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SCH 529074

  Cat. No.:  DC23318   Featured
Chemical Structure
922150-11-6
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More than 5000 active chemicals with high quality for research!
Field of application
SCH 529074 is a small molecule mutant p53 reactivator that binds p53 DNA binding domain with Kd of 1-2 uM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 922150-11-6
Chemical Name: SCH529074
Synonyms: SCH 529074;N1-(2-((4-(bis(4-chlorophenyl)methyl)piperazin-1-yl)methyl)quinazolin-4-yl)-N3,N3-dimethylpropane-1,3-diamine;N3-[2-[[4-[Bis(4-chlorophenyl)methyl]-1-piperazinyl]methyl]-4-quinazolinyl]-N1,N1-dimethyl-1,3-propanediamine (ACI);Sch 529074;SCH529074
SMILES: ClC1C=CC(C(N2CCN(CC3N=C(NCCCN(C)C)C4C(=CC=CC=4)N=3)CC2)C2C=CC(Cl)=CC=2)=CC=1
Formula: C31H36Cl2N6
M.Wt: 563.563744544983
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: SCH 529074 is a small molecule mutant p53 reactivator that binds p53 DNA binding domain with Kd of 1-2 uM; restores growth-suppressive function to mutant p53 and inhibits ubiquitination of p53 by HDM2.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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