(R)-ZINC-3573 |CAS 2089389-15-9|DC Chemicals

Cas No.:	2089389-15-9
Chemical Name:	(R)-Zinc-3573
Synonyms:	(R)-Dimethyl-[1-(5-phenyl-pyrazolo[1,5-a]pyrimidin-7-yl)-pyrrolidin-3-yl]-amine;GTPL9566;J3.638.819F;(3R)-N,N-Dimethyl-1-(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)-3-pyrrolidinamine;(3R)-N,N-dimethyl-1-(5-phenylpyrazolo[1,5-a]pyrimidin-7-yl)pyrrolidin-3-amine;(R)-Zinc-3573;ZINC-3573
SMILES:	N1(C2=CC(C3C=CC=CC=3)=NC3=CC=NN23)CC[C@H](C1)N(C)C
Formula:	C₁₈H₂₁N₅
M.Wt:	307.392843008041
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

(R)-ZINC-3573 is a potent, selective agonist of the atypical opioid receptor MRGPRX2 (EC50=0.76 uM), showing little activity against 315 other GPCRs and 97 representative kinases; activates endogenous MRGPRX2 in a human mast cell line, inducing degranulation and calcium release.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

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