DC23856 |
CEP-7055 |
CEP-7055 is a potent, orally active, pan inhibitor of VEGFR, CEP-7055 is the dimethylglycine ester prodrug of CEP-5214, which inhibits human VEGFR2/KDR kinase, VEGFR1/FLT-1 kinase, and VEGFR3/FLT-4 kinase with IC50 of 18 nM, 12 nM, and 17 nM. |
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DC7347 |
Cephalosporin C Na salt
Featured
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Cephalosporin C Na salt is used to study the effect of transpeptidase expression, binding, and inhibition on bacterial cell wall mucopeptide synthesis. |
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DC7346 |
Cephalosporin C zinc salt
Featured
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Cephalosporin C zinc salt is used to study the effect of transpeptidase expression, binding, and inhibition on bacterial cell wall mucopeptide synthesis. |
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DC9649 |
Cephalotaxlen
Featured
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Cephalotaxine is an antiviral as well as antitumor agent. |
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DC10226 |
Cefradine |
Cephradine is a semi-synthetic cephalosporin antibiotic. |
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DC9765 |
CERC-501(LY-2456302,Aticaprant)
Featured
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CERC-501(LY-2456302) is a potent, selective antagonist of the kappa opioid receptor (KOR) (Ki = 0.81 nM vs. 24.0 nM and 155 nM for the μ-opioid receptor (MOR) and δ-opioid receptor (DOR), respectively. |
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DC7814 |
Cerdulatinib(PRT-062070; PRT2070)
Featured
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Cerdulatinib(PRT-062070; PRT2070) is an novel oral dual Syk/JAK inhibitor. |
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DC9154 |
Cetirizine 2HCl |
Cetirizine 2Hcl, a second-generation antihistamine, is a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria. |
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DC9500 |
Cevimeline (hydrochloride hemihydrate)
Featured
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Cevimeline hydrochloride hemihydrate, a novel muscarinic receptor agonist, is a candidate therapeutic drug for xerostomia in Sjogren's syndrome. |
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DC7899 |
Cevipabulin(TTI 237) |
Cevipabulin, also known as TTI-237, an antimicrotubule agent, is a small synthetic molecule of triazolopyrimidine derivative with potential antitumor activity. |
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DC10440 |
Namodenoson (CF-102)
Featured
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CF-102(2-Cl-IB-MECA) is a selective A3 adenosine receptor agonist (Ki = 0.33 nM). Displays 2500- and 1400-fold selectivity over A1 and A2A receptors respectively.
target: A3 adenosine receptor agonist; |
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DC22052 |
CFI02 |
CFI02 (CFI-02) is a specific inhibitor of human cytomegalovirus (HCMV) glycoprotein B-mediated fusion with IC50 of 40 nM against laboratory adapted HCMV strain AD169. |
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DC10069 |
CFI-400437
Featured
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CFI-400437 is potent against PLK4 (IC50 = 0.6 nM) and selective against other members of the PLK family (>10 uM). |
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DC23338 |
CFI-401980 |
CFI-401980 is a potent, selective, novel class TTK (Tyrosine Threonine Kinase) inhibitor with Ki of 0.8 nM, HCT116 GI50 of 13 nM. |
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DC9340 |
CFM-2 |
CFM-2 is a selective non-competitive AMPAR antagonist.
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DC11133 |
CFM-4.16 |
CFM-4.16 is a CARP-1 functional mimetic (CFM) compound bind with CARP-1, stimulates CARP-1 expression and apoptosis. |
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DC22809 |
c-FMS-IN-8
Featured
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c-FMS-IN-8 is a potent, selective c-FMS kinase inhibitor with IC50 of 0.8 nM, shows activity in collagen-induced model of arthritis in mice.. |
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DC7039 |
CFTR Inhibitor II
Featured
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CFTR Inhibitor II is a cell-permeable glycinyl hydrazone compound that acts as a potent, selective and reversible open-channel blocker of CFTR with intermediate speed (< 1 min; 95% inhibition at 50 µM; Ki = 4.3 µM in CFTR-expressing FRT cells. |
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DC12580 |
CG-806
Featured
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CG-806 (CG806, CG'806) is a novel potent, pan-FLT3/BTK multi-kinase inhibitor with impressive inhibition of leukemic cell proliferation with IC50 at sub-nanomolar or low nanomolar levels. |
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DC7380 |
CGI-1746
Featured
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CGI1746 is a small-molecule Btk inhibitor chemotype with a new binding mode that stabilizes an inactive nonphosphorylated enzyme conformation. |
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DC7101 |
CGK733
Featured
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CGK 733 is a potent and selective inhibitor of ATM/ATR with IC50 of ~200 nM. |
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DC10843 |
CGP 52432
Featured
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CGP 52432 is a potent, selective GABAB receptor antagonist (IC50 = 85 nM). |
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DC7381 |
CGP-57380
Featured
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CGP 57380 is a cell-permeable pyrazolo-pyrimidine compound that acts as a selective inhibitor of Mnk1 (IC50 = 2.2 μM) with no inhibitory activity against p38, JNK1, ERK1/2, PKC, or Src-like kinases. |
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DC10722 |
CGP-71683A
Featured
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CGP 71683A is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity. |
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DC9849 |
CGP37849 |
CGP37849 is a potent, selective and competitive NMDA receptor antagonist (Ki = 35 nM). Anticonvulsive following oral administration in vivo. |
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DC23919 |
CGP-42112
Featured
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CGP-42112 (CGP42112A) is a highly potent, selective Angiotensin-II subtype 2 receptor(AT2 receptor) agonist with Ki of 0.24 nM. |
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DC23830 |
CGP-53353 |
CGP-53353 (DAPH-7) is a selective inhibitor of PKCβII with IC50 of 0.41 uM, shows weak activity on PKCβI with IC50 of 3.8 uM. |
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DC20887 |
CGP-74514A hydrochloride |
CGP-74514A hydrochloride is a potent CDK1 inhibitor with IC50 of 25 nM. |
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DC8471 |
CGS 21680 hydrochloride
Featured
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CGS 21680 hydrochloride is an A2A adenosine receptor agonist (Ki = 27 nM). |
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DC24112 |
CGS 21680 |
CGS 21680 is a specific adenosine A2A subtype receptor agonist with Ki of 27 nM. |
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