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PF-06928215

  Cat. No.:  DC21478   Featured
Chemical Structure
2378173-15-8
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More than 5000 active chemicals with high quality for research!
Field of application
PF-06928215 (PF06928215) is a high affinity Cyclic GMP-AMP synthase (cGAS) inhibitor with Kd of 200 nM, IC50 of 4.9 uM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2378173-15-8
Chemical Name: PF-06928215
Synonyms: (1R,2S)-2-{[(7-Hydroxy-5-phenylpyrazolo[1,5-a]pyrimidin-3-yl)carbonyl]amino}cyclohexanecarboxylic ac;PF-06928215;CID 137300622;(1R,2S)-2-[(7-oxo-5-phenyl-1H-pyrazolo[1,5-a]pyrimidine-3-carbonyl)amino]cyclohexane-1-carboxylic acid;(1R,2S)-2-[[(7-hydroxy-5-phenylpyrazolo[1,5-a]pyrimidin-3-yl)carbonyl]amino]-cyclohexanecarboxylic acid;(1R,2S)-2-[(7-hydroxy-5-phenylpyrazolo[1,5-a]pyrimidine-3-carbonyl)amino]cyclohexane-1-carboxylic acid;GTPL11324;BDBM50250108;(1R,2S)-2-(7-Hydroxy-5-phenylpyrazolo[1,5-a]pyrimidine-3-carboxamido)cyclohexanecarboxylic ac
SMILES: O([H])C([C@]1([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])[C@]1([H])N([H])C(C1=C([H])N([H])N2C(C([H])=C(C3C([H])=C([H])C([H])=C([H])C=3[H])N=C21)=O)=O)=O
Formula: C20H20N4O4
M.Wt: 380.3972
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: PF-06928215 (PF06928215) is a high affinity Cyclic GMP-AMP synthase (cGAS) inhibitor with Kd of 200 nM, IC50 of 4.9 uM.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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