is a potent and selective dual Bcr-Abl/Lyn inhibitor with IC50 of 5.8 nM and 19 nM, respectively. |
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DC8858 |
Bafilomycin A1(Baf-A1)
Featured
|
Bafilomycin A1 is a vacuolar H+-ATPase inhibitor with IC50 of 0.44 nM. |
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DC20740 |
BAL30072 |
BAL30072 is a monocyclic beta-lactam antibiotic that shows potent activity against MDR Pseudomonas aeruginosa and Acinetobacter sp. Isolates with MIC90 of 8 and 4 ug/ml. |
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DC10994 |
Balamapimod |
Balamapimod (MKI-833) is an orally active, reversible Ras/Raf/MEK inhibitor developed for antineoplastic potential.. |
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